GB1088550A - N-substituted 3-imino-benzisothiazolines and their production - Google Patents
N-substituted 3-imino-benzisothiazolines and their productionInfo
- Publication number
- GB1088550A GB1088550A GB3397166A GB3397166A GB1088550A GB 1088550 A GB1088550 A GB 1088550A GB 3397166 A GB3397166 A GB 3397166A GB 3397166 A GB3397166 A GB 3397166A GB 1088550 A GB1088550 A GB 1088550A
- Authority
- GB
- United Kingdom
- Prior art keywords
- carbon atoms
- alkyl
- substituted
- nitro
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 N-substituted 3-imino-benzisothiazolines Chemical class 0.000 title abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 8
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- 229910052736 halogen Inorganic materials 0.000 abstract 4
- 150000002367 halogens Chemical group 0.000 abstract 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 4
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 abstract 3
- 239000003085 diluting agent Substances 0.000 abstract 3
- 239000007788 liquid Substances 0.000 abstract 3
- 239000007787 solid Substances 0.000 abstract 3
- 241000607479 Yersinia pestis Species 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 229910021529 ammonia Inorganic materials 0.000 abstract 2
- 230000001857 anti-mycotic effect Effects 0.000 abstract 2
- 239000002543 antimycotic Substances 0.000 abstract 2
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 150000005840 aryl radicals Chemical class 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 2
- 150000004820 halides Chemical class 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
The invention comprises N-substituted 3-imino-benzisothiazoline of the formula <FORM:1088550/C2/1> in which R1 is an alkyl of 1 to 7 carbon atoms, a cycloalkyl, an aralkyl or an aryl radical, which may be substituted by halogen, nitro, alkyl or alkoxy containing 1 to 6 carbon atoms or dialkylamino containing 2 to 12 carbon atoms, and R2 is at least one of hydrogen, halogen, nitro, alkyl and alkoxy containing 1 to 6 carbon atoms and strong acid salts thereof. The compounds may be made by reacting an N - substituted 3 - halogeno - benzisothiazo lium halide with ammonia, prefarably by intro ducing the halide into an excess of ammonia in methanol. Antimycotic compositions, for use in human or veterinary medicine, comprise the above compounds in admixture with a solid or liquid diluent or carrier.ALSO:An antimycotic composition comprises a compound of the formula: <FORM:1088550/A5-A6/1> wherein R1 is an alkyl of 1 to 7 carbon atoms, a cycloalkyl, an aralkyl or an aryl radical, which may be substituted by halogen, nitro, alkyl or alkoxy containing 1 to 6 carbon atoms or dialkylamino containing 2 to 12 carbon atoms, and R2 is at least one of hydrogen, halogen, nitro, alkyl and alkoxy containing 1 to 6 carbon atoms or a strong acid salt thereof, in admixture with a solid or liquid diluent or carrier. A method of combating mycotic pests comprises applying to a mycotic pest habitat, such as plants, a compound according to the above formula, alone or in admixture with a solid or liquid diluent or carrier.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DEF0046742 | 1965-07-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1088550A true GB1088550A (en) | 1967-10-25 |
Family
ID=7101207
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB3397166A Expired GB1088550A (en) | 1965-07-29 | 1966-07-28 | N-substituted 3-imino-benzisothiazolines and their production |
Country Status (7)
| Country | Link |
|---|---|
| BE (1) | BE684739A (en) |
| CH (1) | CH484181A (en) |
| CY (1) | CY541A (en) |
| DE (1) | DE1545844A1 (en) |
| GB (1) | GB1088550A (en) |
| IL (1) | IL26178A (en) |
| NL (1) | NL6610677A (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1670967B2 (en) * | 1967-12-27 | 1977-10-13 | Bayer Ag, 5090 Leverkusen | 3-IMINO-1,2-BENZISOTHIAZOLINE SALT AND METHOD FOR THEIR PRODUCTION |
| US6376530B1 (en) | 1999-05-10 | 2002-04-23 | Merck & Co., Inc. | Cyclic amidines useful as NMDA NR2B antagonists |
-
1965
- 1965-07-29 DE DE19651545844 patent/DE1545844A1/en not_active Withdrawn
-
1966
- 1966-07-19 IL IL2617866A patent/IL26178A/en unknown
- 1966-07-20 CH CH1046366A patent/CH484181A/en not_active IP Right Cessation
- 1966-07-28 BE BE684739D patent/BE684739A/xx unknown
- 1966-07-28 NL NL6610677A patent/NL6610677A/xx unknown
- 1966-07-28 GB GB3397166A patent/GB1088550A/en not_active Expired
-
1970
- 1970-06-05 CY CY54170A patent/CY541A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CY541A (en) | 1970-06-05 |
| IL26178A (en) | 1970-03-22 |
| CH484181A (en) | 1970-01-15 |
| DE1545844A1 (en) | 1969-12-18 |
| NL6610677A (en) | 1967-01-30 |
| BE684739A (en) | 1967-01-30 |
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