FI950023L - Uudet D-vitamiinianalogit - Google Patents
Uudet D-vitamiinianalogit Download PDFInfo
- Publication number
- FI950023L FI950023L FI950023A FI950023A FI950023L FI 950023 L FI950023 L FI 950023L FI 950023 A FI950023 A FI 950023A FI 950023 A FI950023 A FI 950023A FI 950023 L FI950023 L FI 950023L
- Authority
- FI
- Finland
- Prior art keywords
- analogues
- new vitamin
- vitamin
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Nutrition Science (AREA)
- Dermatology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9214202 | 1992-07-03 | ||
| GB929214202A GB9214202D0 (en) | 1992-07-03 | 1992-07-03 | Chemical compounds |
| DK9300196 | 1993-06-07 | ||
| PCT/DK1993/000196 WO1994001398A1 (en) | 1992-07-03 | 1993-06-07 | Vitamin d analogues |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI950023L true FI950023L (fi) | 1995-01-02 |
| FI950023A0 FI950023A0 (fi) | 1995-01-02 |
| FI106120B FI106120B (fi) | 2000-11-30 |
Family
ID=10718182
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI950023A FI106120B (fi) | 1992-07-03 | 1995-01-02 | Menetelmä uusien D-vitamiinianalogien valmistamiseksi |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5545633A (fi) |
| EP (1) | EP0648207B1 (fi) |
| JP (1) | JPH08504746A (fi) |
| KR (1) | KR100285146B1 (fi) |
| AT (1) | ATE150013T1 (fi) |
| AU (1) | AU667378B2 (fi) |
| CA (1) | CA2131631A1 (fi) |
| DE (1) | DE69308852T2 (fi) |
| DK (1) | DK0648207T3 (fi) |
| ES (1) | ES2101319T3 (fi) |
| FI (1) | FI106120B (fi) |
| GB (1) | GB9214202D0 (fi) |
| GR (1) | GR3023407T3 (fi) |
| HU (1) | HU222775B1 (fi) |
| NZ (1) | NZ253026A (fi) |
| RU (1) | RU2114825C1 (fi) |
| WO (1) | WO1994001398A1 (fi) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9226860D0 (en) * | 1992-12-23 | 1993-02-17 | Leo Pharm Prod Ltd | Novel treatment |
| DE4427690A1 (de) * | 1994-08-04 | 1996-02-08 | Bogdahn Ulrich Prof | Deuterium enthaltende pharmazeutische Zusammensetzung als Zytostatikum oder Tumor-Therapeutikum |
| ES2130522T3 (es) * | 1994-12-14 | 1999-07-01 | Duphar Int Res | Compuestos de vitamina d y metodo para preparar estos compuestos. |
| TW422696B (en) | 1995-03-20 | 2001-02-21 | Katsuhiko Mukai | Ophthalmic composition containing active vitamin D |
| GB9526208D0 (en) * | 1995-12-21 | 1996-02-21 | Res Inst Medicine Chem | Chemical compounds |
| GB9721156D0 (en) | 1997-10-06 | 1997-12-03 | Leo Pharm Prod Ltd | Novel vitamin d analogues |
| US20030220234A1 (en) * | 1998-11-02 | 2003-11-27 | Selvaraj Naicker | Deuterated cyclosporine analogs and their use as immunodulating agents |
| ES2266564T3 (es) | 2001-10-19 | 2007-03-01 | Isotechnika Inc. | Sintesis de analogos de cicloporinas. |
| US8404667B2 (en) * | 2006-12-29 | 2013-03-26 | Wisconsin Alumni Research Foundation | Compounds, compositions, kits and methods of use to orally and topically treat acne and other skin conditions by 19-Nor vitamin D analog |
| WO2006051106A1 (en) | 2004-11-12 | 2006-05-18 | Bioxell Spa | Combined use of vitamin d derivatives and anti-proliferative agents for treating bladder cancer |
| EP1817279B1 (en) | 2004-11-22 | 2010-05-26 | Wisconsin Alumni Research Foundation | 17,20(z)-dehydro vitamin d analogs and their uses |
| US8193169B2 (en) * | 2006-04-06 | 2012-06-05 | Wisconsin Alumni Research Foundation | (20R)-2α-methyl-19,26,2-trinor-vitamin D analogs |
| US8193170B2 (en) | 2008-07-10 | 2012-06-05 | Wisconsin Alumni Research Foundation | 2-methylene-19,26-dinor-(20R,22E,25R)-vitamin D analogs |
| US7879829B2 (en) * | 2008-07-10 | 2011-02-01 | Wisconsin Alumni Research Foundation | 19-nor-vitamin D analogs with 1,2-dihydrofuran ring |
| US7888339B2 (en) | 2008-07-10 | 2011-02-15 | Wisconsin Alumni Research Foundation | 2-methylene-20(21)-dehydro-19-nor-vitamin D analogs |
| US8222236B2 (en) * | 2008-07-10 | 2012-07-17 | Wisconsin Alumni Research Foundation | 2-methylene-(20E)-20(22)-dehydro-19-nor-vitamin D analogs |
| US7893043B2 (en) | 2008-07-10 | 2011-02-22 | Wisconsin Alumni Research Foundation | 2-methylene-(17Z)-17(20)-dehydro-19,21-dinor-vitamin D analogs |
| US7648974B1 (en) * | 2008-07-10 | 2010-01-19 | Wisconsin Alumni Research Foundation | 19-nor-vitamin D analogs with 3,2-dihydrofuran ring |
| US7713953B2 (en) * | 2008-07-10 | 2010-05-11 | Wisconsin Alumni Research Foundation | 2-methylene-(22E)-25-(1-methylene-hexyl)-26,27-cyclo-22-dehydro-19-nor-vitamin D analogs |
| US8399439B2 (en) * | 2008-07-10 | 2013-03-19 | Wisconsin Alumni Research Foundation | 2-methylene-19,26-dinor-(20S,22E,25R)-vitamin D analogs |
| RU2509773C2 (ru) * | 2008-07-15 | 2014-03-20 | Теракос, Инк. | Дейтерированные бензилбензольные производные и способы применения |
| CN102341110B (zh) | 2009-01-27 | 2017-04-12 | 博格有限责任公司 | 用于减轻与化疗有关的副作用的维生素d3及其类似物 |
| CN105663146B (zh) | 2009-08-14 | 2020-09-11 | 博格有限责任公司 | 用于治疗脱发的维生素d3及其类似物 |
| WO2011041596A2 (en) | 2009-10-02 | 2011-04-07 | Wisconsin Alumni Research Foundation | 19-nor-vitamin d analogs with 1,2-or 3,2-cyclopentene ring |
| MX2012003883A (es) | 2009-10-02 | 2012-06-27 | Wisconsin Alumni Res Found | Analogos de (20s,22e)-2-metileno-19-nor-22-ene-1a,25-dihidroxovita mina d3. |
| AU2012262174B2 (en) | 2011-06-03 | 2016-12-01 | Wisconsin Alumni Research Foundation | (22E)-2-methylene-26,27-cyclo-22-dehydro-1alpha-hydroxy-19-norvitamin D3 derivatives |
| US10479764B2 (en) | 2011-06-28 | 2019-11-19 | Wisconsin Alumni Research Foundation | 2-methylene-(22E)-25-hexanoyl-24-oxo-26,27-cyclo-22-dehydro-19-nor-vitamin D analogs |
| US20130178449A1 (en) | 2011-07-18 | 2013-07-11 | Wisconsin Alumni Research Foundation | 2-Methylene-20(21)-Dehydro-19,24,25,26,27-Pentanor-Vitamin D Analogs |
| US9416102B2 (en) | 2013-01-23 | 2016-08-16 | Wisconsin Alumni Research Foundation | (22E)-2-methylene-22-dehydro-1α,24,25-trihydroxy-19-nor-vitamin D3 analogs |
| SG11201509715UA (en) | 2013-05-29 | 2015-12-30 | Berg Llc | Preventing or mitigating chemotherapy induced alopecia using vitamin d |
| AU2015352677B2 (en) | 2014-11-25 | 2019-10-24 | Trophea Development AB | Treatment of skin atrophy with a combination of triiodothyroacetic acid (TRIAC) and dehydroepiandrosterone (DHEA) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4804502A (en) * | 1988-01-20 | 1989-02-14 | Hoffmann-La Roche Inc. | Vitamin D compounds |
| GB9017890D0 (en) * | 1990-08-15 | 1990-09-26 | Leo Pharm Prod Ltd | Chemical compounds i |
-
1992
- 1992-07-03 GB GB929214202A patent/GB9214202D0/en active Pending
-
1993
- 1993-06-07 CA CA002131631A patent/CA2131631A1/en not_active Abandoned
- 1993-06-07 DE DE69308852T patent/DE69308852T2/de not_active Expired - Fee Related
- 1993-06-07 JP JP6502829A patent/JPH08504746A/ja not_active Withdrawn
- 1993-06-07 AT AT93912681T patent/ATE150013T1/de not_active IP Right Cessation
- 1993-06-07 AU AU43111/93A patent/AU667378B2/en not_active Ceased
- 1993-06-07 EP EP93912681A patent/EP0648207B1/en not_active Expired - Lifetime
- 1993-06-07 DK DK93912681.9T patent/DK0648207T3/da active
- 1993-06-07 NZ NZ253026A patent/NZ253026A/en unknown
- 1993-06-07 US US08/295,755 patent/US5545633A/en not_active Expired - Fee Related
- 1993-06-07 HU HU9402484A patent/HU222775B1/hu not_active IP Right Cessation
- 1993-06-07 WO PCT/DK1993/000196 patent/WO1994001398A1/en not_active Ceased
- 1993-06-07 ES ES93912681T patent/ES2101319T3/es not_active Expired - Lifetime
- 1993-06-07 KR KR1019940703687A patent/KR100285146B1/ko not_active Expired - Fee Related
- 1993-06-07 RU RU94046411A patent/RU2114825C1/ru not_active IP Right Cessation
-
1995
- 1995-01-02 FI FI950023A patent/FI106120B/fi active
-
1997
- 1997-05-12 GR GR970401061T patent/GR3023407T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2114825C1 (ru) | 1998-07-10 |
| HU9402484D0 (en) | 1994-11-28 |
| ATE150013T1 (de) | 1997-03-15 |
| DE69308852D1 (de) | 1997-04-17 |
| ES2101319T3 (es) | 1997-07-01 |
| HUT68025A (en) | 1995-05-29 |
| FI106120B (fi) | 2000-11-30 |
| KR100285146B1 (ko) | 2001-04-02 |
| KR950700876A (ko) | 1995-02-20 |
| NZ253026A (en) | 1997-07-27 |
| EP0648207B1 (en) | 1997-03-12 |
| EP0648207A1 (en) | 1995-04-19 |
| HU222775B1 (hu) | 2003-10-28 |
| DE69308852T2 (de) | 1997-11-27 |
| AU667378B2 (en) | 1996-03-21 |
| GR3023407T3 (en) | 1997-08-29 |
| DK0648207T3 (da) | 1997-06-23 |
| GB9214202D0 (en) | 1992-08-12 |
| CA2131631A1 (en) | 1994-01-20 |
| US5545633A (en) | 1996-08-13 |
| JPH08504746A (ja) | 1996-05-21 |
| WO1994001398A1 (en) | 1994-01-20 |
| AU4311193A (en) | 1994-01-31 |
| RU94046411A (ru) | 1996-10-10 |
| FI950023A0 (fi) | 1995-01-02 |
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