FR2765221B1 - DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION - Google Patents
DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONInfo
- Publication number
- FR2765221B1 FR2765221B1 FR9707900A FR9707900A FR2765221B1 FR 2765221 B1 FR2765221 B1 FR 2765221B1 FR 9707900 A FR9707900 A FR 9707900A FR 9707900 A FR9707900 A FR 9707900A FR 2765221 B1 FR2765221 B1 FR 2765221B1
- Authority
- FR
- France
- Prior art keywords
- anilide
- imidazol
- piperidin
- derivatives
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- -1 1H-IMIDAZOL-4-YL Chemical class 0.000 title 2
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9707900A FR2765221B1 (en) | 1997-06-25 | 1997-06-25 | DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| PCT/FR1998/001288 WO1999000379A1 (en) | 1997-06-25 | 1998-06-19 | 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide derivatives, their preparation and application in therapy |
| AU82206/98A AU8220698A (en) | 1997-06-25 | 1998-06-19 | 4-{(1h-imidazol-4-yl)piperidin-1-yl}anilide derivatives, their preparation and application in therapy |
| EP98932237A EP0991639A1 (en) | 1997-06-25 | 1998-06-19 | 4- (1h-imidazol-4-yl)piperidin-1-yl]anilide derivatives, their preparation and application in therapy |
| JP50531399A JP2002506458A (en) | 1997-06-25 | 1998-06-19 | 4-[(1H-Imidazol-4-yl) piperidin-1-yl] anilide Derivatives, Their Preparation and Their Application in Therapy |
| ZA985518A ZA985518B (en) | 1997-06-25 | 1998-06-24 | 4-[(1H-imidazol-4-YL) piperidin-1-YL] anilide derivatives their preparation and their application in therapeutics |
| ARP980103032A AR013127A1 (en) | 1997-06-25 | 1998-06-24 | DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-IL) PIPERIDIN-1-IL] ANILIDE, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9707900A FR2765221B1 (en) | 1997-06-25 | 1997-06-25 | DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2765221A1 FR2765221A1 (en) | 1998-12-31 |
| FR2765221B1 true FR2765221B1 (en) | 1999-07-30 |
Family
ID=9508386
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR9707900A Expired - Lifetime FR2765221B1 (en) | 1997-06-25 | 1997-06-25 | DERIVATIVES OF 4 - [(1H-IMIDAZOL-4-YL) PIPERIDIN-1-YL] ANILIDE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP0991639A1 (en) |
| JP (1) | JP2002506458A (en) |
| AR (1) | AR013127A1 (en) |
| AU (1) | AU8220698A (en) |
| FR (1) | FR2765221B1 (en) |
| WO (1) | WO1999000379A1 (en) |
| ZA (1) | ZA985518B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6887870B1 (en) | 1999-10-12 | 2005-05-03 | Bristol-Myers Squibb Company | Heterocyclic sodium/proton exchange inhibitors and method |
| US7501889B2 (en) | 2004-04-26 | 2009-03-10 | Rgb Systems, Inc. | Method and apparatus for implementing soft switching in a class D amplifier |
| WO2013012848A1 (en) * | 2011-07-18 | 2013-01-24 | Merck Patent Gmbh | Benzamides |
| AU2022221359A1 (en) * | 2021-02-12 | 2023-09-21 | Albany College Of Pharmacy And Health Sciences In The City Of Albany | Novel compounds comprising a new class of transthyretin ligands for treatment of common age-related comorbidities |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2579596B1 (en) * | 1985-03-26 | 1987-11-20 | Inst Nat Sante Rech Med | (IMIDAZOLYL-4) PIPERIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| FR2671083B1 (en) * | 1990-12-31 | 1994-12-23 | Inst Nat Sante Rech Med | NEWS 4- (4-IMIDAZOLYL) PIPERIDINES SUBSTITUTED IN 1, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS. |
| FR2674855B1 (en) * | 1991-04-03 | 1994-01-14 | Synthelabo | PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION. |
| FR2696177B1 (en) * | 1992-09-28 | 1995-05-12 | Synthelabo | Piperidine derivatives, their preparation and their therapeutic application. |
| DE4325822A1 (en) * | 1993-07-31 | 1995-02-02 | Hoechst Ag | Substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic agent, and medicament containing them |
-
1997
- 1997-06-25 FR FR9707900A patent/FR2765221B1/en not_active Expired - Lifetime
-
1998
- 1998-06-19 EP EP98932237A patent/EP0991639A1/en not_active Withdrawn
- 1998-06-19 WO PCT/FR1998/001288 patent/WO1999000379A1/en not_active Ceased
- 1998-06-19 AU AU82206/98A patent/AU8220698A/en not_active Abandoned
- 1998-06-19 JP JP50531399A patent/JP2002506458A/en active Pending
- 1998-06-24 ZA ZA985518A patent/ZA985518B/en unknown
- 1998-06-24 AR ARP980103032A patent/AR013127A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2002506458A (en) | 2002-02-26 |
| AU8220698A (en) | 1999-01-19 |
| ZA985518B (en) | 1999-01-28 |
| WO1999000379A1 (en) | 1999-01-07 |
| EP0991639A1 (en) | 2000-04-12 |
| FR2765221A1 (en) | 1998-12-31 |
| AR013127A1 (en) | 2000-12-13 |
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