FR2882261B1 - Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 - Google Patents
Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2Info
- Publication number
- FR2882261B1 FR2882261B1 FR0501861A FR0501861A FR2882261B1 FR 2882261 B1 FR2882261 B1 FR 2882261B1 FR 0501861 A FR0501861 A FR 0501861A FR 0501861 A FR0501861 A FR 0501861A FR 2882261 B1 FR2882261 B1 FR 2882261B1
- Authority
- FR
- France
- Prior art keywords
- diabetes
- prevention
- preparation
- treatment
- type
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical class C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 230000002265 prevention Effects 0.000 title 1
- 208000001072 type 2 diabetes mellitus Diseases 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/64—Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (24)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0501861A FR2882261B1 (fr) | 2005-02-21 | 2005-02-21 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| FR0504942A FR2882264A1 (fr) | 2005-02-21 | 2005-05-12 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| FR0505228A FR2882265B1 (fr) | 2005-02-21 | 2005-05-23 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2. |
| KR1020077018993A KR20070104913A (ko) | 2005-02-21 | 2006-02-20 | 2형 당뇨병의 예방 및 치료에 사용될 수 있는 약제의제조를 위한 리모나반트의 용도 |
| BRPI0608183-5A BRPI0608183A2 (pt) | 2005-02-21 | 2006-02-20 | utilização do rimonabante para o preparo de medicamentos úteis na prevenção e no tratamento do diabetes do tipo 2 |
| ZA200707012A ZA200707012B (en) | 2005-02-21 | 2006-02-20 | Use of rimonabant for the preparation of medicaments that can be used in the prevention and treatment of type 2 diabetes |
| JP2007555669A JP2008530189A (ja) | 2005-02-21 | 2006-02-20 | 2型糖尿病の防止および処置において使用することができる医薬品を調製するためのリモナバントの使用 |
| CNA2006800052531A CN101119727A (zh) | 2005-02-21 | 2006-02-20 | 利莫那班在制备用于预防和治疗2型糖尿病的药物中的用途 |
| PCT/FR2006/000376 WO2006087481A1 (fr) | 2005-02-21 | 2006-02-20 | Utilisation du rimonabant pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| EA200701781A EA011618B1 (ru) | 2005-02-21 | 2006-02-20 | Применение римонабанта для получения лекарственных средств, пригодных для профилактики и лечения диабета типа 2 |
| AU2006215444A AU2006215444A1 (en) | 2005-02-21 | 2006-02-20 | Use of rimonabant for the preparation of medicaments that can be used in the prevention and treatment of type 2 diabetes |
| UY29386A UY29386A1 (es) | 2005-02-21 | 2006-02-20 | Utilizción de rimonabant para la preparación de medicamentos útiles en la prevención y el tratamiento de la diabetes de tipo2. |
| EP06709344A EP1853264A1 (fr) | 2005-02-21 | 2006-02-20 | Utilisation du rimonabant pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| MX2007009996A MX2007009996A (es) | 2005-02-21 | 2006-02-20 | Utilizacion de rimonabant para la preparacion de medicamentos utiles en la prevencion y el tratamiento de la diabetes de tipo 2. |
| CA002597245A CA2597245A1 (fr) | 2005-02-21 | 2006-02-20 | Utilisation du rimonabant pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| TW095105631A TW200640457A (en) | 2005-02-21 | 2006-02-20 | Use of rimonabant for the preparation of medicaments useful in the prevention and treatment of type 2 diabetes |
| ARP060100611A AR053812A1 (es) | 2005-02-21 | 2006-02-21 | Utilizacion de rimonabant para la preparacion de medicamentos utiles en la prevencion y el tratamiento de la diabetes de tipo2 |
| TNP2007000297A TNSN07297A1 (en) | 2005-02-21 | 2007-07-31 | Use of rimonabant for the preparation of medicaments that can be used in the prevention and treatment of type 2 diabetes |
| US11/832,865 US20080015229A1 (en) | 2005-02-21 | 2007-08-02 | Use of rimonabant for the preparation of medicaments useful in the prevention and treatment of type 2 diabetes |
| CR9293A CR9293A (es) | 2005-02-21 | 2007-08-07 | Utilizacion de rimonabant para la preparacion de medicamentos utiles en la prevencion y el tratamiento de la diabetes de tipo 2 |
| IL185401A IL185401A0 (en) | 2005-02-21 | 2007-08-20 | Use of rimonabant for the preparation of medicaments that can be used in the prevention and treatment of type 2 diabetes |
| MA30158A MA29262B1 (fr) | 2005-02-21 | 2007-08-23 | Utilisation du rimonabant pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
| NO20074767A NO20074767L (no) | 2005-02-21 | 2007-09-18 | Anvendelse av rimonabant for fremstilling av medikamenter som kan anvendes i forebygging og behandling av type 2 diabetes |
| US12/402,988 US20090197917A1 (en) | 2005-02-21 | 2009-03-12 | Use of rimonabant for the preparation of medicaments useful in the prevention and treatment of type 2 diabetes |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0501861A FR2882261B1 (fr) | 2005-02-21 | 2005-02-21 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2882261A1 FR2882261A1 (fr) | 2006-08-25 |
| FR2882261B1 true FR2882261B1 (fr) | 2009-02-06 |
Family
ID=34954874
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR0501861A Expired - Fee Related FR2882261B1 (fr) | 2005-02-21 | 2005-02-21 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 |
Country Status (3)
| Country | Link |
|---|---|
| CN (1) | CN101119727A (fr) |
| FR (1) | FR2882261B1 (fr) |
| ZA (1) | ZA200707012B (fr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN114452831B (zh) * | 2022-01-24 | 2023-04-25 | 中南大学湘雅医院 | 一种表面涂覆体外循环改性膜及其制备方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2789079B3 (fr) * | 1999-02-01 | 2001-03-02 | Sanofi Synthelabo | Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant |
| US20040122033A1 (en) * | 2002-12-10 | 2004-06-24 | Nargund Ravi P. | Combination therapy for the treatment of obesity |
-
2005
- 2005-02-21 FR FR0501861A patent/FR2882261B1/fr not_active Expired - Fee Related
-
2006
- 2006-02-20 CN CNA2006800052531A patent/CN101119727A/zh active Pending
- 2006-02-20 ZA ZA200707012A patent/ZA200707012B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200707012B (en) | 2008-12-31 |
| CN101119727A (zh) | 2008-02-06 |
| FR2882261A1 (fr) | 2006-08-25 |
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| FR2882261B1 (fr) | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du diabete du type 2 | |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |
Effective date: 20101029 |