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GT201300267A - Isoxazolinas como agentes terapéuticos - Google Patents

Isoxazolinas como agentes terapéuticos

Info

Publication number
GT201300267A
GT201300267A GT201300267A GT201300267A GT201300267A GT 201300267 A GT201300267 A GT 201300267A GT 201300267 A GT201300267 A GT 201300267A GT 201300267 A GT201300267 A GT 201300267A GT 201300267 A GT201300267 A GT 201300267A
Authority
GT
Guatemala
Prior art keywords
therapeutic agents
isoxazolins
metaloproteinasa
matríz
isoxazolinas
Prior art date
Application number
GT201300267A
Other languages
English (en)
Inventor
David J Calderwood
Eric C Breinlinger
Steven L Swann
Subhendu Mukherjee
Venkata Srikanth Chitty
Siva Sanjeeva Rao Thunuguntla
Subramanyah Seetharama Shastry Hosahalli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47108012&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT201300267(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT201300267A publication Critical patent/GT201300267A/es

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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
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    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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Abstract

LA PRESENTE INVENCIÓN SE REFIERE A ISOXAZOLINAS COMO AGENTES TERAPÉUTICOS LOS CUALES SE CONSTITUYEN COMO INHIBIDORES SELECTIVOS DE METALOPROTEINASA DE MATRÍZ, MMP-13, Y DE LAS CUALES SE HA INFORMADO QUE MEDIAN EN LA DEGRADACIÓN DEL TEJIDO CONECTIVO EN PROCESOS FISIOLÓGICOS NORMALES
GT201300267A 2011-04-30 2013-10-30 Isoxazolinas como agentes terapéuticos GT201300267A (es)

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DOP2013000251A (es) 2014-02-28
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