ES8305730A1 - Un procedimiento para la preparacion de un derivado del imidazol. - Google Patents
Un procedimiento para la preparacion de un derivado del imidazol.Info
- Publication number
- ES8305730A1 ES8305730A1 ES510875A ES510875A ES8305730A1 ES 8305730 A1 ES8305730 A1 ES 8305730A1 ES 510875 A ES510875 A ES 510875A ES 510875 A ES510875 A ES 510875A ES 8305730 A1 ES8305730 A1 ES 8305730A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- lower alkyl
- hydrogen
- compounds
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 230000000845 anti-microbial effect Effects 0.000 title abstract 2
- 150000002460 imidazoles Chemical class 0.000 title abstract 2
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 244000005700 microbiome Species 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Agronomy & Crop Science (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE IMIDAZOL SUS FORMAS ISOMERICAS POSIBLES SUS SALES DE ADICION DE ACIDO Y SUS COMPLEJOS DE SALES METALICAS, DE FORMULA (I), EN LA QUE N VALE 0-2; Y R , R , R , R Y R PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE TIOACETALIZACION DE UNA CETONA DE FORMULA (II), EN LA QUE R , R Y R TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I), O UN DERIVADO CETALICO ADECUADO, CON UN TIOL. LA REACCION SE LLEVA A CABO EN UN DISOLVENTE INERTE, EN PRESENCIA DE UN ACIDO DE LEWIS, A TEMPERATURAS ELEVADAS. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO AGENTES ANTIMICROBIANOS.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24859481A | 1981-03-27 | 1981-03-27 | |
| US06/342,553 US4483865A (en) | 1981-03-27 | 1982-01-25 | Antimicrobial imidazole derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8305730A1 true ES8305730A1 (es) | 1983-04-16 |
| ES510875A0 ES510875A0 (es) | 1983-04-16 |
Family
ID=26939447
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES510875A Granted ES510875A0 (es) | 1981-03-27 | 1982-03-26 | Un procedimiento para la preparacion de un derivado del imidazol. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4483865A (es) |
| EP (1) | EP0061794B1 (es) |
| AR (1) | AR230633A1 (es) |
| AU (1) | AU551590B2 (es) |
| BR (1) | BR8201733A (es) |
| CA (1) | CA1183855A (es) |
| DE (1) | DE3261889D1 (es) |
| DK (1) | DK140982A (es) |
| ES (1) | ES510875A0 (es) |
| GR (1) | GR70087B (es) |
| IL (1) | IL65353A (es) |
| PT (1) | PT74667B (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4489087A (en) * | 1982-10-13 | 1984-12-18 | Syntex (U.S.A.) Inc. | Spermicidal thioketal substituted N-alkyl imidazoles |
| US4870094A (en) * | 1984-05-02 | 1989-09-26 | Uniroyal Chemical Company, Inc. | Substituted imidazoles and triazoles |
| US4602030A (en) * | 1984-05-24 | 1986-07-22 | Chevron Research Company | Fungicidal 2-substituted-1-(1-imidazolyl)-propyl aryl sulfides, sulfoxides and sulfones |
| DE3587252T2 (de) * | 1985-10-09 | 1993-07-15 | Nihon Nohyaku Co Ltd | Keten-s,s,-acetalderivate, verfahren zu ihrer herstellung und methode zur heilung von mykose unter verwendung dieser derivate. |
| EP0218736B1 (en) * | 1985-10-10 | 1993-04-07 | Nihon Nohyaku Co., Ltd. | A ketene s,s-acetal derivative, a process for manufacturing thereof and a method for curing mycosis by administering it |
| US5502073A (en) * | 1987-06-05 | 1996-03-26 | The Wellcome Foundation | Heterocyclic pesticidal compounds |
| US4943311A (en) * | 1988-05-09 | 1990-07-24 | Uniroyal Chemical Company, Inc. | Azole derivatives of spiroheterocycles |
| GB9125791D0 (en) * | 1991-12-04 | 1992-02-05 | Schering Agrochemicals Ltd | Herbicides |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3193563A (en) * | 1963-05-24 | 1965-07-06 | Syntex Corp | Process for the preparation of steroidal ethers and thioethers |
| US3575999A (en) * | 1968-08-19 | 1971-04-20 | Janssen Pharmaceutica Nv | Ketal derivatives of imidazole |
| US4079062A (en) * | 1974-11-18 | 1978-03-14 | Janssen Pharmaceutica N.V. | Triazole derivatives |
| US4101664A (en) * | 1975-10-06 | 1978-07-18 | Janssen Pharmaceutica N.V. | 1-(2-Ar-4-aryloxymethyl-1,3-dioxolan-2-ylmethyl)-imidazoles |
| US4085209A (en) * | 1975-02-05 | 1978-04-18 | Rohm And Haas Company | Preparation and safening effect of 1-substituted imidazole metal salt complexes |
| US4055652A (en) * | 1975-07-07 | 1977-10-25 | Syntex (U.S.A.) Inc. | 1-[β(R-thio)phenethyl]imidazoles and derivatives thereof |
| US4078071A (en) * | 1976-03-08 | 1978-03-07 | Syntex (U.S.A.) Inc. | Derivatives of substituted N-alkyl imidazoles |
| US4150153A (en) * | 1977-05-13 | 1979-04-17 | Syntex (U.S.A.) Inc. | 1-(Naphthylethyl)imidazole derivatives |
| IT1160898B (it) * | 1977-11-04 | 1987-03-11 | Syntex Inc | Derivati dell'1-(naftiletil)-imidazolo,particolarmente utili come anticonvulsivi ed antisecretivi,e procedimento per la loro preparazione |
| US4359475A (en) * | 1981-12-21 | 1982-11-16 | Syntex (U.S.A.) Inc. | Thioketal substituted N-alkyl imidazoles |
-
1982
- 1982-01-25 US US06/342,553 patent/US4483865A/en not_active Expired - Fee Related
- 1982-02-25 CA CA000397116A patent/CA1183855A/en not_active Expired
- 1982-03-04 GR GR67479A patent/GR70087B/el unknown
- 1982-03-05 EP EP82200282A patent/EP0061794B1/en not_active Expired
- 1982-03-05 DE DE8282200282T patent/DE3261889D1/de not_active Expired
- 1982-03-25 IL IL65353A patent/IL65353A/xx unknown
- 1982-03-26 ES ES510875A patent/ES510875A0/es active Granted
- 1982-03-26 AU AU81972/82A patent/AU551590B2/en not_active Ceased
- 1982-03-26 DK DK140982A patent/DK140982A/da not_active Application Discontinuation
- 1982-03-26 BR BR8201733A patent/BR8201733A/pt unknown
- 1982-03-26 PT PT74667A patent/PT74667B/pt unknown
- 1982-03-26 AR AR288897A patent/AR230633A1/es active
Also Published As
| Publication number | Publication date |
|---|---|
| IL65353A0 (en) | 1982-05-31 |
| CA1183855A (en) | 1985-03-12 |
| BR8201733A (pt) | 1983-02-22 |
| EP0061794B1 (en) | 1985-01-16 |
| AR230633A1 (es) | 1984-05-31 |
| EP0061794A1 (en) | 1982-10-06 |
| AU8197282A (en) | 1982-09-30 |
| ES510875A0 (es) | 1983-04-16 |
| GR70087B (es) | 1982-07-30 |
| AU551590B2 (en) | 1986-05-08 |
| PT74667B (en) | 1985-05-31 |
| PT74667A (en) | 1982-04-01 |
| US4483865A (en) | 1984-11-20 |
| IL65353A (en) | 1985-04-30 |
| DK140982A (da) | 1982-09-28 |
| DE3261889D1 (en) | 1985-02-28 |
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