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FI921562A7 - Gem-difosfonihapot, menetelmä niiden valmistamiseksi ja farmaseuttiset koostumukset, jotka sisältävät niitä - Google Patents

Gem-difosfonihapot, menetelmä niiden valmistamiseksi ja farmaseuttiset koostumukset, jotka sisältävät niitä Download PDF

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Publication number
FI921562A7
FI921562A7 FI921562A FI921562A FI921562A7 FI 921562 A7 FI921562 A7 FI 921562A7 FI 921562 A FI921562 A FI 921562A FI 921562 A FI921562 A FI 921562A FI 921562 A7 FI921562 A7 FI 921562A7
Authority
FI
Finland
Prior art keywords
gem
preparation
pharmaceutical compositions
compositions containing
diphosphonic acids
Prior art date
Application number
FI921562A
Other languages
English (en)
Swedish (sv)
Other versions
FI921562A0 (fi
FI921562L (fi
Inventor
Sergio Tognella
Silvano Spinelli
Valeria Livi
Ernesto Menta
Original Assignee
Boehringer Mannheim Italia S P A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Italia S P A filed Critical Boehringer Mannheim Italia S P A
Publication of FI921562A0 publication Critical patent/FI921562A0/fi
Publication of FI921562L publication Critical patent/FI921562L/fi
Publication of FI921562A7 publication Critical patent/FI921562A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40Esters thereof
    • C07F9/4003Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4025Esters of poly(thio)phosphonic acids
    • C07F9/405Esters of poly(thio)phosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839Polyphosphonic acids
    • C07F9/3873Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/564Three-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Materials For Medical Uses (AREA)
FI921562A 1989-10-12 1990-10-11 Gem-difosfonihapot, menetelmä niiden valmistamiseksi ja farmaseuttiset koostumukset, jotka sisältävät niitä FI921562A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT22004A IT1241674B (it) 1989-10-12 1989-10-12 Acidi gem-difosfonici, un processo per la loro preparazione e composizioni farmaceutiche che li contengono.
PCT/EP1990/001710 WO1991005791A1 (en) 1989-10-12 1990-10-11 Gem-diphosphonic acids, a process for the preparation thereof and pharmaceutical compositions containing them

Publications (3)

Publication Number Publication Date
FI921562A0 FI921562A0 (fi) 1992-04-08
FI921562L FI921562L (fi) 1992-04-08
FI921562A7 true FI921562A7 (fi) 1992-04-08

Family

ID=11190055

Family Applications (1)

Application Number Title Priority Date Filing Date
FI921562A FI921562A7 (fi) 1989-10-12 1990-10-11 Gem-difosfonihapot, menetelmä niiden valmistamiseksi ja farmaseuttiset koostumukset, jotka sisältävät niitä

Country Status (14)

Country Link
US (1) US5300671A (fi)
EP (1) EP0593437B1 (fi)
JP (1) JPH05500949A (fi)
KR (1) KR927003610A (fi)
AT (1) ATE137757T1 (fi)
AU (1) AU639495B2 (fi)
CA (1) CA2067191A1 (fi)
DE (1) DE69026964T2 (fi)
ES (1) ES2090143T3 (fi)
FI (1) FI921562A7 (fi)
HU (1) HUT61027A (fi)
IT (1) IT1241674B (fi)
WO (1) WO1991005791A1 (fi)
ZA (1) ZA908131B (fi)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5183815A (en) * 1991-01-22 1993-02-02 Merck & Co., Inc. Bone acting agents
EP0496520A1 (en) * 1991-01-22 1992-07-29 Merck & Co. Inc. Novel bone acting agents
IT1246777B (it) * 1991-04-12 1994-11-26 Boehringer Mannheim Italia Aminoacil derivati di acidi gem-difosfonici,un processo per la loro preparazione e composizioni farmaceutiche che li contengono
IT1246778B (it) * 1991-04-12 1994-11-26 Boehringer Mannheim Italia Nitrosocarbamoil derivati di acidi gem-difosfonici, un processo per la loro preparazione e composizioni farmaceutiche che li contengono
IT1284070B1 (it) * 1996-06-26 1998-05-08 Boehringer Mannheim Italia Derivati di carbossi gem-difosfonati ad attivita' antitumorale, un processo per la loro preparazione e composizioni farmaceutiche che
IT1290444B1 (it) * 1997-03-27 1998-12-03 Boehringer Mannheim Italia Coniugati di bis-fosfonati con funzionalita' alchilanti aventi attivita' antitumorale
US6828312B2 (en) 1998-09-25 2004-12-07 Sunol Molecular Corporation Pharmaceutically active compounds and methods of use thereof
WO2005090370A1 (en) * 2004-02-05 2005-09-29 The Regents Of The University Of California Pharmacologically active agents containing esterified phosphonates and methods for use thereof
US8642577B2 (en) 2005-04-08 2014-02-04 Chimerix, Inc. Compounds, compositions and methods for the treatment of poxvirus infections
US20070003608A1 (en) * 2005-04-08 2007-01-04 Almond Merrick R Compounds, compositions and methods for the treatment of viral infections and other medical disorders
JP5562255B2 (ja) * 2008-01-25 2014-07-30 キメリクス,インコーポレイテッド ウイルス感染を治療する方法
US8614200B2 (en) 2009-07-21 2013-12-24 Chimerix, Inc. Compounds, compositions and methods for treating ocular conditions
EP2462152A4 (en) 2009-08-03 2013-02-13 Chimerix Inc COMPOSITION AND METHOD FOR THE TREATMENT OF VIRUS INFECTIONS AND TEMPORED VIRUSES
ES2629165T3 (es) 2010-02-12 2017-08-07 Chimerix, Inc. Métodos de tratamiento de una infección vírica
WO2011139709A2 (en) 2010-04-26 2011-11-10 Chimerix, Inc. Methods of treating retroviral infections and related dosage regimes
US11246905B2 (en) 2016-08-15 2022-02-15 President And Fellows Of Harvard College Treating infections using IdsD from Proteus mirabilis

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3425812A1 (de) * 1984-07-13 1986-01-16 Deutsches Krebsforschungszentrum, 6900 Heidelberg Neue 1-hydroxy-1,1-diphosphonsaeureverbindungen, verfahren zu ihrer herstellung und pharmakologische zubereitungen, insbesondere zur behandlung von knochentumoren
DE3512536A1 (de) * 1985-04-06 1986-10-16 Boehringer Mannheim Gmbh, 6800 Mannheim Neue diphosphonsaeure-derivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
JPH05500949A (ja) 1993-02-25
WO1991005791A1 (en) 1991-05-02
IT1241674B (it) 1994-01-27
EP0593437B1 (en) 1996-05-08
FI921562A0 (fi) 1992-04-08
CA2067191A1 (en) 1991-04-13
US5300671A (en) 1994-04-05
AU6510890A (en) 1991-05-16
HU9201215D0 (en) 1992-07-28
IT8922004A0 (it) 1989-10-12
EP0593437A1 (en) 1994-04-27
ATE137757T1 (de) 1996-05-15
DE69026964D1 (de) 1996-06-13
IT8922004A1 (it) 1991-04-12
AU639495B2 (en) 1993-07-29
KR927003610A (ko) 1992-12-18
ES2090143T3 (es) 1996-10-16
HUT61027A (en) 1992-11-30
FI921562L (fi) 1992-04-08
DE69026964T2 (de) 1996-10-24
ZA908131B (en) 1991-07-31

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