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FI941309L - Substituoituja pyridopyrmidiinejä korkean verenpaineen vastaisina aineina - Google Patents

Substituoituja pyridopyrmidiinejä korkean verenpaineen vastaisina aineina Download PDF

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Publication number
FI941309L
FI941309L FI941309A FI941309A FI941309L FI 941309 L FI941309 L FI 941309L FI 941309 A FI941309 A FI 941309A FI 941309 A FI941309 A FI 941309A FI 941309 L FI941309 L FI 941309L
Authority
FI
Finland
Prior art keywords
antihypertensive agents
pyridopyrimidines
substituted
substituted pyridopyrimidines
antihypertensive
Prior art date
Application number
FI941309A
Other languages
English (en)
Swedish (sv)
Other versions
FI941309A0 (fi
FI108135B (fi
Inventor
John Watson Ellingboe
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/179,461 external-priority patent/US5466692A/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of FI941309A0 publication Critical patent/FI941309A0/fi
Publication of FI941309L publication Critical patent/FI941309L/fi
Application granted granted Critical
Publication of FI108135B publication Critical patent/FI108135B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI941309A 1993-03-24 1994-03-21 Menetelmä terapeuttisesti aktiivisten 7-okso-8-[2'-(1H-tetrasol-5-yyli)bifenyl-4-yylimetyyli]-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidiinijohdannaisten valmistamiseksi FI108135B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US3661593A 1993-03-24 1993-03-24
US3661593 1993-03-24
US08/179,461 US5466692A (en) 1993-03-24 1994-01-10 Substituted pyridopyrimidines and antihypertensives
US17946194 1994-01-10

Publications (3)

Publication Number Publication Date
FI941309A0 FI941309A0 (fi) 1994-03-21
FI941309L true FI941309L (fi) 1994-09-25
FI108135B FI108135B (fi) 2001-11-30

Family

ID=26713326

Family Applications (1)

Application Number Title Priority Date Filing Date
FI941309A FI108135B (fi) 1993-03-24 1994-03-21 Menetelmä terapeuttisesti aktiivisten 7-okso-8-[2'-(1H-tetrasol-5-yyli)bifenyl-4-yylimetyyli]-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidiinijohdannaisten valmistamiseksi

Country Status (16)

Country Link
EP (2) EP0618207B1 (fi)
JP (1) JPH06321945A (fi)
AT (1) ATE175413T1 (fi)
AU (1) AU669966B2 (fi)
BR (1) BR9401261A (fi)
CA (1) CA2119692A1 (fi)
DE (1) DE69415706T2 (fi)
DK (1) DK0618207T3 (fi)
ES (1) ES2126061T3 (fi)
FI (1) FI108135B (fi)
GR (1) GR3029879T3 (fi)
HU (1) HU222240B1 (fi)
LV (1) LV12261B (fi)
NZ (1) NZ260164A (fi)
PH (1) PH30373A (fi)
SG (1) SG47714A1 (fi)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1149196C (zh) 1998-07-06 2004-05-12 布里斯托尔-迈尔斯斯奎布公司 作为血管紧张肽和内皮肽受体双重拮抗剂的联苯基磺酰胺
HRP20151233T1 (hr) * 2007-06-07 2015-12-18 Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. 5beta,14beta-androstanski derivati, korisni u lijeäśenju bolesti uzrokovanih fibrozom organa

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US521797A (en) * 1894-06-26 Half to john m
BG94957A (bg) * 1990-08-10 1993-12-24 Ciba - Geigy Ag Пиримидинови производни и средство за борба срещу вредители по растенията
US5290780A (en) * 1991-01-30 1994-03-01 American Cyanamid Co. Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
IL100917A0 (en) * 1991-02-16 1992-11-15 Fisons Plc Pyridinone and pyrimidinone derivatives,their preparation and pharmaceutical compositions containing them
IL101860A0 (en) * 1991-05-31 1992-12-30 Ici Plc Heterocyclic derivatives
US5149699A (en) * 1991-10-24 1992-09-22 American Home Products Corporation Substituted pyridopyrimidines useful as antgiotensin II antagonists
TW226375B (fi) * 1991-10-24 1994-07-11 American Home Prod
GB9125842D0 (en) * 1991-12-04 1992-02-05 Ici Plc Heterocyclic derivatives

Also Published As

Publication number Publication date
JPH06321945A (ja) 1994-11-22
NZ260164A (en) 1996-02-27
EP0618207A1 (en) 1994-10-05
LV12261B (en) 1999-09-20
AU669966B2 (en) 1996-06-27
FI941309A0 (fi) 1994-03-21
CA2119692A1 (en) 1994-09-25
LV12261A (lv) 1999-04-20
DE69415706D1 (de) 1999-02-18
PH30373A (en) 1997-04-02
SG47714A1 (en) 1998-04-17
FI108135B (fi) 2001-11-30
DE69415706T2 (de) 1999-05-20
ATE175413T1 (de) 1999-01-15
DK0618207T3 (da) 1999-08-30
HUT66964A (en) 1995-01-30
ES2126061T3 (es) 1999-03-16
AU5799794A (en) 1994-09-29
HU222240B1 (hu) 2003-05-28
EP0863143A1 (en) 1998-09-09
EP0618207B1 (en) 1999-01-07
GR3029879T3 (en) 1999-07-30
BR9401261A (pt) 1994-11-22
HU9400822D0 (en) 1994-06-28
HK1011358A1 (en) 1999-07-09

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