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ES8105262A1 - Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina. - Google Patents

Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina.

Info

Publication number
ES8105262A1
ES8105262A1 ES489469A ES489469A ES8105262A1 ES 8105262 A1 ES8105262 A1 ES 8105262A1 ES 489469 A ES489469 A ES 489469A ES 489469 A ES489469 A ES 489469A ES 8105262 A1 ES8105262 A1 ES 8105262A1
Authority
ES
Spain
Prior art keywords
biphenyl
production
preparations containing
containing same
cardiovascular preparations
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES489469A
Other languages
English (en)
Other versions
ES489469A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES489469A0 publication Critical patent/ES489469A0/es
Publication of ES8105262A1 publication Critical patent/ES8105262A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • C07C211/27Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring having amino groups linked to the six-membered aromatic ring by saturated carbon chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/092Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

PROCEDIMIENTO DE OBTENCION DE DERIVADOS DE 1,1''BIFENIL-2-IL-ALQUILAMINA. CONSISTE EN HACER REACCIONAR UNA CETONA DE FORMULA GENERAL (II) CON UN REACTIVO DE GRIGNARD DE FORMULA (III), OBTENIENDOSE DERIVADOS DE FORMULA GENERAL (I), EN QUE X ES HIDROGENO, R'' ES HIDROXI, R ELEVADO A 2 ES HIDROGENO O ALQUILO, Z ES -(CH2)N Y R ELEVADO A 4, R ELEVADO A 3 SON HIDROGENO, ALQUILO, CH2-ALQUENILO, FENILALQUILO. *FORMULA* QUIMIOTERAPIA DE ALTERACIONES CARDIOVASCULARES. R
ES489469A 1979-03-12 1980-03-12 Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina. Expired ES8105262A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1953479A 1979-03-12 1979-03-12

Publications (2)

Publication Number Publication Date
ES489469A0 ES489469A0 (es) 1981-05-16
ES8105262A1 true ES8105262A1 (es) 1981-05-16

Family

ID=21793713

Family Applications (6)

Application Number Title Priority Date Filing Date
ES489469A Expired ES8105262A1 (es) 1979-03-12 1980-03-12 Un procedimiento para la preparacion de 1, 1'-bifenil-2-il- alquilamina.
ES497208A Expired ES8201527A1 (es) 1979-03-12 1980-11-27 Un procedimiento para las preparaciones de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497206A Granted ES497206A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497209A Expired ES8201528A1 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497207A Granted ES497207A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-binefil-2-il-alquilamina
ES497210A Granted ES497210A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina

Family Applications After (5)

Application Number Title Priority Date Filing Date
ES497208A Expired ES8201527A1 (es) 1979-03-12 1980-11-27 Un procedimiento para las preparaciones de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497206A Granted ES497206A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497209A Expired ES8201528A1 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-bifenil-2-il-alquilamina
ES497207A Granted ES497207A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1,1'-binefil-2-il-alquilamina
ES497210A Granted ES497210A0 (es) 1979-03-12 1980-11-27 Un procedimiento para la preparacion de nuevos derivados de 1-1'-bifenil-2-il-alquilamina

Country Status (31)

Country Link
EP (1) EP0015776B1 (es)
JP (1) JPS55127347A (es)
KR (1) KR840000103B1 (es)
AR (1) AR228852A1 (es)
AT (1) AT367395B (es)
AU (1) AU528060B2 (es)
BE (1) BE882167A (es)
CA (1) CA1144926A (es)
CH (1) CH644094A5 (es)
CS (1) CS215052B2 (es)
DD (1) DD149664A5 (es)
DE (1) DE3060611D1 (es)
DK (1) DK103480A (es)
ES (6) ES8105262A1 (es)
FI (1) FI800736A7 (es)
FR (1) FR2451363A1 (es)
GB (1) GB2046256B (es)
GR (1) GR68036B (es)
HU (1) HU180334B (es)
IE (1) IE49552B1 (es)
IL (1) IL59557A (es)
IT (1) IT1140773B (es)
LU (1) LU82237A1 (es)
MX (1) MX6219E (es)
NZ (1) NZ193079A (es)
PH (1) PH14749A (es)
PL (1) PL121662B1 (es)
PT (1) PT70928A (es)
RO (1) RO79906A (es)
SU (2) SU940645A3 (es)
ZA (1) ZA801421B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100470454B1 (ko) * 2002-05-14 2005-02-05 대한민국 돼지 사료공급을 위한 자동조절급이기
EP1768951A4 (en) * 2004-06-17 2011-06-15 Musc Found For Res Dev NON-NATURAL AMINO ACIDS
ES2742261T3 (es) * 2011-04-15 2020-02-13 Hivih Inhibidores de la replicación viral, su proceso de preparación y sus usos terapéuticos
EP2821104A1 (en) 2013-07-05 2015-01-07 Laboratoire Biodim Inhibitors of viral replication, their process of preparation and their therapeutical uses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES236010A1 (es) * 1956-06-29 1957-12-16 Lab Pharmaceutica Dr C Janssen UN PROCEDIMIENTO PARA PREPARAR NUEVOS DERIVADOS PARASIMPATICOLiTICAMENTE ACTIVOS DE ALFAS-DEFENIL PROPANO
US3433836A (en) * 1966-01-14 1969-03-18 Rexall Drug Chemical Alpha-diaryl alpha,omega-alkylene glycol-dilower-alkylamines
GB1475314A (en) * 1973-11-02 1977-06-01 Cm Ind Phenyl-propylamine derivatives
IL48319A0 (en) * 1974-10-26 1975-12-31 Merck Patent Gmbh Araliphatic nitrogen compounds and a process for their preparation
GB1523655A (en) * 1975-02-10 1978-09-06 Armour Pharma 4-(4-biphenylyl) butylamines and treatment of the animal organism therewith

Also Published As

Publication number Publication date
IE800493L (en) 1980-09-12
BE882167A (fr) 1980-09-11
IL59557A (en) 1983-10-31
ES489469A0 (es) 1981-05-16
PT70928A (en) 1980-04-01
ES497208A0 (es) 1981-12-16
ES8201526A1 (es) 1981-12-16
EP0015776A1 (en) 1980-09-17
ES8201529A1 (es) 1981-12-16
IT8020503A0 (it) 1980-03-11
ES8201525A1 (es) 1981-12-16
AT367395B (de) 1982-06-25
JPS55127347A (en) 1980-10-02
DD149664A5 (de) 1981-07-22
ES497206A0 (es) 1981-12-16
ATA134580A (de) 1981-11-15
IL59557A0 (en) 1980-06-30
DK103480A (da) 1980-09-13
CA1144926A (en) 1983-04-19
MX6219E (es) 1984-12-21
NZ193079A (en) 1982-05-31
PL121662B1 (en) 1982-05-31
FI800736A7 (fi) 1981-01-01
GR68036B (es) 1981-10-27
CH644094A5 (fr) 1984-07-13
ES497207A0 (es) 1981-12-16
KR830001854A (ko) 1983-05-19
AU5630280A (en) 1980-09-18
IE49552B1 (en) 1985-10-30
SU1022655A3 (ru) 1983-06-07
IT1140773B (it) 1986-10-10
HU180334B (en) 1983-02-28
KR840000103B1 (ko) 1984-02-11
ES497210A0 (es) 1981-12-16
ZA801421B (en) 1981-10-28
RO79906A (ro) 1982-10-11
ES497209A0 (es) 1981-12-16
ES8201528A1 (es) 1981-12-16
EP0015776B1 (en) 1982-06-30
CS215052B2 (en) 1982-07-30
PH14749A (en) 1981-11-20
AU528060B2 (en) 1983-04-14
DE3060611D1 (en) 1982-08-19
GB2046256A (en) 1980-11-12
FR2451363B1 (es) 1983-01-14
ES8201527A1 (es) 1981-12-16
LU82237A1 (fr) 1980-06-06
PL222601A1 (es) 1981-01-30
GB2046256B (en) 1983-04-20
AR228852A1 (es) 1983-04-29
SU940645A3 (ru) 1982-06-30
FR2451363A1 (fr) 1980-10-10

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19980202