ES8601153A1 - Procedimiento para la obtencion de derivados de acido barbi-turico - Google Patents
Procedimiento para la obtencion de derivados de acido barbi-turicoInfo
- Publication number
- ES8601153A1 ES8601153A1 ES540040A ES540040A ES8601153A1 ES 8601153 A1 ES8601153 A1 ES 8601153A1 ES 540040 A ES540040 A ES 540040A ES 540040 A ES540040 A ES 540040A ES 8601153 A1 ES8601153 A1 ES 8601153A1
- Authority
- ES
- Spain
- Prior art keywords
- image
- acid derivatives
- barbituric acid
- zooparasitic
- helminths
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000007656 barbituric acids Chemical class 0.000 title 1
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 1
- 125000006527 (C1-C5) alkyl group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- HNMQOBQNWWMABB-UHFFFAOYSA-N 2,4,6-trioxo-n-phenyl-1,3-diazinane-5-carboxamide Chemical class O=C1NC(=O)NC(=O)C1C(=O)NC1=CC=CC=C1 HNMQOBQNWWMABB-UHFFFAOYSA-N 0.000 abstract 1
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 230000000507 anthelmentic effect Effects 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 239000000969 carrier Substances 0.000 abstract 1
- 244000000013 helminth Species 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229910052717 sulfur Chemical group 0.000 abstract 1
- 239000011593 sulfur Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
- C07D239/62—Barbituric acids
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Pest Control & Pesticides (AREA)
- Tropical Medicine & Parasitology (AREA)
- Agronomy & Crop Science (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DEL ACIDO BARBITURICO DE SUS FORMAS TAUTOMERAS Y DE SUS SALES DE FORMULA (I) EN LA QUE X REPRESENTA OXIGGENO O AZUFRE; Y R1 R2 R3 R4 Y R5 PUEDEN SER VARIOS TIPOS DE RADICALES. COMPRENDE LA REACCION DE CONDENSACION DE ACIDO BARBITURICO SUSTITUIDO DE FORMULA (II) CON UN ISOCIANATO DE FENILO SUSTITUIDO DE FORMULA (III) EN LAS QUE TODOS LOS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE ORGANICO INERTE EN PRESENCIA DE UNA BASE A UNA TEMPERATURA COMPRENDIDA ENTRE 100JC Y 220JC. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS PARA EL TRATAMIENTO DE LOS HELMINTOS.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH453583 | 1983-08-19 | ||
| CH352684 | 1984-07-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8601153A1 true ES8601153A1 (es) | 1985-11-01 |
| ES540040A0 ES540040A0 (es) | 1985-11-01 |
Family
ID=25693240
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES535293A Granted ES535293A0 (es) | 1983-08-19 | 1984-08-20 | Procedimiento para la obtencion de derivados de acido barbiturico |
| ES540040A Granted ES540040A0 (es) | 1983-08-19 | 1985-02-01 | Procedimiento para la obtencion de derivados de acido barbi-turico |
| ES540037A Expired ES8601152A1 (es) | 1983-08-19 | 1985-02-01 | Procedimiento para la obtencion de derivados de acido barbi-turico |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES535293A Granted ES535293A0 (es) | 1983-08-19 | 1984-08-20 | Procedimiento para la obtencion de derivados de acido barbiturico |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES540037A Expired ES8601152A1 (es) | 1983-08-19 | 1985-02-01 | Procedimiento para la obtencion de derivados de acido barbi-turico |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4748178A (es) |
| EP (1) | EP0135155B1 (es) |
| KR (1) | KR850001907A (es) |
| AU (1) | AU583796B2 (es) |
| CA (1) | CA1264745A (es) |
| DD (1) | DD222876A5 (es) |
| DE (1) | DE3483294D1 (es) |
| DK (1) | DK396384A (es) |
| EG (1) | EG17262A (es) |
| ES (3) | ES535293A0 (es) |
| GB (1) | GB2145087B (es) |
| HU (1) | HU192991B (es) |
| IL (1) | IL72716A (es) |
| MX (1) | MX160630A (es) |
| MY (1) | MY101864A (es) |
| NZ (1) | NZ209267A (es) |
| PH (1) | PH23080A (es) |
| ZW (1) | ZW13584A1 (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2145087B (en) * | 1983-08-19 | 1987-02-04 | Ciba Geigy Ag | Barbituric acid derivatives |
| CH657015A5 (de) * | 1984-06-27 | 1986-08-15 | Ciba Geigy Ag | Motten- und kaeferschutzmittel. |
| PH24423A (en) * | 1985-02-15 | 1990-06-25 | Ciba Geigy Ag | 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives as anthelmintics |
| US4753940A (en) * | 1985-02-15 | 1988-06-28 | Ciba-Geigy Corporation | Barbituric acid derivatives |
| GB8531815D0 (en) * | 1985-12-24 | 1986-02-05 | Wellcome Found | Insecticidal compounds |
| EP0430885A3 (en) * | 1989-12-01 | 1991-11-06 | Ciba-Geigy Ag | Anthelmintical compounds |
| NL9001075A (es) * | 1990-05-04 | 1991-12-02 | Duphar Int Res | |
| AUPO190596A0 (en) | 1996-08-26 | 1996-09-19 | Alchemia Pty Ltd | Oligosaccharide synthesis |
| AUPO937597A0 (en) * | 1997-09-24 | 1997-10-16 | Alchemia Pty Ltd | Protecting and linking groups for organic synthesis |
| KR101272098B1 (ko) * | 2005-02-08 | 2013-06-07 | 가부시키가이샤 한도오따이 에네루기 켄큐쇼 | 발광소자, 발광장치 및 전자기기 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2405733C2 (de) * | 1974-02-07 | 1984-12-13 | Bayer Ag, 5090 Leverkusen | Amidocarbonylthiobarbitursäurederivate und deren Salze, Verfahren zu ihrer Herstellung sowie ihre Verwendung zur Bekämpfung von Insekten, Milben und Pilzen |
| PL103086B1 (pl) * | 1976-05-06 | 1979-05-31 | Ciba Geigy Ag | Srodek owadobojczy |
| DE2832698A1 (de) * | 1978-07-26 | 1980-02-07 | Bayer Ag | Substituierte 5-phenylcarbamoyl- barbitursaeuren, verfahren zu ihrer herstellung und ihre verwendung als insektizide |
| US4283444A (en) * | 1978-09-12 | 1981-08-11 | Ciba-Geigy Corporation | Method of protecting keratinous material from attack by insects that feed on keratin by treatment with 5-phenylcarbamoylbarbituric acid compounds |
| GB2126582B (en) * | 1982-08-26 | 1986-03-05 | Ciba Geigy Ag | Phenyl carbamoyl barbituric acid anthelmintics |
| CH658770A5 (de) * | 1982-08-26 | 1986-12-15 | Ciba Geigy Ag | Motten- und kaeferschutzmittel. |
| GB2145087B (en) * | 1983-08-19 | 1987-02-04 | Ciba Geigy Ag | Barbituric acid derivatives |
| IL73840A (en) * | 1983-12-19 | 1988-11-15 | Uniroyal Chem Co Inc | 2-thio-5-(thio)carbamoyl barbituric acid derivatives,their preparation and pharmaceutical compositions containing them |
| CH657015A5 (de) * | 1984-06-27 | 1986-08-15 | Ciba Geigy Ag | Motten- und kaeferschutzmittel. |
| EP0167491A3 (de) * | 1984-07-06 | 1986-12-30 | Ciba-Geigy Ag | Thiobarbitursäurederivate |
| PH24423A (en) * | 1985-02-15 | 1990-06-25 | Ciba Geigy Ag | 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives as anthelmintics |
-
1984
- 1984-08-15 GB GB08420712A patent/GB2145087B/en not_active Expired
- 1984-08-16 EP EP84109765A patent/EP0135155B1/de not_active Expired - Lifetime
- 1984-08-16 DE DE8484109765T patent/DE3483294D1/de not_active Expired - Lifetime
- 1984-08-17 DD DD84266391A patent/DD222876A5/de unknown
- 1984-08-17 AU AU32040/84A patent/AU583796B2/en not_active Ceased
- 1984-08-17 ZW ZW135/84A patent/ZW13584A1/xx unknown
- 1984-08-17 DK DK396384A patent/DK396384A/da not_active Application Discontinuation
- 1984-08-17 CA CA000461250A patent/CA1264745A/en not_active Expired - Lifetime
- 1984-08-17 HU HU843130A patent/HU192991B/hu unknown
- 1984-08-17 NZ NZ209267A patent/NZ209267A/en unknown
- 1984-08-17 IL IL72716A patent/IL72716A/xx unknown
- 1984-08-17 PH PH31116A patent/PH23080A/en unknown
- 1984-08-18 KR KR1019840004982A patent/KR850001907A/ko not_active Ceased
- 1984-08-19 EG EG530/84A patent/EG17262A/xx active
- 1984-08-20 ES ES535293A patent/ES535293A0/es active Granted
- 1984-08-20 MX MX8345A patent/MX160630A/es unknown
-
1985
- 1985-02-01 ES ES540040A patent/ES540040A0/es active Granted
- 1985-02-01 ES ES540037A patent/ES8601152A1/es not_active Expired
-
1986
- 1986-02-13 US US06/829,589 patent/US4748178A/en not_active Expired - Fee Related
-
1987
- 1987-09-25 MY MYPI87001955A patent/MY101864A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES540037A0 (es) | 1985-11-01 |
| EP0135155B1 (de) | 1990-09-26 |
| NZ209267A (en) | 1988-01-08 |
| ES8506290A1 (es) | 1985-07-16 |
| IL72716A (en) | 1987-10-20 |
| GB8420712D0 (en) | 1984-09-19 |
| DK396384D0 (da) | 1984-08-17 |
| CA1264745A (en) | 1990-01-23 |
| ZW13584A1 (en) | 1985-03-06 |
| US4748178A (en) | 1988-05-31 |
| DD222876A5 (de) | 1985-05-29 |
| AU583796B2 (en) | 1989-05-11 |
| ES535293A0 (es) | 1985-07-16 |
| PH23080A (en) | 1989-04-10 |
| EG17262A (en) | 1991-08-30 |
| MX160630A (es) | 1990-03-29 |
| HUT35653A (en) | 1985-07-29 |
| HU192991B (en) | 1987-08-28 |
| ES8601152A1 (es) | 1985-11-01 |
| DE3483294D1 (de) | 1990-10-31 |
| ES540040A0 (es) | 1985-11-01 |
| DK396384A (da) | 1985-02-20 |
| AU3204084A (en) | 1985-02-21 |
| GB2145087B (en) | 1987-02-04 |
| GB2145087A (en) | 1985-03-20 |
| EP0135155A3 (en) | 1986-01-02 |
| KR850001907A (ko) | 1985-04-10 |
| EP0135155A2 (de) | 1985-03-27 |
| IL72716A0 (en) | 1984-11-30 |
| MY101864A (en) | 1992-01-31 |
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