FI944086L - Antiparasiittiset avermektiini- ja milbemysiinijohdannaiset - Google Patents

Antiparasiittiset avermektiini- ja milbemysiinijohdannaiset Download PDF

Info

Publication number: FI944086L
Authority: FI; Finland
Prior art keywords: milbemycin derivatives; avermectin; antiparasitic; antiparasitic avermectin; milbemycin
Prior art date: 1992-03-07

Application number

FI944086A

Other languages

English (en)

Swedish (sv)

Other versions

FI944086A0 (fi

FI944086A7 (fi

Inventor

Bernard Joseph Banks

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-03-07

Filing date

1993-02-23

Publication date

1994-09-06

1993-02-23 Application filed by Pfizer filed Critical Pfizer

1994-09-06 Publication of FI944086L publication Critical patent/FI944086L/fi

1994-09-06 Publication of FI944086A0 publication Critical patent/FI944086A0/fi

1994-09-06 Publication of FI944086A7 publication Critical patent/FI944086A7/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Molecular Biology (AREA)
Engineering & Computer Science (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Animal Behavior & Ethology (AREA)
Tropical Medicine & Parasitology (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Saccharide Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Fodder In General (AREA)

FI944086A 1992-03-07 1993-02-23 Antiparasiittiset avermektiini- ja milbemysiinijohdannaiset FI944086A7 (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB929205007A GB9205007D0 (en)	1992-03-07	1992-03-07	Antiparasitic agents
PCT/EP1993/000423 WO1993018041A1 (en)	1992-03-07	1993-02-23	Antiparasitic avermectin and milbemycin derivatives

Publications (3)

Publication Number	Publication Date
FI944086L true FI944086L (fi)	1994-09-06
FI944086A0 FI944086A0 (fi)	1994-09-06
FI944086A7 FI944086A7 (fi)	1994-09-06

Family

ID=10711698

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI944086A FI944086A7 (fi)	1992-03-07	1993-02-23	Antiparasiittiset avermektiini- ja milbemysiinijohdannaiset

Country Status (24)

Country	Link
US (1)	US5556868A (fi)
EP (1)	EP0629202B1 (fi)
JP (1)	JP2690195B2 (fi)
KR (1)	KR950700307A (fi)
CN (1)	CN1083818A (fi)
AT (1)	ATE151425T1 (fi)
AU (1)	AU658268B2 (fi)
BR (1)	BR9306037A (fi)
CA (1)	CA2130664C (fi)
DE (1)	DE69309665T2 (fi)
DK (1)	DK0629202T3 (fi)
ES (1)	ES2099422T3 (fi)
FI (1)	FI944086A7 (fi)
GB (1)	GB9205007D0 (fi)
GR (1)	GR3023625T3 (fi)
HR (1)	HRP930226B1 (fi)
HU (1)	HU9402562D0 (fi)
IL (1)	IL104899A0 (fi)
MX (1)	MX9301255A (fi)
NO (1)	NO943289L (fi)
RU (1)	RU94040915A (fi)
WO (1)	WO1993018041A1 (fi)
YU (1)	YU14993A (fi)
ZA (1)	ZA931584B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6426333B1 (en)	1996-09-19	2002-07-30	Merial	Spot-on formulations for combating parasites
GB9312154D0 (en) *	1993-06-12	1993-07-28	Pfizer Ltd	Antiparasitic agents
GB9315108D0 (en) *	1993-07-21	1993-09-01	Pfizer Ltd	Antiparasitic agents
WO1995009863A1 (en) *	1993-10-05	1995-04-13	Pfizer Inc.	Process and antiparasitic intermediates for doramectin
GB9402916D0 (en)	1994-02-16	1994-04-06	Pfizer Ltd	Antiparasitic agents
US20050192319A1 (en) *	1996-09-19	2005-09-01	Albert Boeckh	Spot-on formulations for combating parasites
US6998131B2 (en) *	1996-09-19	2006-02-14	Merial Limited	Spot-on formulations for combating parasites
DK1001962T3 (da) *	1997-07-23	2002-12-16	Pfizer	Fremstilling af avermectinforbindelser
RU2143904C1 (ru) *	1997-11-27	2000-01-10	Пермская государственная медицинская академия	Способ профилактики иксодовых клещевых боррелиозов
US6265571B1 (en)	1999-07-12	2001-07-24	Magellan Laboratories, Inc.	Purification process for anti-parasitic fermentation product
US20040077703A1 (en)	2002-10-02	2004-04-22	Soll Mark D.	Nodulisporic acid derivative spot-on formulations for combating parasites
GB0302547D0 (en) *	2003-02-04	2003-03-12	Syngenta Participations Ag	Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0313937D0 (en) *	2003-06-16	2003-07-23	Syngenta Participations Ag	Avermectin B1 monosaccharide derivatives having an aminosulfonyloxy substituentin the 4'-position
GB0320176D0 (en) *	2003-08-28	2003-10-01	Syngenta Participations Ag	Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
CN102558082B (zh)	2004-03-05	2015-09-30	日产化学工业株式会社	异噁唑啉取代苯甲酰胺化合物的制备中间体
AU2005284422A1 (en) *	2004-09-16	2006-03-23	Bayer Healthcare Ag	Dermally applicable formulations for treating skin diseases in animals
TWI556741B (zh) *	2007-08-17	2016-11-11	英特威特國際股份有限公司	異唑啉組成物及其作為抗寄生蟲藥上的應用
AU2015339096B2 (en)	2014-10-31	2018-08-02	Boehringer Ingelheim Animal Health USA Inc.	Parasiticidal composition comprising fipronil

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS4914624A (fi) *	1972-06-08	1974-02-08
SE434277B (sv) *	1976-04-19	1984-07-16	Merck & Co Inc	Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
US4423209A (en) *	1982-02-26	1983-12-27	Merck & Co., Inc.	Processes for the interconversion of avermectin compounds
DE3519834C2 (de) *	1984-06-05	1993-12-16	American Cyanamid Co	Neue antibiotische Wirkstoffe, Verfahren zu ihrer Gewinnung und ihre Anwendung zur Bekämpfung von Infektionen bei Tieren und Pflanzen
GB2166436B (en) *	1984-09-14	1989-05-24	Glaxo Group Ltd	Antibiotic compounds and their preparation
ES8800986A1 (es) *	1985-07-27	1987-12-01	Pfizer	Un procedimiento para la produccion de un nuevo derivado de avermectina
DE3750495T2 (de) *	1986-07-24	1995-02-23	Beecham Group Plc	Milbemycin-Derivate mit parasitenabtötender Aktivität, ein Verfahren zu ihrer Herstellung und die sie enthaltenden Zusammensetzungen.
ES2058082T3 (es) *	1986-09-12	1994-11-01	American Cyanamid Co	Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249.
GB8721647D0 (en) *	1987-09-15	1987-10-21	Pfizer Ltd	Antiparasitic agents
GB8726730D0 (en) *	1987-11-14	1987-12-16	Pfizer Ltd	Antiparasitic agents
GB8801908D0 (en) *	1988-01-28	1988-02-24	Glaxo Group Ltd	Chemical compounds
GB8807280D0 (en) *	1988-03-26	1988-04-27	Pfizer Ltd	Antiparasitic agents
GB8809232D0 (en) *	1988-04-19	1988-05-25	Pfizer Ltd	Antiparasitic agents
GB8813150D0 (en) *	1988-06-03	1988-07-06	American Cyanamid Co	Chemical compounds
GB8815967D0 (en) *	1988-07-05	1988-08-10	Pfizer Ltd	Antiparasitic agents
GB8917064D0 (en) *	1989-07-26	1989-09-13	Pfizer Ltd	Antiparasitic agent
US5030650A (en) *	1989-09-11	1991-07-09	American Cyanamid Company	13-halo-23-imino derivatives of LL-F28249 compounds and their use as endo- and ectoparasiticidal, insecticidal, acaricidal and nematocidal agents
US5229415A (en) *	1992-03-24	1993-07-20	Merck & Co., Inc.	Alkylthio alkyl avermectins are active antiparasitic agents

1992
- 1992-03-07 GB GB929205007A patent/GB9205007D0/en active Pending
1993
- 1993-02-23 HU HU9402562A patent/HU9402562D0/hu unknown
- 1993-02-23 DK DK93904009.3T patent/DK0629202T3/da active
- 1993-02-23 WO PCT/EP1993/000423 patent/WO1993018041A1/en not_active Ceased
- 1993-02-23 JP JP5515287A patent/JP2690195B2/ja not_active Expired - Fee Related
- 1993-02-23 CA CA002130664A patent/CA2130664C/en not_active Expired - Fee Related
- 1993-02-23 EP EP93904009A patent/EP0629202B1/en not_active Expired - Lifetime
- 1993-02-23 AU AU34987/93A patent/AU658268B2/en not_active Ceased
- 1993-02-23 DE DE69309665T patent/DE69309665T2/de not_active Expired - Fee Related
- 1993-02-23 AT AT93904009T patent/ATE151425T1/de not_active IP Right Cessation
- 1993-02-23 ES ES93904009T patent/ES2099422T3/es not_active Expired - Lifetime
- 1993-02-23 BR BR9306037A patent/BR9306037A/pt not_active Application Discontinuation
- 1993-02-23 FI FI944086A patent/FI944086A7/fi unknown
- 1993-02-23 US US08/302,655 patent/US5556868A/en not_active Expired - Fee Related
- 1993-02-24 HR HR9205007.9A patent/HRP930226B1/xx not_active IP Right Cessation
- 1993-03-01 IL IL104899A patent/IL104899A0/xx unknown
- 1993-03-04 YU YU14993A patent/YU14993A/sh unknown
- 1993-03-05 ZA ZA931584A patent/ZA931584B/xx unknown
- 1993-03-05 MX MX9301255A patent/MX9301255A/es unknown
- 1993-03-06 CN CN93104321A patent/CN1083818A/zh active Pending
1994
- 1994-09-06 NO NO943289A patent/NO943289L/no unknown
- 1994-09-06 RU RU94040915/04A patent/RU94040915A/ru unknown
- 1994-09-06 KR KR1019940703110A patent/KR950700307A/ko not_active Ceased
1997
- 1997-05-30 GR GR970401269T patent/GR3023625T3/el unknown

Also Published As

Publication number	Publication date
CA2130664C (en)	1999-09-14
BR9306037A (pt)	1997-11-18
CN1083818A (zh)	1994-03-16
WO1993018041A1 (en)	1993-09-16
ZA931584B (en)	1994-09-05
HRP930226A2 (en)	1997-06-30
DE69309665T2 (de)	1997-07-24
RU94040915A (ru)	1996-07-20
HU9402562D0 (en)	1994-11-28
KR950700307A (ko)	1995-01-16
GB9205007D0 (en)	1992-04-22
DK0629202T3 (da)	1997-05-05
NO943289D0 (no)	1994-09-06
MX9301255A (es)	1993-09-01
YU14993A (sh)	1996-07-24
GR3023625T3 (en)	1997-08-29
AU3498793A (en)	1993-10-05
JPH07500844A (ja)	1995-01-26
JP2690195B2 (ja)	1997-12-10
FI944086A0 (fi)	1994-09-06
EP0629202A1 (en)	1994-12-21
US5556868A (en)	1996-09-17
EP0629202B1 (en)	1997-04-09
ATE151425T1 (de)	1997-04-15
CA2130664A1 (en)	1993-09-08
IL104899A0 (en)	1993-07-08
AU658268B2 (en)	1995-04-06
ES2099422T3 (es)	1997-05-16
HRP930226B1 (en)	1998-10-31
NO943289L (no)	1994-10-31
DE69309665D1 (de)	1997-05-15
FI944086A7 (fi)	1994-09-06

Publication	Publication Date	Title
FI944086L (fi)	1994-09-06	Antiparasiittiset avermektiini- ja milbemysiinijohdannaiset
FI20000516A7 (fi)	2000-03-07	Bis-indolyylimaleimidijohdannaiset ja niiden valmistus
ATA75293A (de)	1997-11-15	Indolderivate
ZA89538B (en)	1989-09-27	Avermectin derivatives
FI943912L (fi)	1995-06-05	Tienopyrimidiinijohdannaiset, niiden valmistus ja käyttö
ZA899818B (en)	1990-09-26	Avermectin derivatives
FI940167A7 (fi)	1994-03-03	Puriinijohdannaisia
FI940166A0 (fi)	1994-01-13	Uusia adenosiinijohdannaisia
EP0428286A3 (en)	1991-10-23	24- and 25-substituted avermectin and milbemycin derivatives
ZA904211B (en)	1991-03-27	Avermectin derivatives
FI953127L (fi)	1995-08-21	Puriinijohdannaisia
FI933443A7 (fi)	1994-03-02	4-hydroksikumariinijohdannaisia
FI942294A7 (fi)	1994-11-19	Bentsopyraanijohdannaiset ja niiden käyttö
FI922014A7 (fi)	1992-05-05	Nukleosidijohdannaiset
FI944016A0 (fi)	1994-09-01	Makrolidien fluorisokerijohdannaiset
AU615831B2 (en)	1991-10-10	Avermectin derivatives
FI892788A7 (fi)	1989-12-11	Kasvaimen vastainen BU-3420T antibiootti
ZA904207B (en)	1991-03-27	Avermectin derivatives
FI944015L (fi)	1994-09-01	Makrolidien 2-aminosokerijohdannaiset
LV10955A (lv)	1995-12-20	Benzopirana atvasinajumi
GB8909518D0 (en)	1989-06-14	Antiparasitic avermectin derivatives
IE880911L (en)	1988-09-27	Parasiticidal and insecticidal milbemycin derivatives
IL94006A0 (en)	1991-03-10	Antiparasitic formulations comprising avermectin derivatives
IE901978L (en)	1990-12-02	Avermectin derivatives
IE901977L (en)	1990-12-02	Avermectin derivatives