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FI903752A0 - Foerfarande foer framstaellning av 1,2,3,4-tetrahydro-9-akridinaminderivat. - Google Patents

Foerfarande foer framstaellning av 1,2,3,4-tetrahydro-9-akridinaminderivat.

Info

Publication number
FI903752A0
FI903752A0 FI903752A FI903752A FI903752A0 FI 903752 A0 FI903752 A0 FI 903752A0 FI 903752 A FI903752 A FI 903752A FI 903752 A FI903752 A FI 903752A FI 903752 A0 FI903752 A0 FI 903752A0
Authority
FI
Finland
Prior art keywords
tetrahydro
acridinaminderivat
agents
cerebral
frequency fragmentation
Prior art date
Application number
FI903752A
Other languages
English (en)
Other versions
FI903752A7 (fi
Inventor
Colin Granger
Jeffrey Alan Kester
Walter Hamilton Moos
Anthony Jerome Thomas
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of FI903752A0 publication Critical patent/FI903752A0/fi
Publication of FI903752A7 publication Critical patent/FI903752A7/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D219/00Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D219/00Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08Nitrogen atoms
    • C07D219/10Nitrogen atoms attached in position 9
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Psychiatry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Water Treatment By Electricity Or Magnetism (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI903752A 1989-07-31 1990-07-27 Menetelmä 1,2,3,4-tetrahydro-9-akridiiniamiinin johdannaisten valmistamiseksi FI903752A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/387,722 US4999430A (en) 1989-07-31 1989-07-31 Derivatives of 1,2,3,4-tetrahydro-9-acrisinamine

Publications (2)

Publication Number Publication Date
FI903752A0 true FI903752A0 (fi) 1990-07-27
FI903752A7 FI903752A7 (fi) 1991-02-01

Family

ID=23531113

Family Applications (1)

Application Number Title Priority Date Filing Date
FI903752A FI903752A7 (fi) 1989-07-31 1990-07-27 Menetelmä 1,2,3,4-tetrahydro-9-akridiiniamiinin johdannaisten valmistamiseksi

Country Status (17)

Country Link
US (1) US4999430A (fi)
EP (2) EP0411534B1 (fi)
JP (1) JP2930245B2 (fi)
KR (1) KR910002802A (fi)
AT (2) ATE119885T1 (fi)
AU (1) AU5994590A (fi)
CA (1) CA2022297C (fi)
DE (2) DE69033369T2 (fi)
DK (2) DK0411534T3 (fi)
ES (2) ES2141787T3 (fi)
FI (1) FI903752A7 (fi)
GR (1) GR3032539T3 (fi)
IE (1) IE66823B1 (fi)
NO (1) NO903359L (fi)
NZ (1) NZ234672A (fi)
PT (1) PT94849A (fi)
ZA (1) ZA905978B (fi)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0282959A3 (en) * 1987-03-17 1989-05-31 Hoechst-Roussel Pharmaceuticals Incorporated Substituted 9-amino-tetrahydro-acridines and related compounds, a process for their preparation and their use as medicaments
FR2640508B1 (fr) * 1988-12-19 1994-07-01 Dietlin Francois Nouvelles compositions et nouveaux produits pharmaceutiques assurant la regeneration de leucocytes et leur emploi pour le traitement du syndrome immuno-deficitaire
JP2546919B2 (ja) * 1989-11-08 1996-10-23 三菱化学株式会社 9ーアシルアミノテトラヒドロアクリジン誘導体
CA2029497C (en) * 1989-11-08 2002-06-04 Kunihiro Ninomiya (Deceased) 4-acylaminopyridine derivative
US5179100A (en) * 1992-03-09 1993-01-12 Hoechst-Roussel Pharmaceuticals Inc. 4,5-dihydropyrazolo[3,4-a]acridines
US5466696A (en) * 1992-09-10 1995-11-14 Warner Lambert Company Tacrine and cytochrome P450 oxidase inhibitors and methods of use
US5422350A (en) * 1992-09-10 1995-06-06 Warner-Lambert Company Nitrogen substituted acridine and cytochrome P450 inhibitors and methods of use
HU213107B (en) * 1994-02-23 1997-02-28 Egyt Gyogyszervegyeszeti Gyar Process for producing acetic acid derivatives and pharmaceutical compositions containing them
GB9716879D0 (en) * 1997-08-08 1997-10-15 Shire Int Licensing Bv Treatment of attention deficit disorders
US6218383B1 (en) 1998-08-07 2001-04-17 Targacept, Inc. Pharmaceutical compositions for the prevention and treatment of central nervous system disorders
ES2168926B1 (es) * 1999-12-14 2003-10-16 Prous Science S A Derivados de ciclopenta- ciclohexa- y ciclohepta (b)quinoleina, procedimiento para su fabricacion, utilizacion y composicion farmaceutica correspondiente.
EP1779867A4 (en) * 2004-07-01 2009-12-02 Eisai R&D Man Co Ltd MEANS FOR PROMOTING NERVE REVENERATION
CN1315810C (zh) * 2004-08-30 2007-05-16 北京理工大学 哌嗪桥联他克林双体衍生物及其合成方法
US20080188510A1 (en) * 2005-05-23 2008-08-07 Eisai R & D Management Co., Ltd. Novel methods using zonisamide
WO2011070177A2 (en) * 2009-12-11 2011-06-16 Baltic Technology Development, Ltd. Methods of facilitating neural cell survival using gdnf family ligand (gfl) mimetics or ret signaling pathway activators
CN102905532A (zh) 2010-02-09 2013-01-30 约翰斯.霍普金斯大学 用于改善认知功能的方法和组合物
HK1215170A1 (zh) 2012-11-14 2016-08-19 The Johns Hopkins University 治療精神分裂症的方法和組合物
CA2904767C (en) 2013-03-15 2022-06-21 Agenebio, Inc. Methods and compositions for improving cognitive function
WO2014144663A1 (en) 2013-03-15 2014-09-18 The Johns Hopkins University Methods and compositions for improving cognitive function
EA034167B8 (ru) 2015-05-22 2021-04-27 Эйджинбайо, Инк. Фармацевтические композиции леветирацетама пролонгированного высвобождения

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3889302T2 (de) * 1987-12-03 1994-10-20 Mitsubishi Chem Ind 9-(Acylamino)tetrahydroacridinderivate und wahrnehmungssteigernde Mittel davon als aktiver Wirkstoff.

Also Published As

Publication number Publication date
JP2930245B2 (ja) 1999-08-03
JPH0366670A (ja) 1991-03-22
EP0628548A1 (en) 1994-12-14
ATE186908T1 (de) 1999-12-15
NO903359D0 (no) 1990-07-30
GR3032539T3 (en) 2000-05-31
ATE119885T1 (de) 1995-04-15
EP0411534A3 (en) 1991-06-05
EP0411534B1 (en) 1995-03-15
KR910002802A (ko) 1991-02-26
ES2068955T3 (es) 1995-05-01
FI903752A7 (fi) 1991-02-01
CA2022297A1 (en) 1991-02-01
DE69033369D1 (de) 1999-12-30
AU5994590A (en) 1991-01-31
US4999430A (en) 1991-03-12
IE66823B1 (en) 1996-02-07
DK0628548T3 (da) 2000-05-08
DE69017789T2 (de) 1995-07-13
IE902751A1 (en) 1991-02-27
DE69033369T2 (de) 2000-05-11
EP0628548B1 (en) 1999-11-24
NZ234672A (en) 1991-11-26
CA2022297C (en) 2001-09-18
DK0411534T3 (da) 1995-07-24
ES2141787T3 (es) 2000-04-01
EP0411534A2 (en) 1991-02-06
NO903359L (no) 1991-02-01
PT94849A (pt) 1991-04-18
ZA905978B (en) 1992-04-29
DE69017789D1 (de) 1995-04-20

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Legal Events

Date Code Title Description
FD Application lapsed

Owner name: WARNER-LAMBERT COMPANY