FI20116033A7 - Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina - Google Patents

Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina

Info

Publication number: FI20116033A7
Authority: FI; Finland
Prior art keywords: androgen receptor; receptor modulators; new non; steroidal compounds; steroidal
Prior art date: 2011-10-18

Application number

FI20116033A

Other languages

English (en)

Swedish (sv)

Other versions

FI20116033A0 (fi

Inventor

Juha Pulkkinen

Pekka Poutiainen

Tuomas Oravilahti

Jorma Palvimo

Mikael Peraekylae

Reino Laatikainen

Tarja Ihalainen

Original Assignee

Juha Pulkkinen

Pekka Poutiainen

Tuomas Oravilahti

Jorma Palvimo

Mikael Peraekylae

Reino Laatikainen

Tarja Ihalainen

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-10-18

Filing date

2011-10-18

Publication date

2013-04-19

2011-10-18 Application filed by Juha Pulkkinen, Pekka Poutiainen, Tuomas Oravilahti, Jorma Palvimo, Mikael Peraekylae, Reino Laatikainen, Tarja Ihalainen filed Critical Juha Pulkkinen

2011-10-18 Priority to FI20116033A priority Critical patent/FI20116033A7/fi

2011-10-18 Publication of FI20116033A0 publication Critical patent/FI20116033A0/fi

2012-10-17 Priority to PCT/FI2012/050995 priority patent/WO2013057372A1/en

2012-10-17 Priority to EP12841630.2A priority patent/EP2768814A4/en

2012-10-17 Priority to US14/352,052 priority patent/US9278942B2/en

2013-04-19 Publication of FI20116033A7 publication Critical patent/FI20116033A7/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

FI20116033A 2011-10-18 2011-10-18 Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina FI20116033A7 (fi)

Priority Applications (4)

Application Number	Priority Date	Filing Date	Title
FI20116033A FI20116033A7 (fi)	2011-10-18	2011-10-18	Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina
PCT/FI2012/050995 WO2013057372A1 (en)	2011-10-18	2012-10-17	Novel non-steroidal compounds as androgen receptor modulators
EP12841630.2A EP2768814A4 (en)	2011-10-18	2012-10-17	NEW NON-TEROIDAL COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS
US14/352,052 US9278942B2 (en)	2011-10-18	2012-10-17	Non-steroidal compounds as androgen receptor modulators

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FI20116033A FI20116033A7 (fi)	2011-10-18	2011-10-18	Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina

Publications (2)

Publication Number	Publication Date
FI20116033A0 FI20116033A0 (fi)	2011-10-18
FI20116033A7 true FI20116033A7 (fi)	2013-04-19

Family

ID=44883700

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI20116033A FI20116033A7 (fi)	2011-10-18	2011-10-18	Uudet ei-steroidiset yhdisteet androgeenireseptorin muuntelijoina

Country Status (4)

Country	Link
US (1)	US9278942B2 (fi)
EP (1)	EP2768814A4 (fi)
FI (1)	FI20116033A7 (fi)
WO (1)	WO2013057372A1 (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9682960B2 (en)	2013-12-19	2017-06-20	Endorecherche, Inc.	Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5114960A (en) *	1989-07-20	1992-05-19	Hoffmann-La Roche Inc.	Substituted isoxazole derivatives
KR20050044902A (ko)	2002-08-12	2005-05-13	다케다 야쿠힌 고교 가부시키가이샤	축합 벤젠 유도체 및 용도
ES2370788T3 (es)	2005-02-07	2011-12-22	Aerocrine Ab	Controlar flujo de aliento exhalado durante análisis.
WO2008033513A1 (en)	2006-09-15	2008-03-20	Janssen Pharmaceutica N.V.	ISOXAZOLINE ALPHA 1a/1d ADRENORECEPTOR ANTAGONISTS
FI20070897A0 (fi)	2007-11-23	2007-11-23	Juha Pulkkinen	Uudet estrogeeniaktiivisuutta omaavat 4,5-dihydroisoksatsolit

2011
- 2011-10-18 FI FI20116033A patent/FI20116033A7/fi not_active Application Discontinuation
2012
- 2012-10-17 US US14/352,052 patent/US9278942B2/en not_active Expired - Fee Related
- 2012-10-17 WO PCT/FI2012/050995 patent/WO2013057372A1/en not_active Ceased
- 2012-10-17 EP EP12841630.2A patent/EP2768814A4/en not_active Withdrawn

Also Published As

Publication number	Publication date
EP2768814A1 (en)	2014-08-27
FI20116033A0 (fi)	2011-10-18
US9278942B2 (en)	2016-03-08
WO2013057372A1 (en)	2013-04-25
US20140275186A1 (en)	2014-09-18
EP2768814A4 (en)	2015-06-24

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SMT201600271B (it)	2016-08-31	BENZOSSAZEPINONI FUSI COME MODULATORI DI CANALl IONICI
ME03081B (me)	2019-01-20	Modulatora receptora androgena patentni zahtevi
EP2874651A4 (en)	2016-04-27	COMPOUNDS FOR TARGETED IMMUNOTHERAPY
IL230595A0 (en)	2014-03-31	Aniline type compounds
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BR112014012016A2 (pt)	2017-05-16	compostos
IL227559A0 (en)	2013-09-30	Glucagon receptor modulator
EP2764887A4 (en)	2015-12-09	APPLICATOR
CO6910197A2 (es)	2014-03-31	Compuestos novedosos
DK3385252T3 (da)	2022-10-24	Cannabinoidreceptormodulatorer
EP2708280A4 (en)	2015-01-14	LIGHT REACTION MICRO REACTOR
DK2730310T3 (da)	2022-09-05	Applikator
IL239447A0 (en)	2015-07-30	Novel compounds
EP2737924A4 (en)	2015-05-27	APPLICATOR
EP2911666A4 (en)	2016-10-12	MODULATORS OF A RESISTANT ANDROGEN RECEPTOR
DK2804611T3 (da)	2020-11-09	Chitosanafledte forbindelser
IL231440A0 (en)	2014-04-30	Selective androgen receptor modulators
EP2702896A4 (en)	2014-12-03	APPLICATOR
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DK2768442T3 (da)	2019-07-15	Fastgørelsesmekanisme til stomiposer
BR112013028029A2 (pt)	2017-08-08	composto

Legal Events

Date	Code	Title	Description
2013-05-08	FD	Application lapsed