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FI921814L - 2-aminopyrimidin-4-karboxiamidderivat, deras framstaellning och terapeutisk anvaendning av dem - Google Patents

2-aminopyrimidin-4-karboxiamidderivat, deras framstaellning och terapeutisk anvaendning av dem Download PDF

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Publication number
FI921814L
FI921814L FI921814A FI921814A FI921814L FI 921814 L FI921814 L FI 921814L FI 921814 A FI921814 A FI 921814A FI 921814 A FI921814 A FI 921814A FI 921814 L FI921814 L FI 921814L
Authority
FI
Finland
Prior art keywords
anvaendning
aminopyrimidin
dem
therapeutic
deras framstaellning
Prior art date
Application number
FI921814A
Other languages
English (en)
Other versions
FI921814A7 (fi
FI921814A0 (fi
Inventor
Pascal George
Philippe Monoury
Michel Mangane
Jean-Pierre Merly
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI921814A0 publication Critical patent/FI921814A0/fi
Publication of FI921814L publication Critical patent/FI921814L/fi
Publication of FI921814A7 publication Critical patent/FI921814A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI921814A 1991-04-24 1992-04-23 2-aminopyrimidiini-4-karboksiamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö FI921814A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9105043A FR2675799B1 (fr) 1991-04-24 1991-04-24 Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Publications (3)

Publication Number Publication Date
FI921814A0 FI921814A0 (fi) 1992-04-23
FI921814L true FI921814L (fi) 1992-10-25
FI921814A7 FI921814A7 (fi) 1992-10-25

Family

ID=9412198

Family Applications (1)

Application Number Title Priority Date Filing Date
FI921814A FI921814A7 (fi) 1991-04-24 1992-04-23 2-aminopyrimidiini-4-karboksiamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö

Country Status (18)

Country Link
US (1) US5229392A (fi)
EP (1) EP0511072A1 (fi)
JP (1) JPH05117243A (fi)
KR (1) KR920019760A (fi)
CN (1) CN1066066A (fi)
AU (1) AU1507992A (fi)
CA (1) CA2066960A1 (fi)
CS (1) CS124492A3 (fi)
FI (1) FI921814A7 (fi)
FR (1) FR2675799B1 (fi)
HU (1) HUT61002A (fi)
IE (1) IE921319A1 (fi)
IL (1) IL101617A0 (fi)
MX (1) MX9201866A (fi)
NO (1) NO921563L (fi)
NZ (1) NZ242464A (fi)
PL (1) PL294309A1 (fi)
ZA (1) ZA922952B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2699171B1 (fr) * 1992-12-14 1995-02-03 Synthelabo Dérivés de 2-amino-N[[[4-aminocarbonyl) pyrimidin-2-yl]amino]alkyl]pyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique.
ATE123025T1 (de) * 1992-07-03 1995-06-15 Synthelabo 2-amino-n-(((4-(aminocarbonyl)pyrimidin-2- yl>amino>alkyl>-pyrimidin-4- carbonsäureamidderivate, ihre herstellung und ihre anwendung in der therapeutica.
FR2697253B1 (fr) * 1992-10-22 1994-12-02 Synthelabo Dérivés de 2-aminopyrimidine-4-carboxamide, leur préparation et leur application en thérapeutique.
ES2074946B1 (es) * 1993-07-19 1996-06-16 Ferrer Int Nuevos compuestos derivados de la 1,2-etanodiamina-n,n,n',n'-tetrasustituida.
WO1995005366A1 (en) * 1993-08-19 1995-02-23 Janssen Pharmaceutica N.V. Vasoconstrictive substituted aryloxyalkyl diamines
FR2724383B1 (fr) * 1994-09-13 1996-10-18 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique
MXPA00010805A (es) * 1998-05-06 2002-05-08 Univ Duke Metodo para el tratamiento de sindromes de la vejiga y del tracto urinario inferior.
JP7186170B2 (ja) * 2016-10-25 2022-12-08 アリゾナ ボード オブ リージェンツ オン ビハーフ オブ アリゾナ ステート ユニバーシティ 無溶媒イオン性液体エポキシ樹脂
JP7508467B2 (ja) 2019-02-18 2024-07-01 アリゾナ ボード オブ リージェンツ オン ビハーフ オブ アリゾナ ステート ユニバーシティ 無溶剤イオン性液体エポキシ樹脂

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1191845B (it) * 1986-01-20 1988-03-23 Dompe Farmaceutici Spa Alchiloli derivati farmacologicamente attivi

Also Published As

Publication number Publication date
CS124492A3 (en) 1992-11-18
MX9201866A (es) 1992-10-01
KR920019760A (ko) 1992-11-19
CA2066960A1 (en) 1992-10-25
HUT61002A (en) 1992-11-30
US5229392A (en) 1993-07-20
ZA922952B (en) 1993-01-27
FR2675799A1 (fr) 1992-10-30
NO921563L (no) 1992-10-26
CN1066066A (zh) 1992-11-11
JPH05117243A (ja) 1993-05-14
NO921563D0 (no) 1992-04-23
IL101617A0 (en) 1992-12-30
HU9201358D0 (en) 1992-07-28
AU1507992A (en) 1992-10-29
FI921814A7 (fi) 1992-10-25
EP0511072A1 (fr) 1992-10-28
NZ242464A (en) 1993-05-26
IE921319A1 (en) 1992-11-04
FR2675799B1 (fr) 1993-12-24
FI921814A0 (fi) 1992-04-23
PL294309A1 (en) 1992-11-02

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