FI932145A7 - Uudet b-karboliinijohdannaiset, niiden valmistus ja käyttö lääkeaineis sa - Google Patents

Uudet b-karboliinijohdannaiset, niiden valmistus ja käyttö lääkeaineis sa Download PDF

Info

Publication number: FI932145A7
Authority: FI; Finland
Prior art keywords: pharmaceuticals; preparation; new; carboline derivatives; carboline
Prior art date: 1991-09-13

Application number

FI932145A

Other languages

English (en)

Swedish (sv)

Other versions

FI932145L (fi

FI932145A0 (fi

Inventor

Dieter Rahtz

Herbert Hans Schneider

Andreas Huth

Dieter Seidelmann

Ralph Schmiechen

Lecboslaw Turski

Margit Hillmann

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-09-13

Filing date

1992-09-11

Publication date

1993-05-12

1992-09-11 Application filed by Schering Ag filed Critical Schering Ag

1993-05-12 Publication of FI932145A7 publication Critical patent/FI932145A7/fi

1993-05-12 Publication of FI932145L publication Critical patent/FI932145L/fi

1993-05-12 Publication of FI932145A0 publication Critical patent/FI932145A0/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

FI932145A 1991-09-13 1992-09-11 Nya b-karbolinderivat, deras framstaellning och anvaendning i laekemedel FI932145A0 (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE4130933A DE4130933A1 (de)	1991-09-13	1991-09-13	Neue (beta)-carbolinderivate, deren herstellung und verwendung in arzneimitteln
PCT/DE1992/000786 WO1993006100A1 (de)	1991-09-13	1992-09-11	NEUE β-CARBOLINDERIVATE, DEREN HERSTELLUNG UND VERWENDUNG IN ARZNEIMITTELN

Publications (3)

Publication Number	Publication Date
FI932145A7 true FI932145A7 (fi)	1993-05-12
FI932145L FI932145L (fi)	1993-05-12
FI932145A0 FI932145A0 (fi)	1993-05-12

Family

ID=6440817

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI932145A FI932145A0 (fi)	1991-09-13	1992-09-11	Nya b-karbolinderivat, deras framstaellning och anvaendning i laekemedel

Country Status (17)

Country	Link
US (1)	US5506234A (fi)
EP (1)	EP0557497A1 (fi)
JP (1)	JPH06502871A (fi)
KR (1)	KR930703313A (fi)
CN (1)	CN1033391C (fi)
AU (1)	AU655503B2 (fi)
CA (1)	CA2096138A1 (fi)
CZ (1)	CZ72593A3 (fi)
DE (1)	DE4130933A1 (fi)
FI (1)	FI932145A0 (fi)
HU (1)	HUT64343A (fi)
IL (1)	IL103151A0 (fi)
MX (1)	MX9205164A (fi)
NZ (1)	NZ244328A (fi)
PT (1)	PT100860A (fi)
WO (1)	WO1993006100A1 (fi)
ZA (1)	ZA926969B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4330175A1 (de) *	1993-08-31	1995-03-02	Schering Ag	Alkoxy-substituierte beta-Carboline
DE19502753A1 (de) *	1995-01-23	1996-07-25	Schering Ag	Neue 9H-Pyrido[3,4-b]indol-Derivate
DE19514524A1 (de) *	1995-04-12	1996-10-17	Schering Ag	Anellierte beta-Carboline
EA008244B1 (ru) *	2002-05-03	2007-04-27	Янссен Фармацевтика Н.В.	Полимерные микроэмульсии
US7504401B2 (en)	2003-08-29	2009-03-17	Locus Pharmaceuticals, Inc.	Anti-cancer agents and uses thereof
BRPI0907122B8 (pt)	2008-01-11	2021-05-25	Albany Molecular Res Inc	compostos de piridoindóis (1-azinona) substituídos, composição farmacêutica compreendendo os referidos compostos, e usos dos mesmos
US8618299B2 (en) *	2009-07-01	2013-12-31	Albany Molecular Research, Inc.	Azinone-substituted azapolycycle MCH-1 antagonists, methods of making, and use thereof
WO2011003007A1 (en) *	2009-07-01	2011-01-06	Albany Molecular Research, Inc.	Azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine mch-1 antagonists, methods of making, and use thereof
US9073925B2 (en) *	2009-07-01	2015-07-07	Albany Molecular Research, Inc.	Azinone-substituted azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine MCH-1 antagonists, methods of making, and use thereof
US8637501B2 (en) *	2009-07-01	2014-01-28	Albany Molecular Research, Inc.	Azinone-substituted azepino[b]indole and pyrido-pyrrolo-azepine MCH-1 antagonists, methods of making, and use thereof
WO2011158108A2 (en)	2010-06-16	2011-12-22	Purdue Pharma L.P.	Aryl substituted indoles and the use thereof
EP2455378A1 (en)	2010-11-03	2012-05-23	Philip Morris Products S.A.	Carbazole and carboline derivatives, and preparation and therapeutic applications thereof
WO2012088124A2 (en)	2010-12-21	2012-06-28	Albany Molecular Research, Inc.	Tetrahydro-azacarboline mch-1 antagonists, methods of making, and uses thereof
US8697700B2 (en)	2010-12-21	2014-04-15	Albany Molecular Research, Inc.	Piperazinone-substituted tetrahydro-carboline MCH-1 antagonists, methods of making, and uses thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS57123180A (en) *	1980-12-17	1982-07-31	Schering Ag	3-substituted beta-carboline, manufacture and psychotropic drug containing same
DE3335323A1 (de) *	1983-09-27	1985-04-04	Schering AG, 1000 Berlin und 4709 Bergkamen	Substituierte ss-carboline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DK240084D0 (da) *	1984-05-15	1984-05-15	Ferrosan As	New beta-carboline-3-oxadiazolyl derivatives
DE3504045A1 (de) *	1985-02-04	1986-08-07	Schering AG, 1000 Berlin und 4709 Bergkamen	Verfahren zur herstellung von ss-carbolinen durch dehydrierung
DE3545776A1 (de) *	1985-12-20	1987-06-25	Schering Ag	5-aminoalkyl-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
DE3608089A1 (de) *	1986-03-08	1987-09-10	Schering Ag	Heteroaryl-oxy-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
IL87563A (en) *	1987-08-28	1993-08-18	Schering Ag	Isoxazole-b-carboline derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
DE3925507A1 (de) *	1989-07-28	1991-01-31	Schering Ag	14,17(alpha)-etheno- und ethanoestratriene, verfahren zur herstellung dieser verbindungen, sowie ihre verwendung zur herstellung von arzneimitteln
DE3943225A1 (de) *	1989-12-23	1991-06-27	Schering Ag	Neue ss-carboline, verfahren zu deren herstellung und deren verwendung in arzneimitteln

1991
- 1991-09-13 DE DE4130933A patent/DE4130933A1/de not_active Withdrawn
1992
- 1992-09-10 MX MX9205164A patent/MX9205164A/es not_active Application Discontinuation
- 1992-09-11 ZA ZA926969A patent/ZA926969B/xx unknown
- 1992-09-11 EP EP92919414A patent/EP0557497A1/de not_active Withdrawn
- 1992-09-11 PT PT100860A patent/PT100860A/pt not_active Application Discontinuation
- 1992-09-11 WO PCT/DE1992/000786 patent/WO1993006100A1/de not_active Ceased
- 1992-09-11 HU HU9301379A patent/HUT64343A/hu unknown
- 1992-09-11 JP JP5505694A patent/JPH06502871A/ja active Pending
- 1992-09-11 CA CA002096138A patent/CA2096138A1/en not_active Abandoned
- 1992-09-11 CZ CS93725A patent/CZ72593A3/cs unknown
- 1992-09-11 KR KR1019930701425A patent/KR930703313A/ko not_active Withdrawn
- 1992-09-11 FI FI932145A patent/FI932145A0/fi not_active Application Discontinuation
- 1992-09-11 AU AU25578/92A patent/AU655503B2/en not_active Ceased
- 1992-09-12 CN CN92110560A patent/CN1033391C/zh not_active Expired - Fee Related
- 1992-09-13 IL IL103151A patent/IL103151A0/xx unknown
- 1992-09-14 NZ NZ244328A patent/NZ244328A/en unknown
- 1992-09-14 US US07/943,177 patent/US5506234A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO1993006100A1 (de)	1993-04-01
IL103151A0 (en)	1993-02-21
EP0557497A1 (de)	1993-09-01
AU2557892A (en)	1993-04-27
CZ72593A3 (en)	1994-01-19
KR930703313A (ko)	1993-11-29
JPH06502871A (ja)	1994-03-31
HU9301379D0 (en)	1993-09-28
US5506234A (en)	1996-04-09
CN1070403A (zh)	1993-03-31
PT100860A (pt)	1993-11-30
ZA926969B (en)	1993-03-17
FI932145L (fi)	1993-05-12
MX9205164A (es)	1993-03-01
AU655503B2 (en)	1994-12-22
CN1033391C (zh)	1996-11-27
CA2096138A1 (en)	1993-03-14
NZ244328A (en)	1995-02-24
HUT64343A (en)	1993-12-28
FI932145A0 (fi)	1993-05-12
DE4130933A1 (de)	1993-03-18

Publication	Publication Date	Title
FI934220A7 (fi)	1994-03-29	Piperidiinijohdannaisia, niiden valmistus ja niiden käyttö terapiassa
FI955248A7 (fi)	1995-11-02	1-Bifenyylimetyyli-imitdatsolin johdannaiset, niiden valmistus ja terapeuttinen käyttö
FI955140L (fi)	1995-10-27	Uusia kinoksaliinidionijohdannaisia, niiden valmistus ja käyttö lääkkeissä
FI935074A7 (fi)	1993-11-16	Uusia tiopyranopyrrolijohdannaisia ja niiden valmistus
FI935897A7 (fi)	1994-06-30	Pyridopyrimidiinijohdannaiset, niiden valmistus ja käyttö
FI944600A0 (fi)	1994-10-03	Imidatsol-4-yylipiperidiinijohdannaisia, niiden valmistus ja niiden käyttö terapiassa
FI944821L (fi)	1995-04-16	Galantamiinijohdannaisia, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineissa
FI940696A7 (fi)	1994-02-15	Uudet pyratsiinijohdannaiset, niiden valmistus ja käyttö
FI921459A7 (fi)	1992-10-04	Piperidiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI944822L (fi)	1995-04-16	Galantamiinijohdannaisia, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineissa
FI914611A7 (fi)	1992-04-03	2-aminopyrimidiini-4-karboksamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI932145A7 (fi)	1993-05-12	Uudet b-karboliinijohdannaiset, niiden valmistus ja käyttö lääkeaineis sa
FI944823L (fi)	1995-04-16	Galantamiinijohdannaisia, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineissa
FI940889A7 (fi)	1994-02-25	Uudet isatsiinioksiimijohdannaiset, niiden valmistus ja käyttö
FI911615A7 (fi)	1991-10-07	Uusia 4-kinolyyli-dihydropyridiinejä, menetelmiä niiden valmistamiseksi ja niiden käyttö lääkeaineissa
FI922982A7 (fi)	1992-12-28	2-aminopyrimidiini-4-karboksamidijohdannaisia, niiden valmistus ja niiden terapeuttinen käyttö
FI934680A7 (fi)	1993-10-22	Aryylimorfoliini, valmistus ja käyttö
FI933544A7 (fi)	1993-08-11	Tiadiatsiinikarboksamidijohdannaiset, menetelmät niiden valmistamiseks i ja lääkkeet
FI930716A7 (fi)	1993-08-21	Uusia aryylikarbonyyliaminoalkyylidihydro-oksopyridiinejä, niiden valmistus ja käyttö
FI955679A0 (fi)	1995-11-24	Piperidiinijohdannaisia, niiden valmistus ja käyttö
FI934221A7 (fi)	1994-03-29	Piperidiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI930293A7 (fi)	1993-01-25	Uusia heteroaryylioksi-b-karboliineja, niiden valmistus ja käyttö lääk keissä
FI941958A7 (fi)	1994-04-28	2-heterosyklinenetyyliamiinijohdannaiset ja niiden käyttö lääkkeinä
FI920663A7 (fi)	1992-08-16	Polyhydroksisyklopentaanin johdannaiset, niiden valmistus ja terapeuttinen käyttö
FI921814A7 (fi)	1992-10-25	2-aminopyrimidiini-4-karboksiamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö

Legal Events

Date	Code	Title	Description
1998-03-31	FD	Application lapsed