GT200900082A - Composiciones de fenilalquilamino-carbamato - Google Patents
Composiciones de fenilalquilamino-carbamatoInfo
- Publication number
- GT200900082A GT200900082A GT200900082A GT200900082A GT200900082A GT 200900082 A GT200900082 A GT 200900082A GT 200900082 A GT200900082 A GT 200900082A GT 200900082 A GT200900082 A GT 200900082A GT 200900082 A GT200900082 A GT 200900082A
- Authority
- GT
- Guatemala
- Prior art keywords
- phenylalquilamine
- carbamate
- carbamate compositions
- compositions
- alkylamin
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- KXDHJXZQYSOELW-UHFFFAOYSA-M Carbamate Chemical compound NC([O-])=O KXDHJXZQYSOELW-UHFFFAOYSA-M 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Inorganic Chemistry (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Psychology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
LA PRESENTE INVENCION ESTA DIRIGIDA A UNA COMPOSICION CONTENIENDO FENILALQUILAMINO-CARBAMATO QUE TIENE UNA ESTABILIDAD MEJORADA Y MAS PARTICULARMENTE, LAS COMPOSICIONES COMPRENDEN EL COMPUESTO ANTES MENCIONADO EN UNA MEZCLA CON FOSFATO DIBASICO DE CALCIO DIHIDRATADO, QUE TIENEN UNA ESTABILIDAD MEJORADA SIENDO DE UTILIDAD EN TRASTORNOS DEL SISTEMA NERVIOSO CENTRAL (SNC).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82934206P | 2006-10-13 | 2006-10-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200900082A true GT200900082A (es) | 2010-02-24 |
Family
ID=39111348
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200900082A GT200900082A (es) | 2006-10-13 | 2009-04-13 | Composiciones de fenilalquilamino-carbamato |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20080090902A1 (es) |
| EP (1) | EP2079449A2 (es) |
| JP (1) | JP2010506845A (es) |
| KR (1) | KR20090082213A (es) |
| CN (1) | CN101557804A (es) |
| AU (1) | AU2007313017A1 (es) |
| BR (1) | BRPI0719275A2 (es) |
| CA (1) | CA2673487A1 (es) |
| CO (1) | CO6180500A2 (es) |
| CR (1) | CR10794A (es) |
| EA (1) | EA200970377A1 (es) |
| GT (1) | GT200900082A (es) |
| IL (1) | IL198145A0 (es) |
| MX (1) | MX2009003926A (es) |
| NI (1) | NI200900053A (es) |
| NO (1) | NO20091530L (es) |
| SV (1) | SV2009003221A (es) |
| WO (1) | WO2008048801A2 (es) |
| ZA (1) | ZA200903283B (es) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI419681B (zh) | 2005-06-08 | 2013-12-21 | Sk生物製藥股份有限公司 | 胺基甲酸酯用於製造供治療白天過度嗜睡(eds)的藥物之用途 |
| JP6095366B2 (ja) | 2009-06-22 | 2017-03-15 | エスケー バイオファーマシューティカルズ カンパニー リミテッド | 疲労を治療又は予防するための方法 |
| EP2496227B1 (en) | 2009-11-06 | 2019-05-22 | SK Biopharmaceuticals Co., Ltd. | Methods for treating fibromyalgia syndrome |
| CN102762201B (zh) | 2009-11-06 | 2013-12-18 | 爱思开生物制药株式会社 | 注意力缺陷/多动症的治疗方法 |
| US8623913B2 (en) * | 2010-06-30 | 2014-01-07 | Sk Biopharmaceuticals Co., Ltd. | Methods for treating restless legs syndrome |
| US9610274B2 (en) | 2010-06-30 | 2017-04-04 | Sk Biopharmaceuticals Co., Ltd. | Methods for treating bipolar disorder |
| CN105228604A (zh) | 2013-03-12 | 2016-01-06 | 比皮艾思药物研发有限公司 | 用于预防或治疗小儿癫痫和癫痫相关综合征的苯基氨基甲酸酯化合物 |
| KR20160004260A (ko) | 2013-03-12 | 2016-01-12 | (주)바이오팜솔루션즈 | 페닐카바메이트 화합물 및 이를 포함하는 신경보호용 조성물 |
| PT2968208T (pt) | 2013-03-13 | 2022-10-28 | Aerial Biopharma Llc | Tratamento da cataplexia |
| EP3021838B1 (en) | 2013-07-18 | 2020-05-27 | Jazz Pharmaceuticals Ireland Limited | Treatment for obesity |
| US10195151B2 (en) | 2016-09-06 | 2019-02-05 | Jazz Pharmaceuticals International Iii Limited | Formulations of (R)-2-amino-3-phenylpropyl carbamate |
| EP3630072A4 (en) | 2017-06-02 | 2021-03-10 | Jazz Pharmaceuticals Ireland Limited | METHODS AND COMPOSITIONS FOR TREATMENT OF EXCESSIVE Drowsiness |
| CN110037995B (zh) * | 2019-04-17 | 2021-07-06 | 石家庄龙泽制药股份有限公司 | 一种稳定的盐酸帕罗西汀片剂及其制备方法 |
| US10940133B1 (en) | 2020-03-19 | 2021-03-09 | Jazz Pharmaceuticals Ireland Limited | Methods of providing solriamfetol therapy to subjects with impaired renal function |
| IT202000013855A1 (it) | 2020-06-10 | 2021-12-10 | Flamma Spa | Un processo per la purificazione del (r)-2-ammino-3-fenilpropil carbammato |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3342687A (en) * | 1964-06-25 | 1967-09-19 | Colgate Palmolive Co | Oral preparation |
| US3420817A (en) * | 1966-12-06 | 1969-01-07 | Hoffmann La Roche | 4,1,5-benzoxadiazocin-2-ons and processes for preparing same |
| US6043211A (en) * | 1988-02-02 | 2000-03-28 | The Regents Of The University Of California | Method for inhibiting the activity of a platelet-derived growth factor receptor binding protein |
| KR100197892B1 (ko) * | 1994-09-09 | 1999-06-15 | 남창우 | 신규한 페닐알킬아미노 카바메이트 화합물과 그의 제조방법 |
| KR0173862B1 (ko) * | 1995-02-11 | 1999-04-01 | 조규향 | O-카바모일-(d)-페닐알라닌올 화합물과 그의 약제학적으로 유용한 염 및 이들의 제조방법 |
| US5756817C1 (en) * | 1995-02-11 | 2001-04-17 | Sk Corp | O-carbamoyl-phenylananinol compounds their pharmaceutically useful salts and process for preparing the same |
| KR0173863B1 (ko) * | 1995-04-10 | 1999-04-01 | 조규향 | 페닐에 치환체가 있는 o-카바모일-페닐알라닌올 화합물과 그의 약제학적으로 유용한 염 및 이들의 제조방법 |
| EP0873308B1 (en) * | 1996-10-10 | 2002-01-02 | SK Corporation | O-carbamoyl-phenylalaninol compounds and their pharmaceutically useful salts |
| US20020151543A1 (en) * | 1998-05-28 | 2002-10-17 | Sepracor Inc. | Compositions and methods employing R (-) fluoxetine and other active ingredients |
| WO2002017921A2 (en) * | 2000-08-28 | 2002-03-07 | Synthon B.V. | Paroxetine compositions and processes for making the same |
-
2007
- 2007-10-08 US US11/868,555 patent/US20080090902A1/en not_active Abandoned
- 2007-10-08 MX MX2009003926A patent/MX2009003926A/es not_active Application Discontinuation
- 2007-10-08 WO PCT/US2007/080675 patent/WO2008048801A2/en not_active Ceased
- 2007-10-08 EA EA200970377A patent/EA200970377A1/ru unknown
- 2007-10-08 AU AU2007313017A patent/AU2007313017A1/en not_active Abandoned
- 2007-10-08 KR KR1020097009750A patent/KR20090082213A/ko not_active Withdrawn
- 2007-10-08 CN CNA2007800458003A patent/CN101557804A/zh active Pending
- 2007-10-08 JP JP2009532514A patent/JP2010506845A/ja active Pending
- 2007-10-08 EP EP07843957A patent/EP2079449A2/en not_active Withdrawn
- 2007-10-08 CA CA002673487A patent/CA2673487A1/en not_active Abandoned
- 2007-10-08 BR BRPI0719275-4A2A patent/BRPI0719275A2/pt not_active IP Right Cessation
-
2009
- 2009-04-13 NI NI200900053A patent/NI200900053A/es unknown
- 2009-04-13 GT GT200900082A patent/GT200900082A/es unknown
- 2009-04-14 CO CO09037414A patent/CO6180500A2/es not_active Application Discontinuation
- 2009-04-14 SV SV2009003221A patent/SV2009003221A/es unknown
- 2009-04-16 IL IL198145A patent/IL198145A0/en unknown
- 2009-04-17 NO NO20091530A patent/NO20091530L/no not_active Application Discontinuation
- 2009-05-12 ZA ZA200903283A patent/ZA200903283B/xx unknown
- 2009-05-13 CR CR10794A patent/CR10794A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200903283B (en) | 2010-07-28 |
| CN101557804A (zh) | 2009-10-14 |
| MX2009003926A (es) | 2009-06-26 |
| WO2008048801A3 (en) | 2008-06-05 |
| CR10794A (es) | 2009-09-29 |
| SV2009003221A (es) | 2010-04-15 |
| US20080090902A1 (en) | 2008-04-17 |
| AU2007313017A1 (en) | 2008-04-24 |
| KR20090082213A (ko) | 2009-07-29 |
| BRPI0719275A2 (pt) | 2014-04-29 |
| EP2079449A2 (en) | 2009-07-22 |
| CA2673487A1 (en) | 2008-04-24 |
| IL198145A0 (en) | 2009-12-24 |
| WO2008048801A2 (en) | 2008-04-24 |
| CO6180500A2 (es) | 2010-07-19 |
| NI200900053A (es) | 2010-02-01 |
| EA200970377A1 (ru) | 2009-10-30 |
| JP2010506845A (ja) | 2010-03-04 |
| NO20091530L (no) | 2009-07-06 |
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