FI864453L - Karboxylsyraesterderivat av deglukoteikoplanin. - Google Patents

Karboxylsyraesterderivat av deglukoteikoplanin. Download PDF

Info

Publication number: FI864453L
Authority: FI; Finland
Prior art keywords: carboxylic acid; deglucoteikoplan; acid ester; ester derivatives; teicoplanin
Prior art date: 1984-06-13

Application number

FI864453A

Other languages

English (en)

Other versions

FI85147B (fi

FI864453A0 (fi

FI85147C (fi

Inventor

Adriano Malabarba

Paolo Strazzolini

Aldo Trani

Ambrogio Magni

Bruno Cavalleri

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-06-13

Filing date

1986-10-31

Publication date

1986-10-31

1986-10-31 Application filed by Lepetit Spa filed Critical Lepetit Spa

1986-10-31 Publication of FI864453A0 publication Critical patent/FI864453A0/fi

1986-10-31 Publication of FI864453L publication Critical patent/FI864453L/fi

1991-11-29 Publication of FI85147B publication Critical patent/FI85147B/fi

1992-03-10 Application granted granted Critical

1992-03-10 Publication of FI85147C publication Critical patent/FI85147C/fi

Links

150000001733 carboxylic acid esters Chemical class 0.000 title abstract 2
230000003115 biocidal effect Effects 0.000 abstract 3
DDTDNCYHLGRFBM-YZEKDTGTSA-N chembl2367892 Chemical compound CC(=O)N[C@H]1[C@@H](O)[C@H](O)[C@H](CO)O[C@H]1O[C@@H]([C@H]1C(N[C@@H](C2=CC(O)=CC(O[C@@H]3[C@H]([C@H](O)[C@H](O)[C@@H](CO)O3)O)=C2C=2C(O)=CC=C(C=2)[C@@H](NC(=O)[C@@H]2NC(=O)[C@@H]3C=4C=C(O)C=C(C=4)OC=4C(O)=CC=C(C=4)[C@@H](N)C(=O)N[C@H](CC=4C=C(Cl)C(O5)=CC=4)C(=O)N3)C(=O)N1)C(O)=O)=O)C(C=C1Cl)=CC=C1OC1=C(O[C@H]3[C@H]([C@@H](O)[C@H](O)[C@H](CO)O3)NC(C)=O)C5=CC2=C1 DDTDNCYHLGRFBM-YZEKDTGTSA-N 0.000 abstract 3
DKVBOUDTNWVDEP-NJCHZNEYSA-N teicoplanin aglycone Chemical compound N([C@H](C(N[C@@H](C1=CC(O)=CC(O)=C1C=1C(O)=CC=C2C=1)C(O)=O)=O)[C@H](O)C1=CC=C(C(=C1)Cl)OC=1C=C3C=C(C=1O)OC1=CC=C(C=C1Cl)C[C@H](C(=O)N1)NC([C@H](N)C=4C=C(O5)C(O)=CC=4)=O)C(=O)[C@@H]2NC(=O)[C@@H]3NC(=O)[C@@H]1C1=CC5=CC(O)=C1 DKVBOUDTNWVDEP-NJCHZNEYSA-N 0.000 abstract 3
108010053950 Teicoplanin Proteins 0.000 abstract 2
229960001608 teicoplanin Drugs 0.000 abstract 2
108010015899 Glycopeptides Proteins 0.000 abstract 1
102000002068 Glycopeptides Human genes 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
239000000126 substance Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Medicinal Chemistry (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

FI864453A 1984-06-13 1986-10-31 Foerfarande foer framstaellning av karboxylsyraesterderivat av deglukoteikoplanin. FI85147C (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GB848415092A GB8415092D0 (en)	1984-06-13	1984-06-13	Ester derivatives
GB8415092		1984-06-13
PCT/EP1985/000262 WO1986000075A1 (en)	1984-06-13	1985-06-02	Carboxylic acid ester derivatives of deglucoteicoplanin
EP8500262		1985-06-02

Publications (4)

Publication Number	Publication Date
FI864453A0 FI864453A0 (fi)	1986-10-31
FI864453L true FI864453L (fi)	1986-10-31
FI85147B FI85147B (fi)	1991-11-29
FI85147C FI85147C (fi)	1992-03-10

Family

ID=10562381

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI864453A FI85147C (fi)	1984-06-13	1986-10-31	Foerfarande foer framstaellning av karboxylsyraesterderivat av deglukoteikoplanin.

Country Status (23)

Country	Link
US (1)	US4954483A (fi)
EP (1)	EP0216775B1 (fi)
JP (1)	JPS61502335A (fi)
KR (1)	KR930000052B1 (fi)
CN (1)	CN85105429A (fi)
AR (1)	AR243898A1 (fi)
AT (1)	ATE42751T1 (fi)
AU (1)	AU585240B2 (fi)
CA (1)	CA1250095A (fi)
DE (1)	DE3569931D1 (fi)
DK (1)	DK52886D0 (fi)
ES (1)	ES8609366A1 (fi)
FI (1)	FI85147C (fi)
GB (1)	GB8415092D0 (fi)
GR (1)	GR851327B (fi)
HU (1)	HU201779B (fi)
IL (1)	IL75475A0 (fi)
NO (1)	NO172051C (fi)
NZ (1)	NZ212388A (fi)
PH (1)	PH21439A (fi)
PT (1)	PT80621B (fi)
WO (1)	WO1986000075A1 (fi)
ZA (1)	ZA854204B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU579120B2 (en) *	1983-12-16	1988-11-17	Gruppo Lepetit S.P.A.	Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
GB8428619D0 (en) *	1984-11-13	1984-12-19	Lepetit Spa	Derivatives of antibiotic l 17046
GB8704847D0 (en) *	1987-03-02	1987-04-08	Lepetit Spa	Substituted alkylamides of teicoplanin compounds
US5135857A (en) *	1987-07-03	1992-08-04	Gruppo Lepetit S.P.A.	Process for the preparation of de-mannosyl teicoplanin derivatives
US5500410A (en) *	1989-03-29	1996-03-19	Gruppo Lepetit S.P.A.	Substituted alkylamide derivatives of teicoplanin
HUT63860A (en) *	1990-12-05	1993-10-28	Lepetit Spa	Process for producing 39-decarboxy-38-(hydroxymethyl) derivatives of teikoplanin antibiotics
US5606036A (en) *	1991-03-27	1997-02-25	Gruppo Lepetit Spa	Antibiotic A 40926 ester derivatives
WO1997002288A1 (en) *	1995-07-05	1997-01-23	Gruppo Lepetit S.P.A.	Purification of dalbaheptide antibiotics by isoelectric focusing
DK0912604T3 (da)	1996-04-23	2002-03-25	Biosearch Italia Spa	Forbedret kemisk fremgangsmåde til fremstilling af amidderivater af A 40926 antibiotikum
PT1565201T (pt) *	2002-11-18	2019-02-05	Vicuron Pharmaceuticals Llc	Métodos de administração de dalbavancina para o tratamento de infeções bacterianas
US20060074014A1 (en) *	2002-11-18	2006-04-06	Vicuron Pharmaceuticals Inc.	Dalbavancin compositions for treatment of bacterial infections
US7119061B2 (en) *	2002-11-18	2006-10-10	Vicuron Pharmaceuticals, Inc.	Dalbavancin compositions for treatment of bacterial infections
EP1740614A2 (en)	2004-04-30	2007-01-10	Theraptosis S.A.	Caspase-2 inhibitors and their biological applications

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4322343A (en) *	1980-12-18	1982-03-30	Eli Lilly And Company	Pseudo-aglycone of actaplanin
RO86375B1 (ro) *	1982-03-24	1985-04-01	Eli Lilly And Company	Procedeu pentru prepararea antibioticului a 41030
ZA831984B (en) *	1982-03-24	1984-04-25	Lilly Co Eli	A41030 antibiotics and their production
FI73697C (fi) *	1982-06-08	1987-11-09	Lepetit Spa	Foerfarande foer framstaellning av individuella faktorer 1, 2, 3, 4 och 5 av teikomysin a2.
US4462942A (en) *	1982-07-30	1984-07-31	Eli Lilly And Company	A47934 Antibiotic and process for production thereof
US4495179A (en) *	1982-12-20	1985-01-22	Eli Lilly And Company	A51568 Antibiotic and process for producing thereof
US4521335A (en) *	1983-07-13	1985-06-04	Smithkline Beckman Corporation	Aglycone and pseudo-aglycones of the AAD 216 antibiotics
US4537715A (en) *	1983-10-21	1985-08-27	Eli Lilly And Company	Glycopeptide antibiotic CUC/CSV and process for its production
US4497802A (en) *	1983-10-21	1985-02-05	Eli Lilly And Company	N-Acyl glycopeptide derivatives
AU579120B2 (en) *	1983-12-16	1988-11-17	Gruppo Lepetit S.P.A.	Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts

1984
- 1984-06-13 GB GB848415092A patent/GB8415092D0/en active Pending
1985
- 1985-05-30 GR GR851327A patent/GR851327B/el unknown
- 1985-06-02 DE DE8585903239T patent/DE3569931D1/de not_active Expired
- 1985-06-02 AU AU45465/85A patent/AU585240B2/en not_active Ceased
- 1985-06-02 JP JP60502999A patent/JPS61502335A/ja active Pending
- 1985-06-02 AT AT85903239T patent/ATE42751T1/de not_active IP Right Cessation
- 1985-06-02 EP EP85903239A patent/EP0216775B1/en not_active Expired
- 1985-06-02 WO PCT/EP1985/000262 patent/WO1986000075A1/en not_active Ceased
- 1985-06-02 US US07/243,168 patent/US4954483A/en not_active Expired - Fee Related
- 1985-06-02 KR KR1019860700082A patent/KR930000052B1/ko not_active Expired - Lifetime
- 1985-06-02 HU HU853054A patent/HU201779B/hu not_active IP Right Cessation
- 1985-06-04 ZA ZA854204A patent/ZA854204B/xx unknown
- 1985-06-10 IL IL75475A patent/IL75475A0/xx not_active IP Right Cessation
- 1985-06-11 PT PT80621A patent/PT80621B/pt not_active IP Right Cessation
- 1985-06-11 AR AR85300685A patent/AR243898A1/es active
- 1985-06-12 CA CA000483725A patent/CA1250095A/en not_active Expired
- 1985-06-12 ES ES544090A patent/ES8609366A1/es not_active Expired
- 1985-06-12 NZ NZ212388A patent/NZ212388A/xx unknown
- 1985-06-13 PH PH32409A patent/PH21439A/en unknown
- 1985-07-16 CN CN198585105429A patent/CN85105429A/zh active Pending
1986
- 1986-02-04 DK DK52886A patent/DK52886D0/da not_active Application Discontinuation
- 1986-02-12 NO NO86860512A patent/NO172051C/no unknown
- 1986-10-31 FI FI864453A patent/FI85147C/fi not_active IP Right Cessation

Also Published As

Publication number	Publication date
PH21439A (en)	1987-10-20
DK52886A (da)	1986-02-04
AR243898A1 (es)	1993-09-30
ES8609366A1 (es)	1986-09-01
EP0216775A1 (en)	1987-04-08
DK52886D0 (da)	1986-02-04
DE3569931D1 (en)	1989-06-08
NO172051C (no)	1993-06-02
KR860700122A (ko)	1986-03-31
FI85147B (fi)	1991-11-29
AU585240B2 (en)	1989-06-15
HUT41820A (en)	1987-05-28
KR930000052B1 (ko)	1993-01-06
GB8415092D0 (en)	1984-07-18
NO172051B (no)	1993-02-22
NZ212388A (en)	1988-11-29
AU4546585A (en)	1986-01-10
CA1250095A (en)	1989-02-14
ZA854204B (en)	1986-02-26
FI864453A0 (fi)	1986-10-31
EP0216775B1 (en)	1989-05-03
US4954483A (en)	1990-09-04
PT80621B (pt)	1987-08-19
IL75475A0 (en)	1985-10-31
JPS61502335A (ja)	1986-10-16
FI85147C (fi)	1992-03-10
HU201779B (en)	1990-12-28
NO860512L (no)	1986-02-12
GR851327B (fi)	1985-11-25
WO1986000075A1 (en)	1986-01-03
CN85105429A (zh)	1987-01-14
PT80621A (en)	1985-07-01
ES544090A0 (es)	1986-09-01
ATE42751T1 (de)	1989-05-15

Publication	Publication Date	Title
FI864453L (fi)	1986-10-31	Karboxylsyraesterderivat av deglukoteikoplanin.
SE8206731L (sv)	1983-05-28	Ester- och amid-derivat av 13,14-didehydro-prostaglandiner
FI944275L (fi)	1994-11-16	Menetelmä syklisten estereiden valmistamiseksi hydroksihapoista ja niiden johdannaisista
MA22733A1 (fr)	1993-07-01	Esters citrates acyles en tant que precurseurs de peracides.
TNSN87021A1 (fr)	1990-01-01	Derives d'indolizine, leur procede de preparation ainsi que les compositions en contenant
IT1183336B (it)	1987-10-22	Procedimento per la produzione di estere metilico della alfa-l-aspartil-fenilalanina oppure del suo alogenidrato
NO884821D0 (no)	1988-10-28	Substituerte alkylamider av teikoplaninforbindelser.
ES2058561T3 (es)	1994-11-01	Esteroides sustituidos con acido fosfonico como inhibidores de la esteroide-5alfa-reductasa.
ES544466A0 (es)	1987-07-01	Procedimiento para la fabricacion de esteres de triterpenilode acidos organicos
NO891703L (no)	1989-04-25	Farmasoeytiske sammensetninger for behandling av psoriasis.
IT1176404B (it)	1987-08-18	Procedimento per la produzione di l-amminoacidi da alfa-chetoacidi
DE3586344D1 (de)	1992-08-20	Esterderivate vom antibiotikum l 17046.
FI920018A7 (fi)	1992-07-05	Menetelmä 3-eksometyleenikefaamisulfoksidiestereiden valmistamiseksi
NO940623L (no)	1994-08-26	Fremgangsmåte for fremstilling av karboksylsyreanhydrider
ES2111791T3 (es)	1998-03-16	Esteres de acidos grasos de derivados de metilglucosido.
NO811340L (no)	1981-10-26	Fremgangsmaate for fremstilling av cyklopropan-karboksylsyreester-derivater.
ES2095459T3 (es)	1997-02-16	Derivados ester del antibiotico a 40926.
SE8301687D0 (sv)	1983-03-28	8-cyano-6,7-dihydro-5-metyl-1-oxo-1h-,5h-benso(ij)kinolizin-2-karboxylsyror och forfarande for framstellning derav
BE894245A (fr)	1983-02-28	Derives d'esters de n-arylsulfinyl-n-phosphonomethylglycinates
NO811339L (no)	1981-10-26	Fremgangsmaate for fremstilling av cyklopropan-karboksylsyreester-derivater.
ES513663A0 (es)	1983-09-01	Procedimiento para obtencion de derivados antibioticos de la cepa streptomyces spec. ws 116
BE894244A (fr)	1983-02-28	Derives d'esters de n-arylsulfinyl-n-phosphonomethylglycinonitriles
FI851306A7 (fi)	1985-10-03	Kefalosporiinijohdannaisten estereitä.
PT82982B (pt)	1988-07-01	Processo de producao de uma composicao antibiotica sinergica dum composto de oxitetraciclina
IT983759B (it)	1974-11-11	Sistema di aggancio rapido per componenti di organi illuminanti quali lampadcari o lampade da muro

Legal Events

Date	Code	Title	Description
1995-01-11	MM	Patent lapsed
2004-08-31	MM	Patent lapsed	Owner name: GRUPPO LEPETIT S.P.A.