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FI945092L - Epoksimeripihkahappojohdannaiset - Google Patents

Epoksimeripihkahappojohdannaiset Download PDF

Info

Publication number
FI945092L
FI945092L FI945092A FI945092A FI945092L FI 945092 L FI945092 L FI 945092L FI 945092 A FI945092 A FI 945092A FI 945092 A FI945092 A FI 945092A FI 945092 L FI945092 L FI 945092L
Authority
FI
Finland
Prior art keywords
acid derivatives
epoxysuccinic acid
epoxysuccinic
derivatives
acid
Prior art date
Application number
FI945092A
Other languages
English (en)
Swedish (sv)
Other versions
FI945092A0 (fi
FI945092A7 (fi
Inventor
Shigetoshi Tsubotani
Masayuki Takizawa
Mikio Shirasaki
Yukio Fujisawa
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of FI945092A0 publication Critical patent/FI945092A0/fi
Publication of FI945092A7 publication Critical patent/FI945092A7/fi
Publication of FI945092L publication Critical patent/FI945092L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/48Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI945092A 1993-10-29 1994-10-28 Epoksimeripihkahappojohdannaiset FI945092L (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP27283593 1993-10-29
JP27280693 1993-10-29
JP18616594 1994-08-08

Publications (3)

Publication Number Publication Date
FI945092A0 FI945092A0 (fi) 1994-10-28
FI945092A7 FI945092A7 (fi) 1995-04-30
FI945092L true FI945092L (fi) 1995-04-30

Family

ID=27325696

Family Applications (1)

Application Number Title Priority Date Filing Date
FI945092A FI945092L (fi) 1993-10-29 1994-10-28 Epoksimeripihkahappojohdannaiset

Country Status (9)

Country Link
US (1) US5556853A (fi)
EP (1) EP0655447A1 (fi)
KR (1) KR950011429A (fi)
CN (1) CN1112555A (fi)
AU (1) AU7755294A (fi)
CA (1) CA2134627A1 (fi)
FI (1) FI945092L (fi)
HU (1) HUT72319A (fi)
NO (1) NO944121L (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5679708A (en) * 1994-05-31 1997-10-21 Takeda Chemical Industries, Ltd. Epoxysuccinic acid derivatives, their production and use
CA2226740A1 (en) * 1995-07-13 1997-01-30 Mitsuyoshi Azuma Piperazine derivative and its uses
ATE201404T1 (de) * 1995-12-12 2001-06-15 Taiho Pharmaceutical Co Ltd Epoxysuccinamid-derivate oder deren salze und medikamente die diese enthalten
US6110967A (en) * 1997-04-18 2000-08-29 Taiho Pharmaceuticals Co., Ltd. Epoxysuccinamide derivative or salt thereof
AU8997898A (en) * 1997-09-04 1999-03-22 Nippon Chemiphar Co. Ltd. Epoxysuccinamide derivatives
US7132539B2 (en) * 2002-10-23 2006-11-07 The Procter & Gamble Company Melanocortin receptor ligands
US20080227806A1 (en) * 2005-09-28 2008-09-18 American Life Science Pharmaceuticals Novel Drugs for Dementia
JP2010500962A (ja) 2006-06-13 2010-01-14 ザ ボード オブ トラスティーズ オブ ザ リーランド スタンフォード ジュニア ユニバーシティ システインプロテアーゼ類のエポキシド阻害剤
US20100216875A1 (en) * 2006-12-20 2010-08-26 Gregory Hook Methods of treating alzheimer's disease
JPWO2009054454A1 (ja) * 2007-10-24 2011-03-03 国立大学法人 東京医科歯科大学 カテプシン阻害剤を有効成分として含有するToll様受容体のシグナル伝達の調整剤
CN107151236B (zh) * 2016-03-03 2021-04-30 中国人民解放军军事医学科学院毒物药物研究所 一种2,3-环氧丁二酰衍生物及其制备方法和用途
CN113387909B (zh) * 2020-03-13 2023-11-14 中国人民解放军军事科学院军事医学研究院 2,3-环氧丁二酰衍生物的医药用途

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55115878A (en) * 1979-02-27 1980-09-06 Taisho Pharmaceut Co Ltd Epoxysuccinic acid derivative
JPS55153778A (en) * 1979-05-17 1980-11-29 Taisho Pharmaceut Co Ltd Epoxysuccinylamino acid derivative
JPS5772913A (en) * 1980-10-22 1982-05-07 Nippon Chemiphar Co Ltd Remedy for cardiac infraction
JPS57169478A (en) * 1981-04-10 1982-10-19 Nippon Chemiphar Co Ltd Piperazine derivative
JPS5855478A (ja) * 1981-09-25 1983-04-01 Nippon Chemiphar Co Ltd エチレンジアミン誘導体と,心筋梗塞の予防および治療剤
JPS58126879A (ja) * 1982-01-25 1983-07-28 Nippon Chemiphar Co Ltd 光学活性なピペラジン誘導体ならびに心筋梗塞の予防および治療剤
JPS608223A (ja) * 1983-06-28 1985-01-17 Taisho Pharmaceut Co Ltd 抗アレルギ−剤
EP0269311A3 (en) * 1986-11-17 1990-06-06 Merck & Co. Inc. Methods of treating bone diseases by administration of a cysteine proteinase inhibitor
JPH02218610A (ja) * 1989-02-21 1990-08-31 Toyo Jozo Co Ltd 骨疾患の予防および治療剤
JPH02304074A (ja) * 1989-05-18 1990-12-17 Taisho Pharmaceut Co Ltd エポキシコハク酸誘導体

Also Published As

Publication number Publication date
HUT72319A (en) 1996-04-29
CN1112555A (zh) 1995-11-29
HU9403116D0 (en) 1994-12-28
FI945092A0 (fi) 1994-10-28
NO944121D0 (no) 1994-10-28
NO944121L (no) 1995-05-02
CA2134627A1 (en) 1995-04-30
FI945092A7 (fi) 1995-04-30
KR950011429A (ko) 1995-05-15
US5556853A (en) 1996-09-17
AU7755294A (en) 1995-05-18
EP0655447A1 (en) 1995-05-31

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Legal Events

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FD Application lapsed