[go: up one dir, main page]

FI884455L - RENIN-HAEMMANDE DIPEPTIDER, FOERFARANDE FOER DERAS FRAMSTAELLNING, DESSA INNEHAOLLANDE LAEKEMEDEL OCH DERAS ANVAENDNING. - Google Patents

RENIN-HAEMMANDE DIPEPTIDER, FOERFARANDE FOER DERAS FRAMSTAELLNING, DESSA INNEHAOLLANDE LAEKEMEDEL OCH DERAS ANVAENDNING. Download PDF

Info

Publication number
FI884455L
FI884455L FI884455A FI884455A FI884455L FI 884455 L FI884455 L FI 884455L FI 884455 A FI884455 A FI 884455A FI 884455 A FI884455 A FI 884455A FI 884455 L FI884455 L FI 884455L
Authority
FI
Finland
Prior art keywords
deras
haemmande
dipeptider
renin
foerfarande foer
Prior art date
Application number
FI884455A
Other languages
Finnish (fi)
Other versions
FI884455A0 (en
FI884455A7 (en
Inventor
Adalbert Wagner
Heinz-Werner Kleemann
Dieter Ruppert
Bernward Schoelkens
Hansjoerg Urbach
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI884455A0 publication Critical patent/FI884455A0/en
Publication of FI884455L publication Critical patent/FI884455L/en
Publication of FI884455A7 publication Critical patent/FI884455A7/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0227Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0205Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)3-C(=0)-, e.g. statine or derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06078Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
FI884455A 1987-09-30 1988-09-28 Renin-inhibiting dipeptides, a method for their preparation, medicaments containing them and their use. FI884455A7 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19873732971 DE3732971A1 (en) 1987-09-30 1987-09-30 RENINE INHIBITING DIPEPTIDES, METHOD FOR THE PRODUCTION THEREOF, THE AGENTS CONTAINING THEM AND THEIR USE

Publications (3)

Publication Number Publication Date
FI884455A0 FI884455A0 (en) 1988-09-28
FI884455L true FI884455L (en) 1989-03-31
FI884455A7 FI884455A7 (en) 1989-03-31

Family

ID=6337246

Family Applications (1)

Application Number Title Priority Date Filing Date
FI884455A FI884455A7 (en) 1987-09-30 1988-09-28 Renin-inhibiting dipeptides, a method for their preparation, medicaments containing them and their use.

Country Status (13)

Country Link
EP (1) EP0310015A3 (en)
JP (1) JPH01121258A (en)
KR (1) KR890005146A (en)
AU (1) AU624579B2 (en)
DE (1) DE3732971A1 (en)
DK (1) DK543788A (en)
FI (1) FI884455A7 (en)
HU (1) HU203118B (en)
IL (1) IL87912A0 (en)
NO (1) NO884324L (en)
NZ (1) NZ226361A (en)
PT (1) PT88622B (en)
ZA (1) ZA887264B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL87614A0 (en) * 1987-09-16 1989-01-31 Abbott Lab Peptidylheterocycles
DE3804793A1 (en) * 1988-02-16 1989-08-24 Hoechst Ag RENIN-INHIBITING AMINOSAUTE DERIVATIVES
DE3814325A1 (en) * 1988-04-28 1989-11-09 Merck Patent Gmbh AMINOSAEUREDERIVATE
DE3841520A1 (en) * 1988-12-09 1990-06-13 Hoechst Ag ENZYME-INFRINGING DERIVATIVES OF DIPEPTIDES, METHOD FOR THE PRODUCTION THEREOF, METHODS CONTAINING THEM AND THEIR USE
DE3913290A1 (en) * 1989-04-22 1990-10-25 Hoechst Ag RENIN-INHIBITING DI- AND TRIPEPTIDES, METHOD FOR THE PRODUCTION THEREOF, THE MEANS CONTAINING THEM AND THEIR USE
TW225540B (en) * 1990-06-28 1994-06-21 Shionogi & Co
US5554641A (en) * 1995-03-20 1996-09-10 Horwell; David C. Nonpeptides as tachykinin antagonists
JP4696352B2 (en) * 2000-11-30 2011-06-08 トヨタ自動車株式会社 Vehicle power supply

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3538749A1 (en) * 1985-10-31 1987-05-07 Merck Patent Gmbh PEPTIDE
DE3601248A1 (en) * 1986-01-17 1987-07-23 Hoechst Ag SUBSTITUTED 4-AMINO-3-HYDROXYBUTTERIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THESE AGENTS AND THEIR USE
ZA87563B (en) * 1986-02-03 1987-09-30 Squibb & Sons Inc N-heterocyclic alcohol renin inhibitors
DE3627877A1 (en) * 1986-07-30 1988-02-04 Hoechst Ag RENINE-INHIBITING DI- AND TRIPEPTIDES, METHOD FOR THE PRODUCTION THEREOF, THESE AGENTS AND THEIR USE
FI892036L (en) * 1986-10-31 1989-04-28 Pfizer POLYPEPTIDER MED RELATIVT LITEN MOLEKYLVIKT SAOSOM RENININHITORER.
NL8800100A (en) * 1987-01-21 1988-08-16 Sandoz Ag NEW PEPTIDE DERIVATIVES AND METHODS FOR PREPARING AND USING THESE DERIVATIVES.

Also Published As

Publication number Publication date
NO884324L (en) 1989-03-31
FI884455A0 (en) 1988-09-28
HU203118B (en) 1991-05-28
AU624579B2 (en) 1992-06-18
JPH01121258A (en) 1989-05-12
DE3732971A1 (en) 1989-04-20
HUT48278A (en) 1989-05-29
EP0310015A2 (en) 1989-04-05
NO884324D0 (en) 1988-09-29
PT88622B (en) 1993-07-30
DK543788D0 (en) 1988-09-29
DK543788A (en) 1989-03-31
FI884455A7 (en) 1989-03-31
EP0310015A3 (en) 1992-05-20
PT88622A (en) 1989-07-31
IL87912A0 (en) 1989-03-31
NZ226361A (en) 1991-12-23
KR890005146A (en) 1989-05-13
AU2295988A (en) 1989-06-29
ZA887264B (en) 1989-06-28

Similar Documents

Publication Publication Date Title
FI884487A7 (en) KATALYSATORER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH ANVAENDNING.
FI890094A7 (en) CYLINDRISK, NMR-BIASERINGSMAGNETANORDNING UTNYTTJANDE PERMANENTA MAGNETAR OCH FOERFARANDE FOER DENSAMMA.
FI882690A7 (en) POLYOLEFINER INNEHAOLLANDE FUNKTIONEN GRUPPER, MASKERADE MONOMERER INNEHAOLLANDE FUNKTIONEN GRUPPER, REAKTIONSBLANDNINGAR OCH FOERFARANDEN FOER DERAS FRAMSTAELLNING.
FI880198A7 (en) VATTENHALTIGA BLEKMEDELSUSPENSIONER INNEHAOLLANDE PEROXIKARBOXYLSYROR, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING.
FI881086A0 (en) OLJA-I-VATTEN-EMULSIONER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING.
FI894566A7 (en) SUBSTITUERADE BENZAZEPINER, DERAS FRAMSTAELLNING OCH DESSA INNEHAOLLANDE FARMACEUTISKA BLANDNINGAR.
FI884886A0 (en) KALIUMKARBONATBAERARE, KALIUMKATALYTER OCH MEDELST DESSA UTFOERDA OLEFINDIMERISERINGSPROCESSER.
FI884505A0 (en) IMMUNOANALYS, I VILKEN ANVAENDS IGG-UPPSNAPPANDE ANTIKROPPAR OCH DETEKTERINGSSYSTEM FOER FLERA MONOCLONALA ANTIKROPPAR.
FI872147L (en) FISKFODER, FOERFARANDE FOER FRAMSTAELLNING AV DETSAMMA OCH UTFODRINGSFOERFARANDE.
FI872965A0 (en) FOERFARANDE OCH ANORDNING FOER KAPNING AV PAPPER, ISYNNERHET FOERPERFORERAT PAPPER.
FI885592L (en) ARYLOXYPHENYLPROPYLAMINER, DERAS FRAMSTAELLNING OCH ANVAENDNING.
FI885596A0 (en) MANIFYCINDERIVAT, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING.
FI880525L (en) SUBSTITUERADE AMINDERIVAT, DERAS FRAMSTAELLNING OCH ANVAENDNING.
FI882442L (en) ELLEDANDE BELAEGGNINGSMASSA, FOERFARANDE FOER FRAMSTAELLNING OCH ANVAENDNING DAERAV.
FI880199A7 (en) VATTENHALTIGA BLEKMEDELSUSPENSIONER INNEHAOLLANDE PEROXIKARBOXYLSYROR, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING.
FI882715A0 (en) FENOLDERIVAT, DERAS FRAMSTAELLNING OCH ANVAENDNING.
FI881609A7 (en) DIHYDROPYRIDINAMIDER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DERAS ANVAENDNING I LAEKEMEDEL.
FI883986L (en) TRICYKLISKA FUSIONERADE PYRIMIDINDERVAT, DERAS FRAMSTAELLNING OCH ANVAENDNING.
FI884863A7 (en) KONDENSERADE DIAZEPINONER, FOERFARANDE FOER DERAS FRAMSTAELLNING OCH DESSA FOERENINGAR INNEHAOLLANDE LAEKEMEDEL.
FI884455A0 (en) RENIN-HAEMMANDE DIPEPTIDER, FOERFARANDE FOER DERAS FRAMSTAELLNING, DESSA INNEHAOLLANDE CEEKEMEDEL OCH DERAS ANVAENDNING.
FI880661A7 (en) VATTEN-I OLJA-EMULSIONER, VILKA INNEHAOLLER AMIDAS OCH BEHANDLINGSFOERFARANDE FOER DYLIKA EMULSIONER.
FI882251A0 (en) KERAMISKT FOEREMAOL, RAOSATSKOMPOSITION OCH FOERFARANDE.
FI873317A7 (en) FOERFARANDE OCH ANORDNING FOER BESTRYKNING AV LAONGSTRAECKTA STAOLSTYCKEN, ISYNNERHET BETONGSTAOL OCH STAOLPROFILER.
FI872588A0 (en) FOERFARANDE, SAENDARE OCH MOTTAGARE FOER OEVERFOERANDE AV DIGITALISK TILLAEGGSINFORMATION.
FI873969A0 (en) TORKNINGSFOERFARANDE, TORKNINGSENHET OCH TORKNINGSSYSTEM.

Legal Events

Date Code Title Description
FA Application withdrawn [patent]

Owner name: HOECHST AKTIENGESELLSCHAFT