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ES557808A0 - Un procedimiento para preparar derivados de octahidro(f) quinoleina - Google Patents

Un procedimiento para preparar derivados de octahidro(f) quinoleina

Info

Publication number
ES557808A0
ES557808A0 ES557808A ES557808A ES557808A0 ES 557808 A0 ES557808 A0 ES 557808A0 ES 557808 A ES557808 A ES 557808A ES 557808 A ES557808 A ES 557808A ES 557808 A0 ES557808 A0 ES 557808A0
Authority
ES
Spain
Prior art keywords
quinoleina
octahidro
procedure
preparing derivatives
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES557808A
Other languages
English (en)
Other versions
ES8900136A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of ES557808A0 publication Critical patent/ES557808A0/es
Publication of ES8900136A1 publication Critical patent/ES8900136A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • C07D221/06Ring systems of three rings
    • C07D221/10Aza-phenanthrenes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
ES557808A 1983-04-27 1988-01-26 Un procedimiento para preparar derivados de octahidro(f) quinoleina Expired ES8900136A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE8302361A SE8302361D0 (sv) 1983-04-27 1983-04-27 New tricyclic amines

Publications (2)

Publication Number Publication Date
ES557808A0 true ES557808A0 (es) 1989-01-16
ES8900136A1 ES8900136A1 (es) 1989-01-16

Family

ID=20350972

Family Applications (5)

Application Number Title Priority Date Filing Date
ES531931A Granted ES531931A0 (es) 1983-04-27 1984-04-26 Un procedimiento para preparar un derivado de octahidro-benzo (f) quinoleina
ES540003A Expired ES8609258A1 (es) 1983-04-27 1985-01-31 Un procedimiento para preparar un derivado de octahidrobenzo(f) quinoleina
ES552962A Expired ES8801634A1 (es) 1983-04-27 1986-03-13 Un procedimiento para preparar un derivado de octahidro-benzo(f)quinoleina
ES557649A Expired ES8802032A1 (es) 1983-04-27 1987-08-01 Un procedimiento para preparar un derivado de octahidrobenzo (f)quinoleina
ES557808A Expired ES8900136A1 (es) 1983-04-27 1988-01-26 Un procedimiento para preparar derivados de octahidro(f) quinoleina

Family Applications Before (4)

Application Number Title Priority Date Filing Date
ES531931A Granted ES531931A0 (es) 1983-04-27 1984-04-26 Un procedimiento para preparar un derivado de octahidro-benzo (f) quinoleina
ES540003A Expired ES8609258A1 (es) 1983-04-27 1985-01-31 Un procedimiento para preparar un derivado de octahidrobenzo(f) quinoleina
ES552962A Expired ES8801634A1 (es) 1983-04-27 1986-03-13 Un procedimiento para preparar un derivado de octahidro-benzo(f)quinoleina
ES557649A Expired ES8802032A1 (es) 1983-04-27 1987-08-01 Un procedimiento para preparar un derivado de octahidrobenzo (f)quinoleina

Country Status (22)

Country Link
US (1) US4612316A (es)
EP (2) EP0127597B1 (es)
JP (1) JPS60501157A (es)
KR (1) KR910007239B1 (es)
AU (1) AU572840B2 (es)
CA (1) CA1264749A (es)
DD (1) DD216716A5 (es)
DE (1) DE3479724D1 (es)
DK (1) DK159848C (es)
ES (5) ES531931A0 (es)
FI (1) FI82930C (es)
GB (1) GB2138815B (es)
GR (1) GR81994B (es)
HU (1) HU193576B (es)
IE (1) IE57883B1 (es)
IS (1) IS1365B6 (es)
NZ (1) NZ207881A (es)
PH (1) PH24764A (es)
PT (1) PT78512B (es)
SE (1) SE8302361D0 (es)
WO (1) WO1984004303A1 (es)
ZA (1) ZA842539B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8302361D0 (sv) * 1983-04-27 1983-04-27 Astra Laekemedel Ab New tricyclic amines
US4764609A (en) * 1986-03-31 1988-08-16 Eli Lilly And Company Synthesis of 2-aminopyrimido[4,5-g]quinolines
JPH0249772A (ja) * 1988-04-07 1990-02-20 Glaxo Group Ltd イミダゾール誘導体
GR1001059B (el) * 1988-12-15 1993-04-28 Abbott Lab Μεθοδος παραγωγης εκλεκτικων παραγοντων 5-ητ.
JPH03502701A (ja) * 1988-12-15 1991-06-20 アボツト・ラボラトリーズ 5‐ht選択性物質
CA2011640A1 (en) * 1989-03-20 1990-09-20 Rene Imhof Quinoline derivatives
US5486611A (en) * 1989-07-13 1996-01-23 The Upjohn Company Carboxamido-(1,2N)-carbocyclic-2-aminotetralin derivatives
CA2057912C (en) * 1989-07-13 1996-10-29 Chiu-Hong Lin (1,2n) and (3,2n)-carbocyclic-2-amino tetralin derivatives
GB8917333D0 (en) * 1989-07-28 1989-09-13 Merck Sharp & Dohme Therapeutic agents
US5294618A (en) * 1989-07-28 1994-03-15 Merck Sharp & Dohme Limited Octahydrobenzisoquinoline derivatives as antipsychotic agents
DE3930282A1 (de) * 1989-09-11 1991-03-21 Boehringer Ingelheim Kg Verwendung von dopamin-autorezeptor-agonisten bei der behandlung von drogenabhaengigkeit
US5244888A (en) * 1989-11-17 1993-09-14 Abbott Laboratories 5-HT selective agents
WO1992020655A1 (en) * 1991-05-20 1992-11-26 The Upjohn Company Carboxamido-(1,2n)-carbocyclic-2-aminotetralin derivatives
ES2169026T3 (es) * 1991-08-21 2002-07-01 Lilly Co Eli Benzo(f)quinolinonas como inhibidores de 5-alfa-reductasa.
US5239075A (en) * 1991-08-21 1993-08-24 Eli Lilly And Company Process for the preparation of benzo (f) quinolinones
TW239127B (es) * 1991-12-20 1995-01-21 Hoffmann La Roche
JPH09509398A (ja) * 1993-11-19 1997-09-22 ザ ボード オブ ガヴァナーズ フォー ハイアー エデュケーション,ステイト オブ ロードアイランド アンド プロヴィデンス プランテーションズ オクタヒドロベンゾ[f]キノリン系受容体アゴニストおよびアンタゴニスト
US5863928A (en) 1993-11-19 1999-01-26 The Board Of Governors For Higher Education The State Of Rhode Island And Providence Plantation. Octahydrobenzo f!quinoline-based receptor agonists and antagonists
US5578724A (en) * 1994-09-20 1996-11-26 Eli Lilly And Company Process for preparation of benzo[f]quinolinones
GB9612153D0 (en) * 1996-06-11 1996-08-14 Smithkline Beecham Plc Compounds
EP1655301B1 (en) * 2003-08-04 2015-03-11 Valery Khazhmuratovich Zhilov Cyclic bioisosters of purine system derivatives and a pharmaceutical composition based thereon
RU2326870C2 (ru) * 2003-08-04 2008-06-20 Валерий Хажмуратович ЖИЛОВ Применение циклических биоизостеров производных пуриновой системы для лечения расстройств, вызванных нарушениями нитрергической и дофаминергической систем

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2486440A (en) * 1946-01-10 1949-11-01 Gen Aniline & Film Corp Production of phenazonium dyestuff images
GB1277789A (en) * 1969-09-08 1972-06-14 Logeais Labor Jacques Improvements in or relating to new polycyclic pyrrole derivatives
CH630902A5 (en) * 1977-01-24 1982-07-15 Sandoz Ag Process for preparing novel derivatives of 1,2,3,4,4a,10b-hexahydrobenzo(f)isoquinoline.
US4341786A (en) * 1981-03-02 1982-07-27 Smithkline Corporation Pharmaceutical compositions and method of producing central alpha1 agonist activity utilizing octahydrobenzo[f]quinoline compounds
PT77267B (en) * 1982-09-07 1986-03-21 Lilly Co Eli Improved process for preparing novel octahydrobenz <f> isoquinolines or compounds relating thereto
SE8302361D0 (sv) * 1983-04-27 1983-04-27 Astra Laekemedel Ab New tricyclic amines

Also Published As

Publication number Publication date
SE8302361D0 (sv) 1983-04-27
DK620784A (da) 1984-12-21
PT78512A (en) 1984-05-01
PH24764A (en) 1990-10-01
DD216716A5 (de) 1984-12-19
HU193576B (en) 1987-10-28
WO1984004303A1 (en) 1984-11-08
JPH0552309B2 (es) 1993-08-05
EP0127597A1 (en) 1984-12-05
US4612316A (en) 1986-09-16
ES552962A0 (es) 1988-02-16
FI852091L (fi) 1985-05-24
DK159848B (da) 1990-12-17
FI82930B (fi) 1991-01-31
AU572840B2 (en) 1988-05-19
JPS60501157A (ja) 1985-07-25
DE3479724D1 (de) 1989-10-19
IS2906A7 (is) 1984-10-28
IE840908L (en) 1984-10-27
HUT38616A (en) 1986-06-30
CA1264749A (en) 1990-01-23
GB2138815B (en) 1987-07-29
EP0172821A1 (en) 1986-03-05
ES8505957A1 (es) 1985-06-16
ES531931A0 (es) 1985-06-16
PT78512B (en) 1986-07-22
ES8801634A1 (es) 1988-02-16
GB2138815A (en) 1984-10-31
ES8609258A1 (es) 1986-09-01
GB8410624D0 (en) 1984-05-31
ES8900136A1 (es) 1989-01-16
EP0127597B1 (en) 1989-06-28
NZ207881A (en) 1987-08-31
ES540003A0 (es) 1986-09-01
ES557649A0 (es) 1988-03-16
ZA842539B (en) 1984-12-24
DK620784D0 (da) 1984-12-21
FI82930C (fi) 1991-05-10
KR840008325A (ko) 1984-12-14
FI852091A0 (fi) 1985-05-24
IE57883B1 (en) 1993-05-05
GR81994B (es) 1984-12-12
EP0172821B1 (en) 1989-09-13
KR910007239B1 (ko) 1991-09-24
IS1365B6 (is) 1989-05-25
AU2866784A (en) 1984-11-19
ES8802032A1 (es) 1988-03-16
DK159848C (da) 1991-05-13

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20010402