ES8800663A1 - Procedimiento para preparar compuestos arilsulfonicos. - Google Patents
Procedimiento para preparar compuestos arilsulfonicos.Info
- Publication number
- ES8800663A1 ES8800663A1 ES553340A ES553340A ES8800663A1 ES 8800663 A1 ES8800663 A1 ES 8800663A1 ES 553340 A ES553340 A ES 553340A ES 553340 A ES553340 A ES 553340A ES 8800663 A1 ES8800663 A1 ES 8800663A1
- Authority
- ES
- Spain
- Prior art keywords
- alkyl
- hydrogen
- halogen
- image
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 150000002367 halogens Chemical class 0.000 abstract 3
- 150000002431 hydrogen Chemical class 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 2
- 125000002030 1,2-phenylene group Chemical group [H]C1=C([H])C([*:1])=C([*:2])C([H])=C1[H] 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 125000006699 (C1-C3) hydroxyalkyl group Chemical group 0.000 abstract 1
- 230000000767 anti-ulcer Effects 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000000325 methylidene group Chemical group [H]C([H])=* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- -1 sulfone compound Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C47/00—Compounds having —CHO groups
- C07C47/02—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen
- C07C47/105—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing rings
- C07C47/11—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing rings monocyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/76—Dibenzothiophenes
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR COMPUESTOS ARILSULFONICOS. CONSISTE EN HACER REACCIONAR A UN DERIVADO HALURO DE FORMULA (II) CON UNA AMINA DE FORMULA (III), EN DIOXANO, EN PRESENCIA DE CARBONATO SODICO Y ENTRE LA TEMPERATURA AMBIENTE Y 150JC, PARA OBTENER UN COMPUESTO DE FORMULA (I) Y SUS SALES FARMACEUTICAMENTE ACEPTABLES. SIENDO: R1 CICLOHEXILO, FENILO Y OTROS; R2, R3, R4 Y R5 H, HAL, CIANO Y OTROS; R6 H, ALQUILO DE C 1 A 3 Y OTROS; R7 H O ALQUILO DE C 1 A 3; X O O METILENO; Y -(CH2)NY U 0,5 O 6. SE UTILIZAN COMO ANTIULCEROSOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP60051202A JPS61210063A (ja) | 1985-03-14 | 1985-03-14 | アリ−ルスルホン類 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES553340A0 ES553340A0 (es) | 1987-12-01 |
| ES8800663A1 true ES8800663A1 (es) | 1987-12-01 |
Family
ID=12880305
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES553340A Expired ES8800663A1 (es) | 1985-03-14 | 1986-03-13 | Procedimiento para preparar compuestos arilsulfonicos. |
| ES557652A Expired ES8801542A1 (es) | 1985-03-14 | 1987-07-15 | Procedimiento para preparar compuestos arilsulfonicos. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES557652A Expired ES8801542A1 (es) | 1985-03-14 | 1987-07-15 | Procedimiento para preparar compuestos arilsulfonicos. |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US4734500A (es) |
| EP (1) | EP0194669B1 (es) |
| JP (1) | JPS61210063A (es) |
| KR (1) | KR870002002B1 (es) |
| CN (1) | CN1006549B (es) |
| AU (1) | AU566680B2 (es) |
| CA (1) | CA1253503A (es) |
| DE (1) | DE3676722D1 (es) |
| DK (1) | DK165634C (es) |
| ES (2) | ES8800663A1 (es) |
| HU (1) | HU196363B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61210063A (ja) * | 1985-03-14 | 1986-09-18 | Mitsubishi Chem Ind Ltd | アリ−ルスルホン類 |
| CN100339365C (zh) * | 2005-10-08 | 2007-09-26 | 浙江大学 | 3－氨基－4－烷氨基苯甲砜的制备方法 |
| DE102007015767A1 (de) | 2007-03-30 | 2008-10-02 | Oerlikon Optics UK Ltd., Yarnton | Methode zum Laserritzen von Solarzellen |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL300886A (es) * | 1962-11-23 | |||
| NL301580A (es) * | 1962-12-11 | |||
| US4011217A (en) * | 1973-04-19 | 1977-03-08 | Merck Sharp & Dohme (I.A.) Corporation | 4-(3-amino-2-acyloxypropoxy)-1,2,5-thiadiazole compounds |
| SE430156B (sv) * | 1975-06-19 | 1983-10-24 | Mitsubishi Chem Ind | Sett att framstella 2-subst-1-(omega-aminoalkoxi)-bensener |
| US4201866A (en) * | 1977-01-17 | 1980-05-06 | American Home Products Corporation | O-Hemi-succinate of propranolol |
| JPS61210063A (ja) * | 1985-03-14 | 1986-09-18 | Mitsubishi Chem Ind Ltd | アリ−ルスルホン類 |
-
1985
- 1985-03-14 JP JP60051202A patent/JPS61210063A/ja active Granted
-
1986
- 1986-02-25 HU HU86792A patent/HU196363B/hu not_active IP Right Cessation
- 1986-03-10 DK DK109686A patent/DK165634C/da not_active IP Right Cessation
- 1986-03-11 US US06/838,569 patent/US4734500A/en not_active Expired - Fee Related
- 1986-03-12 AU AU54661/86A patent/AU566680B2/en not_active Ceased
- 1986-03-12 EP EP86103312A patent/EP0194669B1/en not_active Expired - Lifetime
- 1986-03-12 DE DE8686103312T patent/DE3676722D1/de not_active Expired - Lifetime
- 1986-03-13 ES ES553340A patent/ES8800663A1/es not_active Expired
- 1986-03-13 KR KR1019860001814A patent/KR870002002B1/ko not_active Expired
- 1986-03-13 CN CN86101618A patent/CN1006549B/zh not_active Expired
- 1986-03-14 CA CA000504206A patent/CA1253503A/en not_active Expired
-
1987
- 1987-07-15 ES ES557652A patent/ES8801542A1/es not_active Expired
- 1987-09-14 US US07/095,766 patent/US4814507A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ES8801542A1 (es) | 1988-02-16 |
| JPH051786B2 (es) | 1993-01-11 |
| DK165634C (da) | 1993-06-01 |
| US4734500A (en) | 1988-03-29 |
| EP0194669A3 (en) | 1988-01-27 |
| CA1253503A (en) | 1989-05-02 |
| KR870002002B1 (ko) | 1987-11-30 |
| ES557652A0 (es) | 1988-02-16 |
| CN86101618A (zh) | 1986-12-17 |
| CN1006549B (zh) | 1990-01-24 |
| DE3676722D1 (de) | 1991-02-14 |
| HUT41721A (en) | 1987-05-28 |
| DK165634B (da) | 1992-12-28 |
| JPS61210063A (ja) | 1986-09-18 |
| AU566680B2 (en) | 1987-10-29 |
| DK109686A (da) | 1986-09-15 |
| HU196363B (en) | 1988-11-28 |
| DK109686D0 (da) | 1986-03-10 |
| EP0194669A2 (en) | 1986-09-17 |
| KR870008838A (ko) | 1987-10-21 |
| AU5466186A (en) | 1986-09-18 |
| ES553340A0 (es) | 1987-12-01 |
| US4814507A (en) | 1989-03-21 |
| EP0194669B1 (en) | 1991-01-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19981001 |