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FI92687B - Förfarande för framställning av antracyklinoner - Google Patents

Förfarande för framställning av antracyklinoner Download PDF

Info

Publication number
FI92687B
FI92687B FI914053A FI914053A FI92687B FI 92687 B FI92687 B FI 92687B FI 914053 A FI914053 A FI 914053A FI 914053 A FI914053 A FI 914053A FI 92687 B FI92687 B FI 92687B
Authority
FI
Finland
Prior art keywords
formula
group
compound
daunomycinone
vii
Prior art date
Application number
FI914053A
Other languages
English (en)
Finnish (fi)
Other versions
FI92687C (sv
FI914053A0 (sv
Inventor
Franco Francalanci
Walter Cabri
Ilaria Candiani
Bernardinis Silvia De
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of FI914053A0 publication Critical patent/FI914053A0/sv
Publication of FI92687B publication Critical patent/FI92687B/sv
Application granted granted Critical
Publication of FI92687C publication Critical patent/FI92687C/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C50/00Quinones
    • C07C50/38Quinones containing —CHO or non—quinoid keto groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C46/00Preparation of quinones
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI914053A 1989-03-02 1991-08-28 Förfarande för framställning av antracyklinoner FI92687C (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8904794 1989-03-02
GB898904794A GB8904794D0 (en) 1989-03-02 1989-03-02 Process for preparing anthracyclinones
PCT/EP1990/000334 WO1990009974A1 (en) 1989-03-02 1990-02-28 Process for preparing anthracyclinones
EP9000334 1990-02-28

Publications (3)

Publication Number Publication Date
FI914053A0 FI914053A0 (sv) 1991-08-28
FI92687B true FI92687B (sv) 1994-09-15
FI92687C FI92687C (sv) 1994-12-27

Family

ID=10652605

Family Applications (1)

Application Number Title Priority Date Filing Date
FI914053A FI92687C (sv) 1989-03-02 1991-08-28 Förfarande för framställning av antracyklinoner

Country Status (26)

Country Link
US (1) US5180758A (sv)
EP (1) EP0385354B1 (sv)
JP (1) JP2717023B2 (sv)
KR (1) KR0171047B1 (sv)
CN (1) CN1028518C (sv)
AT (1) ATE88173T1 (sv)
AU (1) AU636134B2 (sv)
CA (1) CA2047748C (sv)
CZ (1) CZ278804B6 (sv)
DE (1) DE69001312T2 (sv)
DK (1) DK0385354T3 (sv)
ES (1) ES2055189T3 (sv)
FI (1) FI92687C (sv)
GB (1) GB8904794D0 (sv)
HU (1) HU207705B (sv)
IE (1) IE63571B1 (sv)
IL (1) IL93559A (sv)
MY (1) MY105260A (sv)
NO (1) NO174546C (sv)
NZ (1) NZ232681A (sv)
PT (1) PT93317B (sv)
RU (1) RU2077526C1 (sv)
SK (1) SK278225B6 (sv)
WO (1) WO1990009974A1 (sv)
YU (1) YU47556B (sv)
ZA (1) ZA901542B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPQ319799A0 (en) * 1999-10-01 1999-10-28 Institute Of Drug Technology Australia Limited Chemical methods
JP4688315B2 (ja) * 2001-02-28 2011-05-25 メルシャン株式会社 4−デメトキシダウノマイシノンの製造
US7053191B2 (en) * 2003-05-21 2006-05-30 Solux Corporation Method of preparing 4-R-substituted 4-demethoxydaunorubicin
WO2006024016A2 (en) * 2004-08-23 2006-03-02 Sicor, Inc. Synthesis of idarubin aglycone
US8357785B2 (en) * 2008-01-08 2013-01-22 Solux Corporation Method of aralkylation of 4′-hydroxyl group of anthracylins
US8846882B2 (en) 2011-04-29 2014-09-30 Synbias Pharma Ag Method of producing 4-demethoxydaunorubicin

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ224252A (en) * 1987-04-21 1991-09-25 Erba Carlo Spa An anthracycline glycoside and its preparation
GB8808475D0 (en) * 1988-04-11 1988-05-11 Erba Carlo Spa Process for preparing 4-demethoxydauno-mycinone
GB8818167D0 (en) * 1988-07-29 1988-09-01 Erba Carlo Spa Novel 4-substituted anthracyclinones & process for their preparation

Also Published As

Publication number Publication date
KR900014286A (ko) 1990-10-23
RU2077526C1 (ru) 1997-04-20
CZ278804B6 (en) 1994-07-13
HU207705B (en) 1993-05-28
CN1028518C (zh) 1995-05-24
NO174546B (no) 1994-02-14
ES2055189T3 (es) 1994-08-16
GB8904794D0 (en) 1989-04-12
NO913382L (no) 1991-08-28
YU39990A (en) 1991-10-31
CA2047748C (en) 1999-05-18
NO174546C (no) 1994-05-25
FI92687C (sv) 1994-12-27
CA2047748A1 (en) 1990-09-03
PT93317A (pt) 1990-11-07
JPH04503803A (ja) 1992-07-09
MY105260A (en) 1994-09-30
KR0171047B1 (ko) 1999-03-30
EP0385354A1 (en) 1990-09-05
CN1045259A (zh) 1990-09-12
DE69001312D1 (de) 1993-05-19
PT93317B (pt) 1996-01-31
NO913382D0 (no) 1991-08-28
HUT58033A (en) 1992-01-28
HU902357D0 (en) 1991-11-28
IL93559A (en) 1994-06-24
US5180758A (en) 1993-01-19
ZA901542B (en) 1990-12-28
CS9000958A2 (en) 1991-08-13
EP0385354B1 (en) 1993-04-14
IL93559A0 (en) 1990-11-29
AU5184890A (en) 1990-09-26
WO1990009974A1 (en) 1990-09-07
AU636134B2 (en) 1993-04-22
NZ232681A (en) 1991-04-26
FI914053A0 (sv) 1991-08-28
DE69001312T2 (de) 1993-07-22
IE900700L (en) 1990-09-02
YU47556B (sh) 1995-10-03
JP2717023B2 (ja) 1998-02-18
ATE88173T1 (de) 1993-04-15
DK0385354T3 (da) 1993-05-17
SK278225B6 (en) 1996-04-03
IE63571B1 (en) 1995-05-17

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Legal Events

Date Code Title Description
BB Publication of examined application
PC Transfer of assignment of patent

Owner name: PHARMACIA & UPJOHN S.P.A.