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FR2765221B1 - DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION - Google Patents

DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Info

Publication number
FR2765221B1
FR2765221B1 FR9707900A FR9707900A FR2765221B1 FR 2765221 B1 FR2765221 B1 FR 2765221B1 FR 9707900 A FR9707900 A FR 9707900A FR 9707900 A FR9707900 A FR 9707900A FR 2765221 B1 FR2765221 B1 FR 2765221B1
Authority
FR
France
Prior art keywords
anilide
imidazol
piperidin
derivatives
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
FR9707900A
Other languages
French (fr)
Other versions
FR2765221A1 (en
Inventor
Gerard Cremer
Marc Daumas
Marie Angele Adler
Genevieve Dellac
Veronique Rouannet
Christian Hoornaert
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR9707900A priority Critical patent/FR2765221B1/en
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to JP50531399A priority patent/JP2002506458A/en
Priority to PCT/FR1998/001288 priority patent/WO1999000379A1/en
Priority to AU82206/98A priority patent/AU8220698A/en
Priority to EP98932237A priority patent/EP0991639A1/en
Priority to ZA985518A priority patent/ZA985518B/en
Priority to ARP980103032A priority patent/AR013127A1/en
Publication of FR2765221A1 publication Critical patent/FR2765221A1/en
Application granted granted Critical
Publication of FR2765221B1 publication Critical patent/FR2765221B1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR9707900A 1997-06-25 1997-06-25 DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION Expired - Lifetime FR2765221B1 (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
FR9707900A FR2765221B1 (en) 1997-06-25 1997-06-25 DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
PCT/FR1998/001288 WO1999000379A1 (en) 1997-06-25 1998-06-19 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide derivatives, their preparation and application in therapy
AU82206/98A AU8220698A (en) 1997-06-25 1998-06-19 4-{(1h-imidazol-4-yl)piperidin-1-yl}anilide derivatives, their preparation and application in therapy
EP98932237A EP0991639A1 (en) 1997-06-25 1998-06-19 4- (1h-imidazol-4-yl)piperidin-1-yl]anilide derivatives, their preparation and application in therapy
JP50531399A JP2002506458A (en) 1997-06-25 1998-06-19 4-[(1H-Imidazol-4-yl) piperidin-1-yl] anilide Derivatives, Their Preparation and Their Application in Therapy
ZA985518A ZA985518B (en) 1997-06-25 1998-06-24 4-[(1H-imidazol-4-YL) piperidin-1-YL] anilide derivatives their preparation and their application in therapeutics
ARP980103032A AR013127A1 (en) 1997-06-25 1998-06-24 DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-IL) PIPERIDIN-1-IL] ANILIDE, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9707900A FR2765221B1 (en) 1997-06-25 1997-06-25 DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (2)

Publication Number Publication Date
FR2765221A1 FR2765221A1 (en) 1998-12-31
FR2765221B1 true FR2765221B1 (en) 1999-07-30

Family

ID=9508386

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9707900A Expired - Lifetime FR2765221B1 (en) 1997-06-25 1997-06-25 DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Country Status (7)

Country Link
EP (1) EP0991639A1 (en)
JP (1) JP2002506458A (en)
AR (1) AR013127A1 (en)
AU (1) AU8220698A (en)
FR (1) FR2765221B1 (en)
WO (1) WO1999000379A1 (en)
ZA (1) ZA985518B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6887870B1 (en) 1999-10-12 2005-05-03 Bristol-Myers Squibb Company Heterocyclic sodium/proton exchange inhibitors and method
US7501889B2 (en) 2004-04-26 2009-03-10 Rgb Systems, Inc. Method and apparatus for implementing soft switching in a class D amplifier
WO2013012848A1 (en) * 2011-07-18 2013-01-24 Merck Patent Gmbh Benzamides
AU2022221359A1 (en) * 2021-02-12 2023-09-21 Albany College Of Pharmacy And Health Sciences In The City Of Albany Novel compounds comprising a new class of transthyretin ligands for treatment of common age-related comorbidities

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2579596B1 (en) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (IMIDAZOLYL-4) PIPERIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2671083B1 (en) * 1990-12-31 1994-12-23 Inst Nat Sante Rech Med NEWS 4- (4-IMIDAZOLYL) PIPERIDINES SUBSTITUTED IN 1, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS.
FR2674855B1 (en) * 1991-04-03 1994-01-14 Synthelabo PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR2696177B1 (en) * 1992-09-28 1995-05-12 Synthelabo Piperidine derivatives, their preparation and their therapeutic application.
DE4325822A1 (en) * 1993-07-31 1995-02-02 Hoechst Ag Substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic agent, and medicament containing them

Also Published As

Publication number Publication date
JP2002506458A (en) 2002-02-26
AU8220698A (en) 1999-01-19
ZA985518B (en) 1999-01-28
WO1999000379A1 (en) 1999-01-07
EP0991639A1 (en) 2000-04-12
FR2765221A1 (en) 1998-12-31
AR013127A1 (en) 2000-12-13

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