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ES525656A0 - Un metodo de preparar profarmacos de pilocarpina - Google Patents

Un metodo de preparar profarmacos de pilocarpina

Info

Publication number
ES525656A0
ES525656A0 ES525656A ES525656A ES525656A0 ES 525656 A0 ES525656 A0 ES 525656A0 ES 525656 A ES525656 A ES 525656A ES 525656 A ES525656 A ES 525656A ES 525656 A0 ES525656 A0 ES 525656A0
Authority
ES
Spain
Prior art keywords
pilocarpine
drugs
preparing
preparing pilocarpine
pilocarpine drugs
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES525656A
Other languages
English (en)
Other versions
ES8502977A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
FALCH ERIK
Original Assignee
FALCH ERIK
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by FALCH ERIK filed Critical FALCH ERIK
Publication of ES8502977A1 publication Critical patent/ES8502977A1/es
Publication of ES525656A0 publication Critical patent/ES525656A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
ES525656A 1982-09-17 1983-09-16 Un metodo de preparar profarmacos de pilocarpina Granted ES525656A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK417082 1982-09-17

Publications (2)

Publication Number Publication Date
ES8502977A1 ES8502977A1 (es) 1985-02-01
ES525656A0 true ES525656A0 (es) 1985-02-01

Family

ID=8130941

Family Applications (1)

Application Number Title Priority Date Filing Date
ES525656A Granted ES525656A0 (es) 1982-09-17 1983-09-16 Un metodo de preparar profarmacos de pilocarpina

Country Status (10)

Country Link
US (1) US4742073A (es)
EP (1) EP0106541A3 (es)
JP (1) JPS59130275A (es)
KR (1) KR840006213A (es)
AU (1) AU557083B2 (es)
CA (1) CA1235416A (es)
ES (1) ES525656A0 (es)
IL (1) IL69593A (es)
NZ (1) NZ205617A (es)
PT (1) PT77347B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL69593A (en) * 1982-09-17 1988-09-30 Bundegaard Hans Pilocarpine prodrugs,their preparation and pharmaceutical compositions containing them
DK406686D0 (da) * 1986-08-26 1986-08-26 Hans Bundgaard Carboxylsyrederivater
US5066663A (en) * 1990-05-21 1991-11-19 Warner-Lambert Company Substituted-hetero-cyclopentanones and cyclopentenones and derivatives thereof acting at muscarinic receptors
US5066665A (en) * 1990-05-21 1991-11-19 Warner-Lambert Co. Substituted isoxazolidin-3-ones and derivatives thereof acting at muscarinic receptors
FI98815C (fi) * 1990-11-30 1997-08-25 Santen Oy Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi
FI98910C (fi) 1992-05-29 1997-09-10 Santen Oy Menetelmä farmaseuttisesti käyttökelpoisten pilokarpiinijohdannaisten valmistamiseksi
US5436350A (en) * 1990-11-30 1995-07-25 Jaervinen; Tomi Bispilocarpic acid ester derivatives and process for their preparation
WO1993024466A1 (en) * 1992-05-29 1993-12-09 Leiras Oy Novel pilocarpine derivatives and process for their preparation
US5521210A (en) * 1993-04-13 1996-05-28 Allergan, Inc. Ophthalmic use of muscarinic agonists having increased duration of activity
CN115536641B (zh) * 2022-09-29 2024-12-27 广州润尔眼科生物科技有限公司 一种内酯化合物及其制备方法与应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3470197A (en) * 1967-08-30 1969-09-30 Miles Lab 1-substituted derivatives of 3-ethyl-4 - (1-methylimidazolyl-(5)-methyl)-2-pyrrolidinone
US3631059A (en) * 1967-09-11 1971-12-28 John T Goorley Process for the extraction and purification of pilocarpine
US4045558A (en) * 1975-10-08 1977-08-30 Merck & Co., Inc. Pilocarpine salts
US4061722A (en) * 1976-04-26 1977-12-06 Interx Research Corporation Selected quaternary ammonium salts of pilocarpine useful in reducing intraocular pressure in warm-blooded animals
IL69593A (en) * 1982-09-17 1988-09-30 Bundegaard Hans Pilocarpine prodrugs,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
JPS59130275A (ja) 1984-07-26
EP0106541A2 (en) 1984-04-25
CA1235416A (en) 1988-04-19
KR840006213A (ko) 1984-11-22
PT77347A (en) 1983-10-01
NZ205617A (en) 1986-06-11
ES8502977A1 (es) 1985-02-01
US4742073A (en) 1988-05-03
PT77347B (en) 1986-03-11
IL69593A (en) 1988-09-30
AU557083B2 (en) 1986-12-04
EP0106541A3 (en) 1985-12-18
AU1849483A (en) 1984-03-22

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