FI906366A0 - Nytt foerfarande foer framstaellning av 1-fenyl-imidazol-2,5-dionderivat. - Google Patents

Nytt foerfarande foer framstaellning av 1-fenyl-imidazol-2,5-dionderivat.

Info

Publication number: FI906366A0
Authority: FI; Finland
Prior art keywords: phenyl; dionderivat; imidazole; formula; image
Prior art date: 1989-12-22

Application number

FI906366A

Other languages

English (en)

Other versions

FI103203B1 (fi

FI906366L (fi

FI103203B (fi

Inventor

Patrick Seuron

Daniel Varraillon

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-12-22

Filing date

1990-12-21

Publication date

1990-12-21

1990-12-21 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1990-12-21 Publication of FI906366A0 publication Critical patent/FI906366A0/fi

1991-06-23 Publication of FI906366L publication Critical patent/FI906366L/fi

1999-05-14 Application granted granted Critical

1999-05-14 Publication of FI103203B1 publication Critical patent/FI103203B1/fi

1999-05-14 Publication of FI103203B publication Critical patent/FI103203B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
- C07D233/74—Two oxygen atoms, e.g. hydantoin with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to other ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Reinforced Plastic Materials (AREA)
Compositions Of Macromolecular Compounds (AREA)
Photoreceptors In Electrophotography (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

FI906366A 1989-12-22 1990-12-21 Uusi menetelmä 1-fenyyli-imidatsolin-2,5-dionin johdannaisten valmista miseksi FI103203B (fi)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8917046A FR2656302B1 (fr)	1989-12-22	1989-12-22	Nouveau procede de preparation de l'anandron et derives de l'anandron.

Publications (4)

Publication Number	Publication Date
FI906366A0 true FI906366A0 (fi)	1990-12-21
FI906366L FI906366L (fi)	1991-06-23
FI103203B1 FI103203B1 (fi)	1999-05-14
FI103203B FI103203B (fi)	1999-05-14

Family

ID=9388859

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI906366A FI103203B (fi)	1989-12-22	1990-12-21	Uusi menetelmä 1-fenyyli-imidatsolin-2,5-dionin johdannaisten valmista miseksi

Country Status (24)

Country	Link
US (1)	US5166358A (fi)
EP (1)	EP0436426B1 (fi)
JP (1)	JP2836041B2 (fi)
KR (1)	KR0173307B1 (fi)
CN (1)	CN1048011C (fi)
AT (1)	ATE107289T1 (fi)
AU (1)	AU628699B2 (fi)
CA (1)	CA2032988C (fi)
CZ (1)	CZ281655B6 (fi)
DE (1)	DE69009964T2 (fi)
DK (1)	DK0436426T3 (fi)
ES (1)	ES2055382T3 (fi)
FI (1)	FI103203B (fi)
FR (1)	FR2656302B1 (fi)
HU (1)	HU207301B (fi)
IE (1)	IE65510B1 (fi)
IL (1)	IL96696A (fi)
NZ (1)	NZ236621A (fi)
PL (1)	PL164694B1 (fi)
PT (1)	PT96313B (fi)
RU (1)	RU1836356C (fi)
SK (1)	SK656790A3 (fi)
UA (1)	UA27220C2 (fi)
ZA (1)	ZA909648B (fi)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5411981A (en) *	1991-01-09	1995-05-02	Roussel Uclaf	Phenylimidazolidines having antiandrogenic activity
FR2693461B1 (fr) *	1992-07-08	1994-09-02	Roussel Uclaf	Nouvelles phénylimidazolidines substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.
FR2694290B1 (fr) *	1992-07-08	1994-09-02	Roussel Uclaf	Nouvelles phénylimidazolidines éventuellement substituées, leur procédé de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.
US5656651A (en) *	1995-06-16	1997-08-12	Biophysica Inc.	Androgenic directed compositions
DE19540027A1 (de) *	1995-10-27	1997-04-30	Gruenenthal Gmbh	Substituierte Imidazolidin-2,4-dion-Verbindungen als pharmazeutische Wirkstoffe
FR2741346B1 (fr) *	1995-11-16	1997-12-19	Roussel Uclaf	Nouveau procede de preparation de derives phenylimidazolidine
FR2741342B1 (fr) *	1995-11-22	1998-02-06	Roussel Uclaf	Nouvelles phenylimidazolidines fluorees ou hydroxylees, procede, intermediaires de preparation, application comme medicaments, nouvelle utilisation et compositions pharmaceutiques
JPH1072446A (ja) *	1996-06-24	1998-03-17	Sumitomo Chem Co Ltd	１−置換−ヒダントイン類の製造法
US20040077605A1 (en)	2001-06-20	2004-04-22	Salvati Mark E.	Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
BR0111298A (pt) *	2000-06-28	2005-05-10	Bristol Myers Squibb Co	Moduladores seletivos dos receptores de andrógenos e métodos para identificação, projeto e uso dos mesmos
US7001911B2 (en)	2000-06-28	2006-02-21	Bristol-Myers Squibb Company	Fused cyclic modulators of nuclear hormone receptor function
US6953679B2 (en)	2000-09-19	2005-10-11	Bristol-Myers Squibb Company	Method for the preparation of fused heterocyclic succinimide compounds and analogs thereof
EP1854798A3 (en)	2000-09-19	2007-11-28	Bristol-Myers Squibb Company	Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
US20040087548A1 (en)	2001-02-27	2004-05-06	Salvati Mark E.	Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
AU2002364082A1 (en)	2001-12-19	2003-07-09	Bristol-Myers Squibb Company	Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function
AU2004305075A1 (en) *	2003-12-19	2005-07-07	The Regents Of The University Of California	Methods and materials for assessing prostate cancer therapies
NZ550102A (en) *	2004-02-24	2010-10-29	Univ California	Methods and materials for assessing prostate cancer therapies and compounds (thiohydantoine derivatives)
US7709517B2 (en) *	2005-05-13	2010-05-04	The Regents Of The University Of California	Diarylhydantoin compounds
AU2007245022A1 (en) *	2006-03-29	2007-11-08	The Regents Of The University Of California	Diarylthiohydantoin compounds
DK3100727T3 (en)	2006-03-27	2018-11-12	Univ California	Androgen receptor modulator for the treatment of prostate cancer and androgen receptor-associated diseases
WO2009055053A2 (en)	2007-10-26	2009-04-30	The Regents Of The University Of California	Diarylhydantoin compounds as androgen receptor modulators
EP3124481B1 (en)	2010-02-16	2018-03-28	Aragon Pharmaceuticals, Inc.	Androgen receptor modulators and uses thereof
SG10201912719TA (en)	2012-09-26	2020-02-27	Aragon Pharmaceuticals Inc	Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer
JOP20200097A1 (ar)	2013-01-15	2017-06-16	Aragon Pharmaceuticals Inc	معدل مستقبل أندروجين واستخداماته
TWI726969B (zh)	2016-01-11	2021-05-11	比利時商健生藥品公司	用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
JP7201694B2 (ja)	2017-10-16	2023-01-10	アラゴンファーマシューティカルズ，インコーポレイテッド	非転移性去勢抵抗性前立腺癌の治療のための抗アンドロゲン剤

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH166004A (de) *	1934-06-06	1933-12-15	Chem Fab Vormals Sandoz	Verfahren zur Darstellung eines Derivates des 5,5-Phenyläthylhydantoins.
US2490813A (en) *	1944-11-29	1949-12-13	Standard Oil Co	Continuous process for making aryl amines
US2759002A (en) *	1954-03-24	1956-08-14	Abbott Lab	3-benzyl hydantoin and process
US3134663A (en) *	1957-07-23	1964-05-26	Geigy Chem Corp	Herbicidal composition and method employing hydantoins
US3914311A (en) *	1973-06-15	1975-10-21	Du Pont	Preparation of aromatic secondary and tertiary amines using a nickel complex catalyst
DE2414613A1 (de) *	1974-03-26	1975-10-16	Bayer Ag	1-aryl-5-alkyliden-2,4-dioxo-imidazolidine
FR2329276A1 (fr) *	1975-10-29	1977-05-27	Roussel Uclaf	Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant
CA1138334A (en) *	1977-10-28	1982-12-28	Karl Bernauer	Pharmaceutical preparations containing certain urea derivatives
GB1598166A (en) *	1978-05-23	1981-09-16	Lilly Industries Ltd	3,5-disubstituted hydantoin derivatives
US4764625A (en) *	1980-12-12	1988-08-16	Xerox Corporation	Process for preparing arylamines
DE3382406D1 (de) *	1982-04-08	1991-10-17	Shell Int Research	Neue hydantoine, ihre herstellung und verwendung.

1989
- 1989-12-22 FR FR8917046A patent/FR2656302B1/fr not_active Expired - Fee Related
1990
- 1990-11-16 IE IE414290A patent/IE65510B1/en not_active IP Right Cessation
- 1990-11-30 ZA ZA909648A patent/ZA909648B/xx unknown
- 1990-12-10 JP JP2407176A patent/JP2836041B2/ja not_active Expired - Lifetime
- 1990-12-17 IL IL9669690A patent/IL96696A/en not_active IP Right Cessation
- 1990-12-18 US US07/629,490 patent/US5166358A/en not_active Expired - Lifetime
- 1990-12-20 PL PL90288365A patent/PL164694B1/pl unknown
- 1990-12-20 AU AU68265/90A patent/AU628699B2/en not_active Expired
- 1990-12-21 KR KR1019900021357A patent/KR0173307B1/ko not_active Expired - Lifetime
- 1990-12-21 DE DE69009964T patent/DE69009964T2/de not_active Expired - Lifetime
- 1990-12-21 NZ NZ236621A patent/NZ236621A/en unknown
- 1990-12-21 HU HU908416A patent/HU207301B/hu unknown
- 1990-12-21 RU SU904894040A patent/RU1836356C/ru active
- 1990-12-21 EP EP90403725A patent/EP0436426B1/fr not_active Expired - Lifetime
- 1990-12-21 ES ES90403725T patent/ES2055382T3/es not_active Expired - Lifetime
- 1990-12-21 SK SK6567-90A patent/SK656790A3/sk not_active IP Right Cessation
- 1990-12-21 CZ CS906567A patent/CZ281655B6/cs not_active IP Right Cessation
- 1990-12-21 AT AT90403725T patent/ATE107289T1/de not_active IP Right Cessation
- 1990-12-21 CA CA002032988A patent/CA2032988C/fr not_active Expired - Lifetime
- 1990-12-21 PT PT96313A patent/PT96313B/pt not_active IP Right Cessation
- 1990-12-21 UA UA4894040A patent/UA27220C2/uk unknown
- 1990-12-21 FI FI906366A patent/FI103203B/fi active IP Right Grant
- 1990-12-21 DK DK90403725.6T patent/DK0436426T3/da active
- 1990-12-22 CN CN90110071A patent/CN1048011C/zh not_active Expired - Lifetime

Also Published As

Publication number	Publication date
SK278447B6 (en)	1997-06-04
US5166358A (en)	1992-11-24
PL288365A1 (en)	1991-09-09
FR2656302B1 (fr)	1992-05-07
CN1052666A (zh)	1991-07-03
PL164694B1 (pl)	1994-09-30
IL96696A (en)	1995-08-31
IL96696A0 (en)	1991-09-16
FR2656302A1 (fr)	1991-06-28
EP0436426A1 (fr)	1991-07-10
HU207301B (en)	1993-03-29
JPH04103573A (ja)	1992-04-06
ZA909648B (en)	1992-02-26
JP2836041B2 (ja)	1998-12-14
CZ656790A3 (en)	1996-08-14
RU1836356C (ru)	1993-08-23
CA2032988A1 (fr)	1991-06-23
DE69009964T2 (de)	1994-10-13
FI103203B1 (fi)	1999-05-14
ES2055382T3 (es)	1994-08-16
EP0436426B1 (fr)	1994-06-15
KR0173307B1 (ko)	1999-02-01
DE69009964D1 (de)	1994-07-21
FI906366L (fi)	1991-06-23
CN1048011C (zh)	2000-01-05
NZ236621A (en)	1992-04-28
PT96313A (pt)	1991-09-30
CA2032988C (fr)	2003-04-29
UA27220C2 (uk)	2000-08-15
IE904142A1 (en)	1991-07-03
CZ281655B6 (cs)	1996-12-11
KR910011799A (ko)	1991-08-07
HU908416D0 (en)	1991-07-29
AU628699B2 (en)	1992-09-17
SK656790A3 (en)	1997-06-04
PT96313B (pt)	1998-06-30
IE65510B1 (en)	1995-11-01
AU6826590A (en)	1991-06-27
DK0436426T3 (da)	1994-07-04
FI103203B (fi)	1999-05-14
ATE107289T1 (de)	1994-07-15

Publication	Publication Date	Title
FI906366A0 (fi)	1990-12-21	Nytt foerfarande foer framstaellning av 1-fenyl-imidazol-2,5-dionderivat.
ES538757A0 (es)	1985-11-01	Procedimiento para la preparacion de 11b-aril-estradienos
IE811931L (en)	1982-02-25	Oxiranes.
BR9203919A (pt)	1993-04-27	Processo para a preparacao de uma n-(aril)-1,2,4-triazolopirimidina-2-sulfonamida
IL60975A (en)	1984-03-30	Substituted oxiranecarboxylic acids,processes for their preparation and pharmaceutical compositions containing them
FR2665446B1 (fr)	1992-11-27	Procede et catalyseur comprenant un compose de lanthanide comme additif promoteur pour la synthese directe du dimethyldichlorosilane.
SE8001556L (sv)	1980-09-03	Tetrahydrobensotiazolylimidazolidinoner
DE3560027D1 (en)	1987-01-15	Process for the preparation of o,o'-dithiobenzamides
FR2443457A1 (fr)	1980-07-04	Derives de 1-phenyl-2-amino-1-propanol, leur procede de preparation et leur utilisation comme medicaments
ATE42542T1 (de)	1989-05-15	3-amino-azetidin, seine salze, verfahren zu deren herstellung und zwischenprodukte.
SE8302824D0 (sv)	1983-05-19	New herbicidal compounds
FR2376139A1 (fr)	1978-07-28	Nouveaux derives d'isoquinoleine-acetamide utiles comme medicaments
GR75012B (fi)	1984-07-12
ATE17710T1 (de)	1986-02-15	Keten-0,0-acetale und verfahren zu ihrer herstellung.
JPS5214773A (en)	1977-02-03	Process for preparing novel benzylpyridine derivatives
ES454038A1 (es)	1977-11-16	Procedimiento para la preparacion de amidas derivadas de la 4-aminopiperidina.
JPS5473775A (en)	1979-06-13	Isoxazoline-3-one derivative
EP0424248A3 (en)	1992-01-22	20,21-dinoreburnamine derivatives, substituted in position 15, process for their preparation and novel intermediates so obtained, their use as medicines and compositions containing them
JPS5283565A (en)	1977-07-12	Novel benzylpyridine derivatives
ES483300A1 (es)	1980-09-01	Un procedimiento para la preparacion de derivados de benzo- diacepina
SE8302547D0 (sv)	1983-05-04	Heterocykliska amider av fenoxifenoxialkansyror
FR2401927A1 (fr)	1979-03-30	Derives de thiazine utiles comme medicaments
JPS5473774A (en)	1979-06-13	Isoxazoline-3-one derivative
JPS5432437A (en)	1979-03-09	2-thio-2-(3-phenoxyphenyl)alkane-carboxylic acid derivatives and their preparation

Legal Events

Date	Code	Title	Description
1990-12-21	FG	Patent granted	Owner name: HOECHST MARION ROUSSEL
1998-10-15	GB	Transfer or assigment of application	Owner name: HOECHST MARION ROUSSEL
2004-08-31	FG	Patent granted	Owner name: AVENTIS PHARMA S.A.