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FI892897A7 - Nya kondenserade diazepinoner, foerfarande foer deras framstaellning och laekemedel som innehaoller dessa foereningar. - Google Patents

Nya kondenserade diazepinoner, foerfarande foer deras framstaellning och laekemedel som innehaoller dessa foereningar. Download PDF

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Publication number
FI892897A7
FI892897A7 FI892897A FI892897A FI892897A7 FI 892897 A7 FI892897 A7 FI 892897A7 FI 892897 A FI892897 A FI 892897A FI 892897 A FI892897 A FI 892897A FI 892897 A7 FI892897 A7 FI 892897A7
Authority
FI
Finland
Prior art keywords
kondenserade
diazepinoner
laekemedel
nya
foerfarande foer
Prior art date
Application number
FI892897A
Other languages
English (en)
Other versions
FI892897A0 (fi
Inventor
Gerhard Mihm
Wolfgang Eberlein
Wolfhard Engel
Guenter Trummlitz
Norbert Mayer
Jonge Adriaan De
Henri Doods
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Priority to FI925819A priority Critical patent/FI925819A0/fi
Publication of FI892897A0 publication Critical patent/FI892897A0/fi
Publication of FI892897A7 publication Critical patent/FI892897A7/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
FI892897A 1988-06-15 1989-06-14 Nya kondenserade diazepinoner, foerfarande foer deras framstaellning och laekemedel som innehaoller dessa foereningar. FI892897A7 (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI925819A FI925819A0 (fi) 1988-06-15 1989-06-14 Foerfarande foer framstaellning av terapeutiskt aktiva 11h-dibentso/b,e//1,4/diazepin-11-oner

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3820346A DE3820346A1 (de) 1988-06-15 1988-06-15 Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
FI892897A0 FI892897A0 (fi) 1989-06-14
FI892897A7 true FI892897A7 (fi) 1989-12-16

Family

ID=6356594

Family Applications (1)

Application Number Title Priority Date Filing Date
FI892897A FI892897A7 (fi) 1988-06-15 1989-06-14 Nya kondenserade diazepinoner, foerfarande foer deras framstaellning och laekemedel som innehaoller dessa foereningar.

Country Status (16)

Country Link
US (1) US5002943A (fi)
EP (1) EP0346745A1 (fi)
JP (1) JPH0240381A (fi)
KR (1) KR900000365A (fi)
AU (1) AU612493B2 (fi)
DD (1) DD284016A5 (fi)
DE (1) DE3820346A1 (fi)
DK (1) DK291189A (fi)
FI (1) FI892897A7 (fi)
HU (1) HU201759B (fi)
IL (1) IL90590A0 (fi)
NO (1) NO168477C (fi)
PH (1) PH27213A (fi)
PT (1) PT90842A (fi)
SU (1) SU1678209A3 (fi)
ZA (1) ZA894461B (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3818299A1 (de) * 1988-05-30 1989-12-07 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DD295849A5 (de) * 1989-06-28 1991-11-14 �������������@��������@��������@����Kk�� Neuartige 5,11-dihydo-6h-dipyrido[3,2-b:2',3'-e]diazepin-6-one und thione und ihre anwendung bei der verhuetung bzw. behandlung von aids
US5179090A (en) * 1989-09-11 1993-01-12 Klaus Rudolf Condensed diazepinones and medicaments containing these compounds
US5418229A (en) * 1990-01-06 1995-05-23 Alker; David Muscarinic receptor antagonists
AU3754495A (en) * 1994-10-31 1996-05-23 Yamanouchi Pharmaceutical Co., Ltd. Novel benzodiazepinone derivative and medicinal composition thereof
IL131685A (en) * 1999-09-01 2007-03-08 Mordechai Erez Antiarrhythmic, antifbirillatory, and defibrillatory pharmaceutical compositions containing dibenzoazepines and dibenzodiazepines and same such novel compounds
RU2543320C2 (ru) * 2013-04-01 2015-02-27 Федеральное государственное бюджетное учреждение науки Институт физиологии Коми научного центра Уральского отделения Российской академии наук Применение 2-морфолино-5-фенил-6н-1,3,4-тиадизин, гидробромида в качестве средства, изменяющего суммарную мощность спектра вариабельности сердечного ритма и обладающего антибрадикардическими свойствами

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4210648A (en) * 1977-05-31 1980-07-01 Boehringer Ingelheim Gmbh II-Aminoacyl-5,11-dihydro-6H-pyrido(2,3-B) (1,4)benzodiazepin-6-ones and salts thereof
EP0024582A1 (de) * 1979-08-10 1981-03-11 Byk Gulden Lomberg Chemische Fabrik GmbH Benzodiazepinone, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel
IL62792A (en) * 1980-05-07 1985-02-28 Byk Gulden Lomberg Chem Fab Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
DE3262922D1 (en) * 1981-02-02 1985-05-15 Byk Gulden Lomberg Chem Fab Tricyclic pyrrols, process for their preparation, their use and compositions containing them
EP0213293B1 (de) * 1985-06-27 1992-01-02 Dr. Karl Thomae GmbH In 11-Stellung substituierte 5,11-Dihydro-6H-pyrido-[2,3-b][1,4]benzodiazepin-6-one, Verfahren zur ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE3626095A1 (de) * 1986-07-31 1988-02-11 Thomae Gmbh Dr K Neue substituierte pyrido(2,3-b)(1,4)benzodiazepin-6-one, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
IT8721978A0 (it) * 1987-09-21 1987-09-21 Angeli Inst Spa Nuovi derivati ammidinici triciclici.
US4931436A (en) * 1988-08-09 1990-06-05 Dr. Karl Thomae Gmbh Condensed diazepinones, processes for preparing them and pharmaceutical compositions containing these compounds

Also Published As

Publication number Publication date
DK291189D0 (da) 1989-06-14
NO168477C (no) 1992-02-26
JPH0240381A (ja) 1990-02-09
NO892432L (no) 1989-12-18
HU201759B (en) 1990-12-28
AU3644689A (en) 1989-12-21
ZA894461B (en) 1991-02-27
DD284016A5 (de) 1990-10-31
NO892432D0 (no) 1989-06-13
PT90842A (pt) 1989-12-29
DK291189A (da) 1989-12-16
KR900000365A (ko) 1990-01-30
DE3820346A1 (de) 1989-12-21
IL90590A0 (en) 1990-01-18
FI892897A0 (fi) 1989-06-14
AU612493B2 (en) 1991-07-11
HUT50472A (en) 1990-02-28
PH27213A (en) 1993-05-04
NO168477B (no) 1991-11-18
SU1678209A3 (ru) 1991-09-15
EP0346745A1 (de) 1989-12-20
US5002943A (en) 1991-03-26

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FD Application lapsed
MM Patent lapsed

Owner name: DR. KARL THOMAE GESELLSCHAFT MIT