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ES548135A0 - Un procedimiento para preparar dioxafosforinanos - Google Patents

Un procedimiento para preparar dioxafosforinanos

Info

Publication number
ES548135A0
ES548135A0 ES548135A ES548135A ES548135A0 ES 548135 A0 ES548135 A0 ES 548135A0 ES 548135 A ES548135 A ES 548135A ES 548135 A ES548135 A ES 548135A ES 548135 A0 ES548135 A0 ES 548135A0
Authority
ES
Spain
Prior art keywords
dioxaphosphorinans
preparing
procedure
preparing dioxaphosphorinans
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES548135A
Other languages
English (en)
Other versions
ES8701187A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
OCE-Andeno BV
Oce Andeno BV
Original Assignee
OCE-Andeno BV
Oce Andeno BV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by OCE-Andeno BV, Oce Andeno BV filed Critical OCE-Andeno BV
Publication of ES8701187A1 publication Critical patent/ES8701187A1/es
Publication of ES548135A0 publication Critical patent/ES548135A0/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6571Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
    • C07F9/6574Esters of oxyacids of phosphorus
    • C07F9/65744Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6571Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
    • C07F9/6574Esters of oxyacids of phosphorus
    • C07F9/65742Esters of oxyacids of phosphorus non-condensed with carbocyclic rings or heterocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES548135A 1984-10-24 1985-10-23 Un procedimiento para preparar dioxafosforinanos Expired ES8701187A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
NL8403224A NL8403224A (nl) 1984-10-24 1984-10-24 Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen.

Publications (2)

Publication Number Publication Date
ES8701187A1 ES8701187A1 (es) 1986-11-16
ES548135A0 true ES548135A0 (es) 1986-11-16

Family

ID=19844654

Family Applications (2)

Application Number Title Priority Date Filing Date
ES548135A Expired ES8701187A1 (es) 1984-10-24 1985-10-23 Un procedimiento para preparar dioxafosforinanos
ES554328A Expired ES8704504A1 (es) 1984-10-24 1986-04-24 Un procedimiento para preparar isomeros opticamente activos de dioxafosforinanos

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES554328A Expired ES8704504A1 (es) 1984-10-24 1986-04-24 Un procedimiento para preparar isomeros opticamente activos de dioxafosforinanos

Country Status (6)

Country Link
US (1) US4814477A (es)
EP (1) EP0180276B1 (es)
JP (1) JPH0662652B2 (es)
DE (1) DE3567022D1 (es)
ES (2) ES8701187A1 (es)
NL (1) NL8403224A (es)

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US7205404B1 (en) 1999-03-05 2007-04-17 Metabasis Therapeutics, Inc. Phosphorus-containing prodrugs
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ATE414070T1 (de) 2000-12-28 2008-11-15 Takeda Pharmaceutical Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen
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US7214668B2 (en) 2002-05-13 2007-05-08 Metabasis Therapeutics, Inc. Phosphonic acid based prodrugs of PMEA and its analogues
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CN1678326A (zh) * 2002-06-28 2005-10-05 埃迪尼克斯(开曼)有限公司 用于治疗黄病毒感染的2'-c-甲基-3'-o-l-缬氨酸酯核糖呋喃基胞苷
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US7964580B2 (en) 2007-03-30 2011-06-21 Pharmasset, Inc. Nucleoside phosphoramidate prodrugs
MX2009013402A (es) 2007-06-13 2010-02-24 Incyte Corp Sales de inhibidor de janus cinasa (r)-3-(4-(7h-pirrolo[2,3-d]piri midin-4-il)-1h-pirazol-1-il)-3-ciclopentilpropanitrilo.
EP3042660A3 (en) 2008-04-15 2016-10-26 RFS Pharma, LLC. Nucleoside derivatives for treatment of caliciviridae infections, including norovirus infections
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TW201113285A (en) * 2009-09-01 2011-04-16 Incyte Corp Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
CN101792398B (zh) * 2010-03-09 2013-06-26 河北科技大学 一种拆分法制备光学纯对羟基苯甘氨酸的方法
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US8563530B2 (en) 2010-03-31 2013-10-22 Gilead Pharmassel LLC Purine nucleoside phosphoramidate
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UA111854C2 (uk) 2011-09-07 2016-06-24 Інсайт Холдінгс Корпорейшн Способи і проміжні сполуки для отримання інгібіторів jak
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PL2919766T3 (pl) 2012-11-15 2021-10-04 Incyte Holdings Corporation Postacie dawkowania ruksolitynibu o przedłużonym uwalnianiu
CN103232491B (zh) * 2013-02-01 2016-06-15 河北科技大学 一种手性环磷酸的制备方法
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Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT951631B (it) * 1971-03-18 1973-07-10 Richardson Merrell Spa Composti utili per la separazione di isomeri ottici geometrici e strutturali e relativo procedimen to di sintesi
NL8403224A (nl) * 1984-10-24 1986-05-16 Oce Andeno Bv Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen.

Also Published As

Publication number Publication date
NL8403224A (nl) 1986-05-16
JPH0662652B2 (ja) 1994-08-17
ES8704504A1 (es) 1987-04-01
DE3567022D1 (en) 1989-02-02
EP0180276B1 (en) 1988-12-28
JPS61103886A (ja) 1986-05-22
ES8701187A1 (es) 1986-11-16
US4814477A (en) 1989-03-21
EP0180276A1 (en) 1986-05-07
ES554328A0 (es) 1987-04-01

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970303