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FI973207A7 - Heterosyklisiä yhdisteitä - Google Patents

Heterosyklisiä yhdisteitä Download PDF

Info

Publication number
FI973207A7
FI973207A7 FI973207A FI973207A FI973207A7 FI 973207 A7 FI973207 A7 FI 973207A7 FI 973207 A FI973207 A FI 973207A FI 973207 A FI973207 A FI 973207A FI 973207 A7 FI973207 A7 FI 973207A7
Authority
FI
Finland
Prior art keywords
heterocyclic compounds
heterocyclic
compounds
Prior art date
Application number
FI973207A
Other languages
English (en)
Swedish (sv)
Other versions
FI973207A0 (fi
Inventor
Makoto Takemura
Youichi Kimura
Katsuhiro Kawakami
Kenichi Kimura
Hitoshi Ohki
Norikazu Matsuhashi
Haruko Kawato
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of FI973207A0 publication Critical patent/FI973207A0/fi
Publication of FI973207A7 publication Critical patent/FI973207A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Earth Drilling (AREA)
  • Stereophonic System (AREA)
  • Use Of Switch Circuits For Exchanges And Methods Of Control Of Multiplex Exchanges (AREA)
FI973207A 1995-02-02 1997-08-01 Heterosyklisiä yhdisteitä FI973207A7 (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP1561495 1995-02-02
JP1948195 1995-02-07
JP1947895 1995-02-07
PCT/JP1996/000208 WO1996023782A1 (en) 1995-02-02 1996-02-01 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
FI973207A0 FI973207A0 (fi) 1997-08-01
FI973207A7 true FI973207A7 (fi) 1997-10-01

Family

ID=27281082

Family Applications (1)

Application Number Title Priority Date Filing Date
FI973207A FI973207A7 (fi) 1995-02-02 1997-08-01 Heterosyklisiä yhdisteitä

Country Status (13)

Country Link
US (1) US5849757A (fi)
EP (2) EP1304329B1 (fi)
KR (1) KR100389773B1 (fi)
AT (2) ATE411309T1 (fi)
CA (1) CA2212007C (fi)
DE (2) DE69627985T2 (fi)
DK (1) DK0807630T3 (fi)
ES (2) ES2315432T3 (fi)
FI (1) FI973207A7 (fi)
NO (1) NO314546B1 (fi)
PT (1) PT807630E (fi)
TW (1) TW487701B (fi)
WO (1) WO1996023782A1 (fi)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6121285A (en) * 1995-11-22 2000-09-19 Daiichi Pharmaceutical Co., Ltd. Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
ATE317393T1 (de) * 1995-11-22 2006-02-15 Daiichi Seiyaku Co Substituierte aminocycloalkylpyrrolidinderivate
TW519542B (en) * 1996-09-27 2003-02-01 Daiichi Seiyaku Co Bicyclic amine derivative
ZA984527B (en) * 1997-05-30 1998-12-03 Daiichi Seiyaku Co Substituted cyclobutylamine derivative
RU2193558C2 (ru) 1997-09-15 2002-11-27 Дзе Проктер Энд Гэмбл Компани Производные хинолона и фармацевтическая композиция на их основе
GB9822440D0 (en) * 1998-10-14 1998-12-09 Smithkline Beecham Plc Medicaments
DE60011264T2 (de) * 1999-03-10 2005-07-14 Daiichi Pharmaceutical Co., Ltd. Aminomethylpyrrolidin-derivate mit aromatischen substituenten
WO2000055116A1 (en) * 1999-03-17 2000-09-21 Daiichi Pharmaceutical Co., Ltd. Process for producing 5-amino-8- alkylquinolo necarboxylic acid derivatives and intermediates in the production thereof
BR0111248A (pt) * 2000-03-31 2003-07-08 Daiichi Seiyaku Co Derivados de ácido quinolonacarboxìlico
IL155976A0 (en) * 2000-11-20 2003-12-23 Daiichi Seiyaku Co Dehalogeno compounds
GB0112834D0 (en) * 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
KR101041277B1 (ko) * 2002-05-17 2011-06-14 다이이찌 세이야꾸 가부시기가이샤 퀴놀론카르복실산 유도체의 제조방법
US6875784B2 (en) * 2002-10-09 2005-04-05 Pharmacia & Upjohn Company Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
EP1632482A4 (en) * 2003-06-06 2009-10-28 Daiichi Seiyaku Co INTERMEDIATES AND PROCESS FOR THE PRODUCTION OF OPTICALLY ACTIVE QUINOLONECARBOXYLIC ACID DERIVATIVES
WO2004113321A1 (ja) * 2003-06-19 2004-12-29 Daiichi Pharmaceutical Co., Ltd. 選択的なアミノ置換基導入法
JP4619952B2 (ja) * 2003-09-29 2011-01-26 第一三共株式会社 8−シアノキノロンカルボン酸誘導体
US7569599B2 (en) 2003-12-12 2009-08-04 Daiichi Pharmaceutical Co., Ltd. Intermediates for the production of optically active cyclopropylamine derivatives and process for the production of the intermediates
WO2007110835A2 (en) 2006-03-28 2007-10-04 The Procter & Gamble Company A coupling process for preparing quinolone intermediates
MY148393A (en) 2006-03-28 2013-04-15 Taigen Biotechnology Co Ltd Malate salts, and polymorphs of (3s, 5s)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
WO2008082009A2 (en) 2007-01-05 2008-07-10 Daiichi Sankyo Company, Limited Fused substituted aminopyrrolidine derivative
US8278313B2 (en) 2008-03-11 2012-10-02 Abbott Laboratories Macrocyclic spiro pyrimidine derivatives
US8436005B2 (en) 2008-04-03 2013-05-07 Abbott Laboratories Macrocyclic pyrimidine derivatives
US10300155B2 (en) 2015-12-31 2019-05-28 Washington University Alpha-synuclein ligands

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5772981A (en) * 1980-10-22 1982-05-07 Dainippon Pharmaceut Co Ltd 1,8-naphthyridine derivative and its salt
JPS60260577A (ja) * 1984-06-06 1985-12-23 Dainippon Pharmaceut Co Ltd 1,8−ナフチリジン誘導体
CS274601B2 (en) * 1983-07-27 1991-09-15 Dainippon Pharmaceutical Co Method of 1,8-naphthyridine derivative production
IL79189A (en) * 1985-06-26 1990-07-12 Daiichi Seiyaku Co Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co Pyridonecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
JP2844079B2 (ja) * 1988-05-23 1999-01-06 塩野義製薬株式会社 ピリドンカルボン酸系抗菌剤
IE66202B1 (en) * 1989-08-16 1995-12-13 Pfizer Azabicyclo quinolone carboxylic acids
RU2100351C1 (ru) * 1991-05-28 1997-12-27 Дайити Фармасьютикал Ко., Лтд. Производные пиридонкарбоновой кислоты и композиция на их основе
KR960011370B1 (ko) * 1991-12-31 1996-08-22 재단법인 한국화학연구소 스피로알킬아민 유도체와 그의 제조방법
EP0550016A1 (en) * 1991-12-31 1993-07-07 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and processes for preparing same
ATE216993T1 (de) * 1994-02-04 2002-05-15 Dainippon Pharmaceutical Co Pyridoncarbonsäurederivate substituiert von bicyclischer aminogruppe, deren ester und salze, und bicyclisches amin als zwischenprodukt davon
ATE317393T1 (de) * 1995-11-22 2006-02-15 Daiichi Seiyaku Co Substituierte aminocycloalkylpyrrolidinderivate

Also Published As

Publication number Publication date
KR100389773B1 (ko) 2003-10-23
NO973530D0 (no) 1997-07-31
DE69627985T2 (de) 2004-02-19
EP0807630A4 (en) 1998-05-13
FI973207A0 (fi) 1997-08-01
NO314546B1 (no) 2003-04-07
ES2315432T3 (es) 2009-04-01
ES2198474T3 (es) 2004-02-01
PT807630E (pt) 2003-08-29
EP1304329B1 (en) 2008-10-15
US5849757A (en) 1998-12-15
EP0807630A1 (en) 1997-11-19
DE69637717D1 (de) 2008-11-27
TW487701B (en) 2002-05-21
NO973530L (no) 1997-10-02
ATE239720T1 (de) 2003-05-15
WO1996023782A1 (en) 1996-08-08
EP1304329A3 (en) 2004-09-15
CA2212007A1 (en) 1996-08-08
DE69627985D1 (de) 2003-06-12
CA2212007C (en) 2004-09-14
DK0807630T3 (da) 2003-09-01
KR19980701860A (ko) 1998-06-25
EP0807630B1 (en) 2003-05-07
ATE411309T1 (de) 2008-10-15
EP1304329A2 (en) 2003-04-23

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