ES518290A0 - Un procedimiento para la preparacion de un derivado de 4a-9b-trans-hexahidro-1h-piridoindol enantiomerico (+) o racemico(+-) - Google Patents

Un procedimiento para la preparacion de un derivado de 4a-9b-trans-hexahidro-1h-piridoindol enantiomerico (+) o racemico(+-)

Info

Publication number: ES518290A0
Authority: ES; Spain
Prior art keywords: racemico; piridoindol; enantiomerico; hexahidro; trans
Prior art date: 1981-01-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES518290A

Other languages

English (en)

Other versions

ES8405002A1 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Corp Belgium

Pfizer Corp SRL

Original Assignee

Pfizer Corp Belgium

Pfizer Corp SRL

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-01-16

Filing date

1982-12-16

Publication date

1984-05-16

1982-12-16 Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium

1984-05-16 Publication of ES8405002A1 publication Critical patent/ES8405002A1/es

1984-05-16 Publication of ES518290A0 publication Critical patent/ES518290A0/es

Status Granted legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Life Sciences & Earth Sciences (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Neurology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Anesthesiology (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

ES518290A 1981-01-16 1982-12-16 Un procedimiento para la preparacion de un derivado de 4a-9b-trans-hexahidro-1h-piridoindol enantiomerico (+) o racemico(+-) Granted ES518290A0 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/225,569 US4337250A (en)	1979-07-30	1981-01-16	Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents

Publications (2)

Publication Number	Publication Date
ES8405002A1 ES8405002A1 (es)	1984-05-16
ES518290A0 true ES518290A0 (es)	1984-05-16

Family

ID=22845384

Family Applications (11)

Application Number	Title	Priority Date	Filing Date
ES508809A Expired ES8304966A1 (es)	1981-01-16	1982-01-15	Un procediemento para la preparacion de un derivado de piridoindol.
ES518291A Granted ES518291A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518297A Expired ES8405391A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de tetrahidro-1h-piridoindol.
ES518295A Granted ES518295A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518288A Expired ES8401962A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518293A Granted ES518293A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518289A Granted ES518289A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518292A Granted ES518292A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518290A Granted ES518290A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de 4a-9b-trans-hexahidro-1h-piridoindol enantiomerico (+) o racemico(+-)
ES518296A Granted ES518296A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518294A Expired ES8405003A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.

Family Applications Before (8)

Application Number	Title	Priority Date	Filing Date
ES508809A Expired ES8304966A1 (es)	1981-01-16	1982-01-15	Un procediemento para la preparacion de un derivado de piridoindol.
ES518291A Granted ES518291A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518297A Expired ES8405391A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de tetrahidro-1h-piridoindol.
ES518295A Granted ES518295A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518288A Expired ES8401962A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518293A Granted ES518293A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518289A Granted ES518289A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518292A Granted ES518292A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
ES518296A Granted ES518296A0 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.
ES518294A Expired ES8405003A1 (es)	1981-01-16	1982-12-16	Un procedimiento para la preparacion de un derivado de piridoindol.

Country Status (27)

Country	Link
US (1)	US4337250A (es)
EP (1)	EP0060610B1 (es)
JP (2)	JPS57139078A (es)
KR (1)	KR860001819B1 (es)
AR (1)	AR230283A1 (es)
AT (1)	ATE15372T1 (es)
AU (1)	AU528710B2 (es)
CA (1)	CA1177830A (es)
CS (1)	CS248020B2 (es)
DD (3)	DD222027A5 (es)
DE (1)	DE3265922D1 (es)
DK (1)	DK15282A (es)
EG (1)	EG15796A (es)
ES (11)	ES8304966A1 (es)
FI (1)	FI71936C (es)
GR (1)	GR74757B (es)
HU (1)	HU189090B (es)
IE (1)	IE51954B1 (es)
IL (1)	IL64774A (es)
NO (1)	NO159090C (es)
NZ (1)	NZ199473A (es)
PH (1)	PH19614A (es)
PL (2)	PL138924B1 (es)
PT (1)	PT74283A (es)
SU (2)	SU1179930A3 (es)
YU (1)	YU45854B (es)
ZA (1)	ZA82264B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4672117A (en) *	1985-09-16	1987-06-09	American Home Products Corporation	Antipsychotic gamma-carbolines
US4636563A (en) *	1985-09-16	1987-01-13	American Home Products Corporation	Antipsychotic γ-carbolines
US4732984A (en) *	1985-10-17	1988-03-22	American Home Products Corporation	Piperazinoisothiazolones with psychotropic activity
US4748182A (en) *	1986-03-05	1988-05-31	Merrell Dow Pharmaceuticals Inc.	Aromatic 2-aminoalkyl-1,2-benzoisothiazol-3(2H)one-1,1-dioxide derivatives and their use as anti-hypertensive and anxiolytic agents
JPH01140486A (ja) *	1987-11-27	1989-06-01	Hitachi Ltd	ブロッホラインメモリ駆動回路
FR2661177A1 (fr) *	1990-04-23	1991-10-25	Rhone Poulenc Sante	Derives du naphtosultame antagonistes de la serotonine, leur preparation et les medicaments les contenant.
TW470745B (en) *	1996-05-23	2002-01-01	Janssen Pharmaceutica Nv	Hexahydro-pyrido[4,3-b]indole derivatives
US5879444A (en) *	1997-09-02	1999-03-09	Bayer Corporation	Organic pigment compositions
DE60206636T2 (de)	2001-08-08	2006-06-22	Pharmacia & Upjohn Co. Llc, Kalamazoo	THERAPEUTISCHE 1H-PYRIDO[4,3-b]INDOLE
US20140206667A1 (en)	2012-11-14	2014-07-24	Michela Gallagher	Methods and compositions for treating schizophrenia

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3687961A (en) *	1971-05-03	1972-08-29	Abbott Lab	8-fluoro-2-{8 3-(4-fluorophenylanilinopropyl{9 -gamma-carboline
AR205452A1 (es) *	1973-12-06	1976-05-07	Endo Lab	Metodo para preparar nuevos trans-2, 3, 4, 4a, 5, 9b-hexahidro-5-fenil-1h-pirido(4,3-b) indoles
JPS50126699A (es) *	1974-03-20	1975-10-04
US4001263A (en) *	1974-04-01	1977-01-04	Pfizer Inc.	5-Aryl-1,2,3,4-tetrahydro-γ-carbolines
SE7702301L (sv) *	1976-04-08	1977-10-09	Endo Lab	Trans-hexahydro-pyrido-indoler
US4224329A (en) *	1979-01-23	1980-09-23	Pfizer Inc.	2-Substituted-trans-5-aryl-2,3,4,4a,5,9b-hexahydro-1H-pyrido[4,3-b]indoles
US4252811A (en) *	1979-07-30	1981-02-24	Pfizer Inc.	Hexahydro-trans-pyridoindole neuroleptic agents

1981
- 1981-01-16 US US06/225,569 patent/US4337250A/en not_active Expired - Lifetime
1982
- 1982-01-12 JP JP57003237A patent/JPS57139078A/ja active Granted
- 1982-01-12 NZ NZ199473A patent/NZ199473A/en unknown
- 1982-01-14 AT AT82300200T patent/ATE15372T1/de not_active IP Right Cessation
- 1982-01-14 EP EP82300200A patent/EP0060610B1/en not_active Expired
- 1982-01-14 CA CA000394123A patent/CA1177830A/en not_active Expired
- 1982-01-14 IL IL64774A patent/IL64774A/xx unknown
- 1982-01-14 DE DE8282300200T patent/DE3265922D1/de not_active Expired
- 1982-01-14 GR GR67010A patent/GR74757B/el unknown
- 1982-01-14 IE IE61/82A patent/IE51954B1/en unknown
- 1982-01-15 DD DD82265316A patent/DD222027A5/de unknown
- 1982-01-15 PH PH26744A patent/PH19614A/en unknown
- 1982-01-15 SU SU823384201A patent/SU1179930A3/ru active
- 1982-01-15 KR KR8200154A patent/KR860001819B1/ko not_active Expired
- 1982-01-15 DD DD82250220A patent/DD211348A5/de unknown
- 1982-01-15 DK DK15282A patent/DK15282A/da not_active Application Discontinuation
- 1982-01-15 HU HU82117A patent/HU189090B/hu unknown
- 1982-01-15 ZA ZA82264A patent/ZA82264B/xx unknown
- 1982-01-15 FI FI820138A patent/FI71936C/fi not_active IP Right Cessation
- 1982-01-15 NO NO820112A patent/NO159090C/no unknown
- 1982-01-15 AU AU79552/82A patent/AU528710B2/en not_active Ceased
- 1982-01-15 DD DD82236804A patent/DD208980A5/de unknown
- 1982-01-15 ES ES508809A patent/ES8304966A1/es not_active Expired
- 1982-01-15 YU YU9882A patent/YU45854B/sh unknown
- 1982-01-15 PT PT74283A patent/PT74283A/pt unknown
- 1982-01-16 EG EG18/82A patent/EG15796A/xx active
- 1982-01-18 CS CS82344A patent/CS248020B2/cs unknown
- 1982-02-22 PL PL1982241179A patent/PL138924B1/pl unknown
- 1982-02-22 PL PL1982235180A patent/PL137682B1/pl unknown
- 1982-10-05 AR AR290872A patent/AR230283A1/es active
- 1982-12-15 SU SU823521750A patent/SU1152522A3/ru active
- 1982-12-16 ES ES518291A patent/ES518291A0/es active Granted
- 1982-12-16 ES ES518297A patent/ES8405391A1/es not_active Expired
- 1982-12-16 ES ES518295A patent/ES518295A0/es active Granted
- 1982-12-16 ES ES518288A patent/ES8401962A1/es not_active Expired
- 1982-12-16 ES ES518293A patent/ES518293A0/es active Granted
- 1982-12-16 ES ES518289A patent/ES518289A0/es active Granted
- 1982-12-16 ES ES518292A patent/ES518292A0/es active Granted
- 1982-12-16 ES ES518290A patent/ES518290A0/es active Granted
- 1982-12-16 ES ES518296A patent/ES518296A0/es active Granted
- 1982-12-16 ES ES518294A patent/ES8405003A1/es not_active Expired
1985
- 1985-02-12 JP JP60025100A patent/JPS60185780A/ja active Pending

Also Published As

Publication number	Publication date
ES8401963A1 (es)	1984-01-01
EG15796A (en)	1986-12-30
FI71936B (fi)	1986-11-28
DD211348A5 (de)	1984-07-11
ES8405617A1 (es)	1984-06-16
ES508809A0 (es)	1983-03-16
US4337250A (en)	1982-06-29
AR230283A1 (es)	1984-03-01
SU1152522A3 (en)	1985-04-23
ATE15372T1 (de)	1985-09-15
CA1177830A (en)	1984-11-13
DK15282A (da)	1982-08-27
AU7955282A (en)	1982-07-22
ES518292A0 (es)	1984-01-01
KR860001819B1 (ko)	1986-10-24
ES8401964A1 (es)	1984-01-01
ES518297A0 (es)	1984-06-01
ES8405785A1 (es)	1984-06-16
PL137682B1 (en)	1986-07-31
SU1179930A3 (ru)	1985-09-15
JPS6130674B2 (es)	1986-07-15
PL235180A1 (en)	1983-11-21
PL241179A1 (en)	1984-03-26
FI71936C (fi)	1987-03-09
YU45854B (sh)	1992-09-07
JPS60185780A (ja)	1985-09-21
IL64774A0 (en)	1982-03-31
ES8304966A1 (es)	1983-03-16
ES8405391A1 (es)	1984-06-01
NZ199473A (en)	1985-10-11
EP0060610B1 (en)	1985-09-04
NO159090B (no)	1988-08-22
ES518288A0 (es)	1984-01-01
PH19614A (en)	1986-05-30
DE3265922D1 (en)	1985-10-10
EP0060610A1 (en)	1982-09-22
ES518293A0 (es)	1984-06-16
IE51954B1 (en)	1987-04-29
ZA82264B (en)	1982-12-29
CS248020B2 (en)	1987-01-15
ES518294A0 (es)	1984-05-16
HU189090B (en)	1986-06-30
FI820138L (fi)	1982-07-17
ES8401962A1 (es)	1984-01-01
JPS57139078A (en)	1982-08-27
ES8405002A1 (es)	1984-05-16
PT74283A (pt)	1982-02-01
ES8404851A1 (es)	1984-05-16
IE820061L (en)	1982-07-16
ES8405003A1 (es)	1984-05-16
IL64774A (en)	1985-06-30
DD222027A5 (de)	1985-05-08
ES8401965A1 (es)	1984-01-01
PL138924B1 (en)	1986-11-29
DD208980A5 (de)	1984-04-18
ES518291A0 (es)	1984-06-16
ES518296A0 (es)	1984-01-01
ES518295A0 (es)	1984-01-01
NO159090C (no)	1988-11-30
YU9882A (en)	1986-04-30
ES518289A0 (es)	1984-05-16
AU528710B2 (en)	1983-05-12
NO820112L (no)	1982-07-19
GR74757B (es)	1984-07-11
KR830009095A (ko)	1983-12-17

Publication	Publication Date	Title
ES528142A0 (es)	1986-04-16	Procedimiento para la obtencion de compuestos de hexapiranosa
ES529349A0 (es)	1985-08-01	Un procedimiento para la preparacion de derivados de acilmorfinano
ES524922A0 (es)	1984-05-16	Un procedimiento para la preparacion de nuevos derivados de 3-amino-pregn-5-eno
MX7419E (es)	1988-10-18	Procedimiento para la preparacion de pss-asa
MX157607A (es)	1988-12-05	Procedimiento para la preparacion de ciclohexilamina
ES536982A0 (es)	1985-07-01	Un procedimiento para la preparacion de un derivado de carbostirilo
AR231288A1 (es)	1984-10-31	Procedimiento para la preparacion de 3-amido-n-/2-5-dimetilaminometil-furan-2-il-metiltio etil-benzamidas
ES518290A0 (es)	1984-05-16	Un procedimiento para la preparacion de un derivado de 4a-9b-trans-hexahidro-1h-piridoindol enantiomerico (+) o racemico(+-)
ES518347A0 (es)	1984-08-01	Un procedimiento para la preparacion de derivados de desoxiuridina
ES526149A0 (es)	1985-04-16	Un procedimiento para la preparacion de derivados de espirotiazolidinil-piperazina
ES503565A0 (es)	1982-05-16	Un procedimiento para la preparacion de tilactona o un esterderivado de la misma
AR229712A1 (es)	1983-10-31	Procedimiento para la preparacion de 2-hidroximetil-3-hidroxi-6-(1-hidroxi-6-(hidroxi-2-t-butilaminoetil)piridina
AR229890A1 (es)	1983-12-30	Procedimiento para la preparacion de 1-carvona
ES544214A0 (es)	1987-05-01	Un procedimiento para la preparacion de un derivado de n-metil-1-alquiltio-2-nitroetonamina
ES520078A0 (es)	1984-04-01	Un procedimiento para la preparacion de un derivado de b -lactama.
ES515365A0 (es)	1983-11-01	Un procedimiento para la preparacion de un derivado de furanocremona.
ES539247A0 (es)	1985-12-01	Un procedimiento para la preparacion de benzotienil-, benzofuranil o naftil-derivados
ES505718A0 (es)	1983-02-01	Un procedimiento para la preparacion de derivados de cefa- losporina
ES517690A0 (es)	1983-12-16	Un procedimiento para la preparacion de un derivado de 3-carboxillavam.
ES504478A0 (es)	1982-06-01	Un procedimiento para la preparacion de 2-benzotiazol-sul- fenamidas
ES524859A0 (es)	1985-01-16	Un procedimiento para la preparacion de feniltetrahidroftalimidas
ES499753A0 (es)	1982-02-16	Un procedimiento para la preparacion de derivados de cefa- losporina
ES538691A0 (es)	1986-01-01	Procedimiento para la obtencion de un derivado de la vincamina
ES514426A0 (es)	1983-05-01	Un procedimiento para la preparacion de un derivado de fenetilamina.
ES500475A0 (es)	1982-02-01	Procedimiento para la preparacion de 2-halogenoacetamidas

Legal Events

Date	Code	Title	Description
2000-01-01	FD1A	Patent lapsed	Effective date: 19991108