[go: up one dir, main page]

FI933376L - 4-amino-3-acylkinolinderivater och deras anvaendning som inhibitorer avmagsyrasekretion - Google Patents

4-amino-3-acylkinolinderivater och deras anvaendning som inhibitorer avmagsyrasekretion Download PDF

Info

Publication number
FI933376L
FI933376L FI933376A FI933376A FI933376L FI 933376 L FI933376 L FI 933376L FI 933376 A FI933376 A FI 933376A FI 933376 A FI933376 A FI 933376A FI 933376 L FI933376 L FI 933376L
Authority
FI
Finland
Prior art keywords
avmagsyrasekretion
acylquinolinderivater
inhibitorer
amino
och deras
Prior art date
Application number
FI933376A
Other languages
English (en)
Other versions
FI933376A0 (fi
FI933376A7 (fi
Inventor
Robert John Ife
Colin Andrew Leach
Original Assignee
Smithkline Beecham Intercredit
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919101918A external-priority patent/GB9101918D0/en
Priority claimed from GB919101919A external-priority patent/GB9101919D0/en
Application filed by Smithkline Beecham Intercredit filed Critical Smithkline Beecham Intercredit
Publication of FI933376A0 publication Critical patent/FI933376A0/fi
Publication of FI933376A7 publication Critical patent/FI933376A7/fi
Publication of FI933376L publication Critical patent/FI933376L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/42Nitrogen atoms attached in position 4
    • C07D215/44Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicinal Preparation (AREA)
FI933376A 1991-01-29 1992-01-27 4-amino-3-acylkinolinderivater och deras anvaendning som inhibitorer avmagsyrasekretion FI933376L (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB919101918A GB9101918D0 (en) 1991-01-29 1991-01-29 Compound
GB919101919A GB9101919D0 (en) 1991-01-29 1991-01-29 Compound
PCT/EP1992/000200 WO1992012969A1 (en) 1991-01-29 1992-01-27 Salts of a 4-amino-3-acyl quinoline derivative and their use as inhibitors of gastric acid secretion

Publications (3)

Publication Number Publication Date
FI933376A0 FI933376A0 (fi) 1993-07-28
FI933376A7 FI933376A7 (fi) 1993-07-28
FI933376L true FI933376L (fi) 1993-07-28

Family

ID=26298350

Family Applications (1)

Application Number Title Priority Date Filing Date
FI933376A FI933376L (fi) 1991-01-29 1992-01-27 4-amino-3-acylkinolinderivater och deras anvaendning som inhibitorer avmagsyrasekretion

Country Status (18)

Country Link
EP (1) EP0569396A1 (fi)
JP (1) JPH06504541A (fi)
CN (1) CN1064268A (fi)
AP (1) AP337A (fi)
AU (1) AU652028B2 (fi)
CA (1) CA2099117A1 (fi)
CZ (1) CZ153293A3 (fi)
FI (1) FI933376L (fi)
HU (1) HUT67609A (fi)
IE (1) IE920267A1 (fi)
IL (1) IL100791A0 (fi)
MA (1) MA22401A1 (fi)
MX (1) MX9200338A (fi)
NO (1) NO932722D0 (fi)
NZ (1) NZ241408A (fi)
PT (1) PT100056A (fi)
SK (1) SK70993A3 (fi)
WO (1) WO1992012969A1 (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9126438D0 (en) * 1991-12-12 1992-02-12 Smithkline Beecham Intercredit New quinoline derivatives
IS4164A (is) * 1993-06-11 1994-12-12 Ab Astra Efnasambönd sem hindra flæði magasýru
US5556863A (en) * 1993-06-11 1996-09-17 Astra Aktiebolag Compound for gastric acid secretion inhibition
USRE43932E1 (en) 1997-07-18 2013-01-15 Novartis Ag Crystal modification of a N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
US6852739B1 (en) 1999-02-26 2005-02-08 Nitromed Inc. Methods using proton pump inhibitors and nitric oxide donors
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
US20050020637A1 (en) * 2001-11-19 2005-01-27 Wolfgang-Alexander Simon Agents for the treatment of airway disorders
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
AU2003254282A1 (en) 2002-08-01 2004-02-23 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
US20080280944A1 (en) 2003-11-03 2008-11-13 Paula Fernstrom Imidazo[1,2-A]Pyridine Derivatives For The Treatment Of Silent Gastro-Esophageal Reflux

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8804444D0 (en) * 1988-02-25 1988-03-23 Smithkline Beckman Intercredit Compounds

Also Published As

Publication number Publication date
EP0569396A1 (en) 1993-11-18
SK70993A3 (en) 1994-01-12
IL100791A0 (en) 1992-09-06
IE920267A1 (en) 1992-07-29
AU1179992A (en) 1992-08-27
NO932722L (no) 1993-07-28
NO932722D0 (no) 1993-07-28
CN1064268A (zh) 1992-09-09
WO1992012969A1 (en) 1992-08-06
CZ153293A3 (en) 1993-12-15
HUT67609A (en) 1995-04-28
AU652028B2 (en) 1994-08-11
FI933376A0 (fi) 1993-07-28
MA22401A1 (fr) 1992-10-01
PT100056A (pt) 1993-03-31
CA2099117A1 (en) 1992-07-30
JPH06504541A (ja) 1994-05-26
NZ241408A (en) 1994-05-26
AP337A (en) 1994-04-08
AP9200352A0 (en) 1992-01-31
FI933376A7 (fi) 1993-07-28
HU9302201D0 (en) 1993-10-28
MX9200338A (es) 1992-12-01

Similar Documents

Publication Publication Date Title
FI921951A7 (fi) Foerfarande foer framstaellning av polycykliska aminfoereningar och enantiomerer daerav anvaendbara som laekemedel
FI921952L (fi) Foerfarande foer framstaellning av dialkylenpiperidinofoereningar och enantiomerer daerav anvaendbara som laekemedel
FI921950L (fi) Foerfarande foer framstaellning av n-alkylenpiperidinofoereningar och enantiomerer daerav anvaendbara som laekemedel
FI933199L (fi) Doseringsanordning som aer laemplig foer baode kontinuerlig och tillfaelliganvaendning
FI924091A7 (fi) Autoriseringsprotokoll som foersiktighetshjaelpmedel
FI933167A0 (fi) N-alkylkinuklidiniumsalter som substans-p antagonister
FI921105L (fi) Segmentpolyteramider och deras syntesprocess
FI921556L (fi) Plasttillslutning som visar otillboerlig anvaendning
FI921182L (fi) Velangummi som snabbt hydratiseras
FI923558A7 (fi) Tetrahydroindazol-, tetrahydrocyklopentapyrazol- och hexahydrocykloheptapyrazolfoereningar och deras anvaendning som inhibitorer av hmg-coa-reduktas
FI912760A7 (fi) Skivfilter och filterelement foer skivfilter
FI920540A7 (fi) Foerfarande foer framstaellning av en armerad fiberkonstruktion som skalllamineras och motsvarande armerad fiberkonstruktion
FI923185L (fi) Foerfarande och anordning foer framstaellning av fogloesa band- och traodoeglor och deras anvaendning som kapverktyg i band- och traodsaogar
FI923756L (fi) Polyolefinkompositioner som omfattar glycerolmonoestrar av c20-24-fettsyror och daerav framstaellda skumprodukter
FI921818L (fi) Hopknippningsanordning och foerfarande
FI923382A7 (fi) Laosanordning som omfattar nyckel och laoscylinder
FI935944L (fi) Pyratsolopyrimidin- samt pyrimidinylbisfosfonestrar som anti- inflammatorer
FI925330L (fi) Substituerade fenylfenoler som leukotrienantagonister
FI920342L (fi) Komplex som innehaoller koaguleringsfaktor ix och foerfarande foer framstaellning daerav.
FI924463L (fi) Garulaer konstgoedningssammansaettning som frigoers laongsamt och foerfarande foer framstaellning daerav
FI921974A7 (fi) Lageranlaeggning och undervattensdrivdraftsenhet som innehaoller den
FI921741L (fi) En katalyt och belaeggningskomposition innehaollande densamma
FI924712A7 (fi) Kemiska kompositioner och anvaendning daerav som braensletillsatsaemnen
FI933376L (fi) 4-amino-3-acylkinolinderivater och deras anvaendning som inhibitorer avmagsyrasekretion
FI931039L (fi) Foerbaettrade smoerjmedelskompositioner och i dessa anvaendbara tillsatsaemnen