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FI971934A7 - Asyloituja bentsyyliglykosideja sileälihassolulisääntymisen inhibiittoreina - Google Patents

Asyloituja bentsyyliglykosideja sileälihassolulisääntymisen inhibiittoreina Download PDF

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Publication number
FI971934A7
FI971934A7 FI971934A FI971934A FI971934A7 FI 971934 A7 FI971934 A7 FI 971934A7 FI 971934 A FI971934 A FI 971934A FI 971934 A FI971934 A FI 971934A FI 971934 A7 FI971934 A7 FI 971934A7
Authority
FI
Finland
Prior art keywords
inhibitors
cell proliferation
smooth muscle
muscle cell
benzyl glycosides
Prior art date
Application number
FI971934A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI971934A0 (fi
Inventor
Thomas T Nguyen
John Watson Ellingboe
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/531,142 external-priority patent/US5773420A/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of FI971934A0 publication Critical patent/FI971934A0/fi
Publication of FI971934A7 publication Critical patent/FI971934A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
FI971934A 1994-11-07 1997-05-06 Asyloituja bentsyyliglykosideja sileälihassolulisääntymisen inhibiittoreina FI971934A7 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33528694A 1994-11-07 1994-11-07
US08/531,142 US5773420A (en) 1994-11-07 1995-10-20 Acylated benzylglycosides as inhibitors of smooth muscle cell proliferation
PCT/US1995/014795 WO1996014325A1 (fr) 1994-11-07 1995-11-03 Benzylglycosides acyles en tant qu'inhibiteurs de la proliferation cellulaire du muscle lisse

Publications (2)

Publication Number Publication Date
FI971934A0 FI971934A0 (fi) 1997-05-06
FI971934A7 true FI971934A7 (fi) 1997-05-06

Family

ID=26989635

Family Applications (1)

Application Number Title Priority Date Filing Date
FI971934A FI971934A7 (fi) 1994-11-07 1997-05-06 Asyloituja bentsyyliglykosideja sileälihassolulisääntymisen inhibiittoreina

Country Status (16)

Country Link
EP (1) EP0791004B1 (fr)
JP (1) JPH10508610A (fr)
AT (1) ATE184283T1 (fr)
AU (1) AU703338B2 (fr)
BR (1) BR9509586A (fr)
CA (1) CA2204530A1 (fr)
DE (1) DE69512081T2 (fr)
DK (1) DK0791004T3 (fr)
ES (1) ES2136314T3 (fr)
FI (1) FI971934A7 (fr)
GR (1) GR3031731T3 (fr)
HU (1) HUT77757A (fr)
IL (1) IL115745A (fr)
MX (1) MX9702966A (fr)
NZ (1) NZ296037A (fr)
WO (1) WO1996014325A1 (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6664243B1 (en) 1998-11-24 2003-12-16 Wyeth Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
US6291434B1 (en) 1998-11-24 2001-09-18 American Home Products Corp. Benzylmaltotriosides as inhibitors of smooth muscle cell proliferation
AU5706699A (en) * 1998-11-24 2000-06-13 American Home Products Corporation Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
WO2000031096A1 (fr) * 1998-11-24 2000-06-02 American Home Products Corporation Benzylmaltosides acetal utilises comme inhibiteurs de la proliferation cellulaire des muscles lisses
US6340670B1 (en) 1998-11-24 2002-01-22 American Home Products Corporation Acetal benzylmaltosides as inhibitors of smooth muscle cell proliferation
US6258784B1 (en) 1998-11-24 2001-07-10 American Home Products Corp. Acetal benzylmaltosides as inhibitors of smooth muscle cell proliferation
BR9915571A (pt) * 1998-11-24 2001-08-14 American Home Prod Benzilmaltosìdeos como inibidores de proliferação de célula muscular lisa
US6339064B1 (en) 1998-11-24 2002-01-15 American Home Products Corporation Benzylglycosylamides as inhibitors of smooth muscle cell proliferation
US6362170B1 (en) 1998-11-24 2002-03-26 American Home Products Corporation Benzylglycosylamides as inhibitors of smooth muscle cell proliferation
JP2003521460A (ja) * 1998-11-24 2003-07-15 ワイス 平滑筋細胞増殖の阻害薬としてのアセチル化ベンジルマルトシド
US7132402B2 (en) 1998-11-24 2006-11-07 Wyeth Acylated benzylmaltosides as inhibitors of smooth muscle cell proliferation
US6451767B1 (en) 1998-11-24 2002-09-17 Wyeth Benzylmaltotriosides as inhibitors of smooth muscle cell proliferation
US6187755B1 (en) 1998-11-24 2001-02-13 American Home Products Corporation Benzylmaltosides as inhibitors of smooth muscle cell proliferation
US7081448B2 (en) 1998-11-24 2006-07-25 Wyeth Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
CA2350759A1 (fr) * 1998-11-24 2000-06-02 Paul Jeffrey Dollings Benzylmaltotriosides inhibiteurs de la proliferation des cellules des muscles lisses
AU1743800A (en) * 1998-11-24 2000-06-26 American Home Products Corporation Acetal benzylmaltosides as inhibitors of smooth muscle cell proliferation
EP2124948B1 (fr) 2007-02-21 2017-07-26 NC bit, Inc. Compositions pour le traitement de troubles vasculaires hyperprolifératifs et de cancers
CN110152001B (zh) * 2019-05-20 2021-08-10 昆山德瑞生物科技有限公司 小分子化合物的用途及其组合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431637A (en) * 1982-10-25 1984-02-14 American Cyanamid Company Polycation salts of bis (or tris) [4-O-polyhexose-oxy]-arylene sulfate derivatives
FR2634485B1 (fr) * 1988-07-21 1992-02-28 Sanopi Glycosaminoglycanes selectivement o-acyles, leur preparation et compositions pharmaceutiques les contenant
US5032679A (en) * 1988-12-15 1991-07-16 Glycomed, Inc. Heparin fragments as inhibitors of smooth muscle cell proliferation
EP0454220B1 (fr) * 1990-04-23 1993-08-18 Akzo Nobel N.V. Dérivés d'hydrates de carbone comprenant une unité trisaccharide

Also Published As

Publication number Publication date
BR9509586A (pt) 1997-12-23
HUT77757A (hu) 1998-07-28
AU3935395A (en) 1996-05-31
IL115745A (en) 2000-11-21
FI971934A0 (fi) 1997-05-06
ES2136314T3 (es) 1999-11-16
DE69512081T2 (de) 2000-02-03
AU703338B2 (en) 1999-03-25
EP0791004B1 (fr) 1999-09-08
NZ296037A (en) 1999-05-28
MX9702966A (es) 1997-06-28
WO1996014325A1 (fr) 1996-05-17
GR3031731T3 (en) 2000-02-29
IL115745A0 (en) 1996-01-19
JPH10508610A (ja) 1998-08-25
DK0791004T3 (da) 1999-11-29
DE69512081D1 (de) 1999-10-14
ATE184283T1 (de) 1999-09-15
CA2204530A1 (fr) 1996-05-17
EP0791004A1 (fr) 1997-08-27

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