GB2039739A - Medicament against glaucoma - Google Patents
Medicament against glaucomaInfo
- Publication number
- GB2039739A GB2039739A GB8007253A GB8007253A GB2039739A GB 2039739 A GB2039739 A GB 2039739A GB 8007253 A GB8007253 A GB 8007253A GB 8007253 A GB8007253 A GB 8007253A GB 2039739 A GB2039739 A GB 2039739A
- Authority
- GB
- United Kingdom
- Prior art keywords
- medicament against
- against glaucoma
- carbon
- carbostyril
- glaucoma
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 208000010412 Glaucoma Diseases 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical class C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 239000004615 ingredient Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Ophthalmology & Optometry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Quinoline Compounds (AREA)
Abstract
A medicament against glaucoma containing as an effective ingredient a carbostyril derivative having an intra- ocular pressure-suppressing action and being represented by the following general formula: <IMAGE> wherein R<1> and R<2> each represent a lower alkyl group, and the carbon-to- carbon bond between the 3-and 4- positions of the carbostyril skeleton is a single or double bond.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8623178A JPS5513241A (en) | 1978-07-14 | 1978-07-14 | Remedy for glaucoma |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| GB2039739A true GB2039739A (en) | 1980-08-20 |
| GB2039739B GB2039739B (en) | 1983-01-26 |
Family
ID=13881010
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB8007253A Expired GB2039739B (en) | 1978-07-14 | 1979-07-13 | Medicament against glaucoma |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP0020765A1 (en) |
| JP (1) | JPS5513241A (en) |
| CH (1) | CH643143A5 (en) |
| DE (1) | DE2952959C2 (en) |
| GB (1) | GB2039739B (en) |
| NL (1) | NL7920004A (en) |
| SE (1) | SE451070B (en) |
| WO (1) | WO1980000215A1 (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU518814B2 (en) * | 1979-01-30 | 1981-10-22 | Otsuka Pharamaceutical Co. | Glaucoma treatment |
| JPS57172004A (en) * | 1981-04-17 | 1982-10-22 | Nichireki Chem Ind Co | Construction of bitminous thin layered pavement |
| FR2539413A1 (en) * | 1983-01-17 | 1984-07-20 | Pos Lab | CARBOSTYRILOXIMINOPROPANOLAMINES USEFUL AS MEDICAMENTS AND PROCESS FOR THEIR PREPARATION |
| JPH0726362B2 (en) * | 1985-04-08 | 1995-03-22 | 日瀝化学工業株式会社 | Bituminous pavement construction method |
| WO1996004911A1 (en) * | 1994-08-10 | 1996-02-22 | Otsuka Pharmaceutical Co., Ltd. | Method of preventing and treating ophthalmic inflammation and/or wound |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5310994B2 (en) * | 1974-06-13 | 1978-04-18 | ||
| US4026897A (en) * | 1974-01-31 | 1977-05-31 | Otsuka Pharmaceutical Company | 5-[1-Hydroxy-2-(substituted-amino)]alkyl-8-hydroxycarbostyril derivatives |
| DK230476A (en) * | 1976-05-26 | 1977-11-27 | E H Sahlertz | LIGHT SIGNS AND WRITING EQUIPMENT |
-
1978
- 1978-07-14 JP JP8623178A patent/JPS5513241A/en active Granted
-
1979
- 1979-07-13 DE DE19792952959 patent/DE2952959C2/en not_active Expired
- 1979-07-13 GB GB8007253A patent/GB2039739B/en not_active Expired
- 1979-07-13 WO PCT/JP1979/000185 patent/WO1980000215A1/en not_active Ceased
- 1979-07-13 CH CH205680A patent/CH643143A5/en not_active IP Right Cessation
- 1979-07-13 NL NL7920004A patent/NL7920004A/en unknown
-
1980
- 1980-02-25 EP EP79900778A patent/EP0020765A1/en not_active Ceased
- 1980-03-13 SE SE8001981A patent/SE451070B/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE2952959T1 (en) | 1981-01-08 |
| SE8001981L (en) | 1980-03-13 |
| GB2039739B (en) | 1983-01-26 |
| JPS5513241A (en) | 1980-01-30 |
| SE451070B (en) | 1987-08-31 |
| CH643143A5 (en) | 1984-05-30 |
| DE2952959C2 (en) | 1986-08-28 |
| WO1980000215A1 (en) | 1980-02-21 |
| EP0020765A4 (en) | 1980-12-02 |
| JPS611007B2 (en) | 1986-01-13 |
| NL7920004A (en) | 1980-05-30 |
| EP0020765A1 (en) | 1981-01-07 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP0256503A3 (en) | Pyridinecarboxamide derivatives and their use as fungicide | |
| FR2361353A1 (en) | CYCLOHEXANE DERIVATIVES USEFUL AS LIQUID CRYSTALS | |
| DE2960820D1 (en) | Carbostyrile derivatives, processes for their preparation and pharmaceutical compositions containing them | |
| FR2391215A1 (en) | NEW IMIDAZOAZINES AND IMIDAZODIAZINES, THEIR PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS | |
| GB2145721B (en) | Compositions for treating glaucoma | |
| CA2013166A1 (en) | Suppression of parathyroid hormone synthesis and secretion | |
| FR2434572A1 (en) | OXIMUM DERIVATIVES FOR THE PROTECTION OF CROPS | |
| GB2039739A (en) | Medicament against glaucoma | |
| IE792329L (en) | Thiazaheterocyclics and process for preparing pyrrolidine¹and piperidine derivatives. | |
| EP0543018A4 (en) | Antidiabetic | |
| IL70797A0 (en) | Triazole derivatives,their preparation and pharmaceutical and agricultural compositions containing them | |
| JPS5424895A (en) | Pyranochromone derivatives and remedies for allergic disorder | |
| FR2393798A1 (en) | TETRAHYDRO-1,3,5-THIADIAZINE-4-ONE DERIVATIVES FOR USE AS INSECTICIDE AND MITICIDE COMPOSITIONS | |
| AU530930B2 (en) | Pharmaceutical compositions and method of treating heart disease | |
| JPS55102516A (en) | Remedy for glaucoma | |
| GB2021588A (en) | Bibenzyl Derivatives, the Preparation thereof and Pharmaceutical Compositions Containing them | |
| FR2364910A1 (en) | NEW THIAZOLIDINES, THEIR PREPARATION AND THEIR APPLICATION AS A PEST CONTROL AGENT | |
| JPS5427564A (en) | 1-branched alkylcarbonyl-3-(3,5-dihalogenophenyl) hydantoins, their preparation, and bactericides for pomicultural and horticultural uses containing the same as active agent. | |
| AU8714082A (en) | N-substituted-tetrahydroisophthalimide derivatives | |
| JPS5419945A (en) | Cyclohexane derivatives, their preparation and herbicides | |
| DE3169918D1 (en) | Cis-c3",c4"-carbonate derivatives of oleandomycin-y, pharmaceutical compositions containing them, and intermediates therefor | |
| JPS5432481A (en) | Carbostyril derivatives | |
| JPS5436287A (en) | Thiadiazolylthiooxacephalosporin | |
| JPS5387330A (en) | Novel thiohydroxymate derivative, its preparation and bactericideand herbicide containing the same | |
| ZA81401B (en) | N-alkyl-carbamic acid indan-4-yl esters,processes for their preparation and their use as fungicides |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PCNP | Patent ceased through non-payment of renewal fee |
Effective date: 19980713 |