ES490799A0 - Un procedimiento para la preparacion de derivados de imida- zolidina - Google Patents
Un procedimiento para la preparacion de derivados de imida- zolidinaInfo
- Publication number
- ES490799A0 ES490799A0 ES490799A ES490799A ES490799A0 ES 490799 A0 ES490799 A0 ES 490799A0 ES 490799 A ES490799 A ES 490799A ES 490799 A ES490799 A ES 490799A ES 490799 A0 ES490799 A0 ES 490799A0
- Authority
- ES
- Spain
- Prior art keywords
- general formula
- signifies
- compound
- see diagramm
- imida
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/30—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by halogen atoms, or by nitro or nitroso groups
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
- C07D233/80—Two oxygen atoms, e.g. hydantoin with hetero atoms or acyl radicals directly attached to ring nitrogen atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Epoxy Resins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH383779 | 1979-04-24 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES490799A0 true ES490799A0 (es) | 1981-04-16 |
| ES8104243A1 ES8104243A1 (es) | 1981-04-16 |
Family
ID=4264536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES490799A Expired ES8104243A1 (es) | 1979-04-24 | 1980-04-23 | Un procedimiento para la preparacion de derivados de imida- zolidina |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0017976B1 (es) |
| JP (1) | JPS55143974A (es) |
| KR (1) | KR850000719B1 (es) |
| AT (1) | ATE3860T1 (es) |
| CA (1) | CA1135706A (es) |
| DE (1) | DE3063837D1 (es) |
| DK (1) | DK174480A (es) |
| ES (1) | ES8104243A1 (es) |
| FI (1) | FI801184A7 (es) |
| GR (1) | GR67605B (es) |
| HU (1) | HU184271B (es) |
| NO (1) | NO801182L (es) |
| PT (1) | PT71135B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5411981A (en) * | 1991-01-09 | 1995-05-02 | Roussel Uclaf | Phenylimidazolidines having antiandrogenic activity |
| USRE35956E (en) * | 1991-01-09 | 1998-11-10 | Roussel Uclaf | Phenylimidazolidines having antiandrogenic activity |
| FR2715402B1 (fr) * | 1994-01-05 | 1996-10-04 | Roussel Uclaf | Nouvelles phénylimidazolines éventuellement substituées, leur procédé et des intermédiaires de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant. |
| FR2724169B1 (fr) * | 1994-09-06 | 1997-01-03 | Roussel Uclaf | Nouvelles phenylimidazolidines eventuellement substituees, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
| TW521073B (en) * | 1994-01-05 | 2003-02-21 | Hoechst Marion Roussel Inc | New optionally substituted phenylimidazolidines, their preparation process, their use as anti-androgenic agent and the pharmaceutical compositions containing them |
| AU2004305075A1 (en) | 2003-12-19 | 2005-07-07 | The Regents Of The University Of California | Methods and materials for assessing prostate cancer therapies |
| NZ550102A (en) | 2004-02-24 | 2010-10-29 | Univ California | Methods and materials for assessing prostate cancer therapies and compounds (thiohydantoine derivatives) |
| AU2007245022A1 (en) | 2006-03-29 | 2007-11-08 | The Regents Of The University Of California | Diarylthiohydantoin compounds |
| US7709517B2 (en) | 2005-05-13 | 2010-05-04 | The Regents Of The University Of California | Diarylhydantoin compounds |
| DK3100727T3 (en) | 2006-03-27 | 2018-11-12 | Univ California | Androgen receptor modulator for the treatment of prostate cancer and androgen receptor-associated diseases |
| WO2009055053A2 (en) | 2007-10-26 | 2009-04-30 | The Regents Of The University Of California | Diarylhydantoin compounds as androgen receptor modulators |
| EP3124481B1 (en) | 2010-02-16 | 2018-03-28 | Aragon Pharmaceuticals, Inc. | Androgen receptor modulators and uses thereof |
| SG10201912719TA (en) | 2012-09-26 | 2020-02-27 | Aragon Pharmaceuticals Inc | Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer |
| JOP20200097A1 (ar) | 2013-01-15 | 2017-06-16 | Aragon Pharmaceuticals Inc | معدل مستقبل أندروجين واستخداماته |
| TWI726969B (zh) | 2016-01-11 | 2021-05-11 | 比利時商健生藥品公司 | 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物 |
| JP7201694B2 (ja) | 2017-10-16 | 2023-01-10 | アラゴン ファーマシューティカルズ,インコーポレイテッド | 非転移性去勢抵抗性前立腺癌の治療のための抗アンドロゲン剤 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB997037A (en) * | 1962-03-19 | 1965-06-30 | Ici Ltd | New hydrantoin derivatives |
| US3340070A (en) * | 1963-08-23 | 1967-09-05 | Shell Oil Co | Artificial sweetening agent |
| FR2329276A1 (fr) * | 1975-10-29 | 1977-05-27 | Roussel Uclaf | Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant |
| MC1220A1 (fr) * | 1977-10-28 | 1979-07-20 | Hoffmann La Roche | Nouveaux derives d'imidazolidine |
| CA1138334A (en) * | 1977-10-28 | 1982-12-28 | Karl Bernauer | Pharmaceutical preparations containing certain urea derivatives |
-
1980
- 1980-04-14 FI FI801184A patent/FI801184A7/fi not_active Application Discontinuation
- 1980-04-16 DE DE8080102042T patent/DE3063837D1/de not_active Expired
- 1980-04-16 EP EP80102042A patent/EP0017976B1/de not_active Expired
- 1980-04-16 AT AT80102042T patent/ATE3860T1/de not_active IP Right Cessation
- 1980-04-18 CA CA000350162A patent/CA1135706A/en not_active Expired
- 1980-04-21 JP JP5180480A patent/JPS55143974A/ja active Pending
- 1980-04-22 GR GR61749A patent/GR67605B/el unknown
- 1980-04-23 HU HU80995A patent/HU184271B/hu unknown
- 1980-04-23 NO NO801182A patent/NO801182L/no unknown
- 1980-04-23 DK DK174480A patent/DK174480A/da not_active Application Discontinuation
- 1980-04-23 ES ES490799A patent/ES8104243A1/es not_active Expired
- 1980-04-23 PT PT71135A patent/PT71135B/pt unknown
- 1980-04-24 KR KR1019800001691A patent/KR850000719B1/ko not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ATE3860T1 (de) | 1983-07-15 |
| EP0017976A2 (de) | 1980-10-29 |
| FI801184A7 (fi) | 1981-01-01 |
| KR830002722A (ko) | 1983-05-30 |
| JPS55143974A (en) | 1980-11-10 |
| KR850000719B1 (ko) | 1985-05-23 |
| GR67605B (es) | 1981-08-31 |
| EP0017976A3 (en) | 1981-04-01 |
| NO801182L (no) | 1980-10-27 |
| PT71135A (en) | 1980-05-01 |
| DE3063837D1 (en) | 1983-07-28 |
| DK174480A (da) | 1980-10-25 |
| HU184271B (en) | 1984-07-30 |
| CA1135706A (en) | 1982-11-16 |
| PT71135B (en) | 1981-08-07 |
| EP0017976B1 (de) | 1983-06-22 |
| ES8104243A1 (es) | 1981-04-16 |
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