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FI880387L - 1-(4-hydroxi-3,5-di-tert -butylbenzoyl) homopiperazin, dess olika derivat, foerfarande foer framstaellning av dessa foereningar, dessa innehaollande laekemdel och deras anvaendning. - Google Patents

1-(4-hydroxi-3,5-di-tert -butylbenzoyl) homopiperazin, dess olika derivat, foerfarande foer framstaellning av dessa foereningar, dessa innehaollande laekemdel och deras anvaendning. Download PDF

Info

Publication number
FI880387L
FI880387L FI880387A FI880387A FI880387L FI 880387 L FI880387 L FI 880387L FI 880387 A FI880387 A FI 880387A FI 880387 A FI880387 A FI 880387A FI 880387 L FI880387 L FI 880387L
Authority
FI
Finland
Prior art keywords
dessa
laekemdel
olika
hydroxi
homopiperazin
Prior art date
Application number
FI880387A
Other languages
English (en)
Other versions
FI85469B (fi
FI85469C (fi
FI880387A0 (fi
Inventor
Erhard Wolf
Erhard Rossmanith
Robert R Bartlett
Rudolf Schleyerbach
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI880387A0 publication Critical patent/FI880387A0/fi
Publication of FI880387L publication Critical patent/FI880387L/fi
Publication of FI85469B publication Critical patent/FI85469B/fi
Application granted granted Critical
Publication of FI85469C publication Critical patent/FI85469C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/08Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Lubricants (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fats And Perfumes (AREA)
FI880387A 1987-01-30 1988-01-28 Foerfarande foer framstaellning av terapeutiskt anvaendbara 1-(4-hydroxi-3,5-di-tert -butylbenzoyl) homopiperazinderivat. FI85469C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3702755 1987-01-30
DE19873702755 DE3702755A1 (de) 1987-01-30 1987-01-30 3,5-di-tert.-butyl-4-hydroxybenzoesaeureamid, verschiedene von dessen derivaten, verfahren zur herstellung dieser verbindungen, die sie enthaltenden arzneimittel und ihre verwendung

Publications (4)

Publication Number Publication Date
FI880387A0 FI880387A0 (fi) 1988-01-28
FI880387L true FI880387L (fi) 1988-07-31
FI85469B FI85469B (fi) 1992-01-15
FI85469C FI85469C (fi) 1992-04-27

Family

ID=6319853

Family Applications (1)

Application Number Title Priority Date Filing Date
FI880387A FI85469C (fi) 1987-01-30 1988-01-28 Foerfarande foer framstaellning av terapeutiskt anvaendbara 1-(4-hydroxi-3,5-di-tert -butylbenzoyl) homopiperazinderivat.

Country Status (20)

Country Link
US (1) US4829061A (fi)
EP (1) EP0276803B1 (fi)
JP (1) JPS63192758A (fi)
KR (1) KR880008997A (fi)
AT (1) ATE68488T1 (fi)
AU (1) AU600793B2 (fi)
CA (1) CA1300619C (fi)
DE (2) DE3702755A1 (fi)
DK (1) DK47888A (fi)
ES (1) ES2041705T3 (fi)
FI (1) FI85469C (fi)
GR (1) GR3003523T3 (fi)
HU (1) HU200334B (fi)
IE (1) IE880249L (fi)
IL (1) IL85228A (fi)
NO (1) NO170332C (fi)
NZ (1) NZ223336A (fi)
PH (1) PH24649A (fi)
PT (1) PT86657B (fi)
ZA (1) ZA88642B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE951044C (de) * 1954-08-24 1956-10-18 Heinrich Gueltig Verfahren zum UEberziehen zugeschnittener Flaschenkorken mit einem mindestens vorwiegend Paraffin enthaltenden UEberzug
DE3834532A1 (de) * 1988-10-11 1990-04-12 Behringwerke Ag Verwendung von homopiperazinen zur herstellung eines arzneimittels fuer das vorbeugen gegen und die behandlung von organabstossungsreaktionen
US5281623A (en) * 1990-08-27 1994-01-25 Eli Lilly And Company Method for treating inflammation
CA2049481A1 (en) * 1990-08-27 1992-02-28 Jill Ann Panetta Method of treating inflammatory bowel disease
US5280046A (en) * 1991-02-22 1994-01-18 The University Of Colorado Foundation, Inc. Method of treating type I diabetes
JP3497164B2 (ja) * 1991-06-28 2004-02-16 スミスクライン・ビーチャム・コーポレイション 二環式フィブリノーゲン拮抗薬
US5939412A (en) * 1992-06-26 1999-08-17 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists
WO1994014776A2 (en) * 1992-12-21 1994-07-07 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists
US6403578B1 (en) 1993-12-21 2002-06-11 Smithkline Beecham Corporation Bicyclic fibrinogen antagonists
MA23420A1 (fr) * 1994-01-07 1995-10-01 Smithkline Beecham Corp Antagonistes bicycliques de fibrinogene.
US6458784B1 (en) 1994-06-29 2002-10-01 Smithkline Beecham Corporation Vitronectin receptor antagonists
US5977101A (en) * 1995-06-29 1999-11-02 Smithkline Beecham Corporation Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity
DE19737334A1 (de) * 1997-08-27 1999-03-04 Solvay Pharm Gmbh 7-Phenyl-1,4-diazepan-Derivate, sowie Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19747644C2 (de) * 1997-10-29 2001-02-22 Inst Polymerforschung Dresden Sterisch gehinderte Phenole und Verfahren zu ihrer Herstellung
US7259157B2 (en) 2001-04-03 2007-08-21 Merck & Co., Inc. N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists
WO2006115509A2 (en) 2004-06-24 2006-11-02 Novartis Vaccines And Diagnostics Inc. Small molecule immunopotentiators and assays for their detection
US10449198B2 (en) 2016-07-01 2019-10-22 The University Of Liverpool Method for treating pain
MX2020003575A (es) 2017-10-27 2020-07-22 Esteve Pharmaceuticals Sa Nuevos derivados de alcoxiamino para tratar dolor y estados relacionados con dolor.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4066614A (en) * 1974-12-30 1978-01-03 American Cyanamid Company Heterocyclicamides of hindered 3,5-dialkyl-4-hydroxybenzoic acids and use as light stabilizers in polyolefins
US4404302A (en) * 1982-05-27 1983-09-13 Ferro Corporation Acylated hindered hexahydropyrimidines and their use as light stabilizing agents
DE3685829T2 (de) * 1985-02-04 1992-12-17 Searle & Co Heterocyclische amide.

Also Published As

Publication number Publication date
DK47888D0 (da) 1988-01-29
NO170332C (no) 1992-10-07
FI85469B (fi) 1992-01-15
PT86657B (pt) 1992-02-28
ZA88642B (en) 1988-09-28
ES2041705T3 (es) 1993-12-01
EP0276803A1 (de) 1988-08-03
NO880407L (no) 1988-08-01
NO170332B (no) 1992-06-29
DE3702755A1 (de) 1988-08-11
FI85469C (fi) 1992-04-27
IL85228A (en) 1993-08-18
NZ223336A (en) 1989-09-27
AU1099988A (en) 1988-08-04
KR880008997A (ko) 1988-09-13
PT86657A (pt) 1988-02-01
ATE68488T1 (de) 1991-11-15
GR3003523T3 (fi) 1993-03-16
EP0276803B1 (de) 1991-10-16
FI880387A0 (fi) 1988-01-28
JPS63192758A (ja) 1988-08-10
DE3865443D1 (de) 1991-11-21
US4829061A (en) 1989-05-09
HUT46683A (en) 1988-11-28
AU600793B2 (en) 1990-08-23
DK47888A (da) 1988-07-31
NO880407D0 (no) 1988-01-29
PH24649A (en) 1990-09-07
HU200334B (en) 1990-05-28
CA1300619C (en) 1992-05-12
IE880249L (en) 1988-07-30
IL85228A0 (en) 1988-07-31

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Owner name: HOECHST AKTIENGESELLSCHAFT