ES476024A1 - Un procedimiento para preparar derivados de cefalosporina - Google Patents
Un procedimiento para preparar derivados de cefalosporinaInfo
- Publication number
- ES476024A1 ES476024A1 ES476024A ES476024A ES476024A1 ES 476024 A1 ES476024 A1 ES 476024A1 ES 476024 A ES476024 A ES 476024A ES 476024 A ES476024 A ES 476024A ES 476024 A1 ES476024 A1 ES 476024A1
- Authority
- ES
- Spain
- Prior art keywords
- cephem
- methyl
- carboxylic acids
- methoxymethyl esters
- substituted imidazolidinyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- GLYWBKWOTGKGEE-HNHGDDPOSA-N (6r)-4-imidazolidin-1-yl-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical class S([C@H]1N(C(C1)=O)C(=C1C)C(O)=O)C1N1CCNC1 GLYWBKWOTGKGEE-HNHGDDPOSA-N 0.000 title 1
- 125000004184 methoxymethyl group Chemical group [H]C([H])([H])OC([H])([H])* 0.000 title 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/58—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with a nitrogen atom, which is a member of a hetero ring, attached in position 7
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1. Un procedimiento para preparar derivados de cefalosporina de fórmula: **Fórmula-01** cuyo procedimiento comprende hacer reaccionar en cualquier orden un compuesto de fórmula: **Fórmula-02** con: a) acetona, y b) bromometil-metil-éter.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/861,334 US4125716A (en) | 1977-12-16 | 1977-12-16 | Methoxymethyl esters of substituted imidazolidinyl-3-methyl-3-cephem-4-carboxylic acids |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES476024A1 true ES476024A1 (es) | 1980-05-16 |
Family
ID=25335521
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES476024A Expired ES476024A1 (es) | 1977-12-16 | 1978-12-14 | Un procedimiento para preparar derivados de cefalosporina |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4125716A (es) |
| JP (1) | JPS5490193A (es) |
| BE (1) | BE872744A (es) |
| CA (1) | CA1100946A (es) |
| CH (1) | CH637968A5 (es) |
| DE (1) | DE2854041A1 (es) |
| ES (1) | ES476024A1 (es) |
| FR (1) | FR2411840A1 (es) |
| GB (1) | GB2010269B (es) |
| GR (1) | GR70245B (es) |
| IT (1) | IT1109343B (es) |
| NL (1) | NL7812236A (es) |
| YU (1) | YU42169B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS54112892A (en) * | 1978-02-23 | 1979-09-04 | Shionogi & Co Ltd | Substituted imidazolidinyl-3-chloro-3-cephem-4-carboxylic acid |
| US4219495A (en) * | 1979-02-28 | 1980-08-26 | Bristol-Myers Company | Methoxymethyl p-toluenesulfonate |
| US4217275A (en) * | 1979-02-28 | 1980-08-12 | Bristol-Myers Company | β-Lactam antibiotic esterification process using methoxymethyl methane sulfonate |
| US20050181353A1 (en) * | 2004-02-17 | 2005-08-18 | Rao Galla C. | Stabilization of cells and biological specimens for analysis |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| USRE29164E (en) | 1967-09-05 | 1977-03-29 | Bristol-Myers Company | 7-Amino-cephalosporanic and decephalosporanic acid derivatives |
| US3489751A (en) * | 1967-09-05 | 1970-01-13 | Bristol Myers Co | 7-amino-cephalosporanic and decephalosporanic acid derivatives |
| US3714146A (en) * | 1970-10-05 | 1973-01-30 | Bristol Myers Co | Novel syntheses of cephalexin and intermediates therefor |
| JPS5513719B2 (es) * | 1972-12-06 | 1980-04-10 | ||
| US3996236A (en) * | 1973-03-24 | 1976-12-07 | Bristol-Myers Company | Methoxymethyl D-6-(2,2-dimethyl-5-oxo-4-phenyl-1-imidazolidinyl)penicillanate |
-
1977
- 1977-12-16 US US05/861,334 patent/US4125716A/en not_active Expired - Lifetime
-
1978
- 1978-12-04 CA CA317,296A patent/CA1100946A/en not_active Expired
- 1978-12-12 FR FR7834873A patent/FR2411840A1/fr active Granted
- 1978-12-13 GB GB7848371A patent/GB2010269B/en not_active Expired
- 1978-12-13 JP JP15322978A patent/JPS5490193A/ja active Pending
- 1978-12-13 YU YU2924/78A patent/YU42169B/xx unknown
- 1978-12-13 BE BE192305A patent/BE872744A/xx not_active IP Right Cessation
- 1978-12-14 ES ES476024A patent/ES476024A1/es not_active Expired
- 1978-12-14 GR GR57871A patent/GR70245B/el unknown
- 1978-12-14 DE DE19782854041 patent/DE2854041A1/de not_active Withdrawn
- 1978-12-15 IT IT52314/78A patent/IT1109343B/it active
- 1978-12-15 NL NL7812236A patent/NL7812236A/xx not_active Application Discontinuation
- 1978-12-15 CH CH1281378A patent/CH637968A5/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| NL7812236A (nl) | 1979-06-19 |
| US4125716A (en) | 1978-11-14 |
| GB2010269A (en) | 1979-06-27 |
| DE2854041A1 (de) | 1979-06-28 |
| YU292478A (en) | 1983-01-21 |
| CH637968A5 (de) | 1983-08-31 |
| IT7852314A0 (it) | 1978-12-15 |
| GR70245B (es) | 1982-09-01 |
| IT1109343B (it) | 1985-12-16 |
| FR2411840A1 (fr) | 1979-07-13 |
| FR2411840B1 (es) | 1983-04-01 |
| BE872744A (fr) | 1979-06-13 |
| CA1100946A (en) | 1981-05-12 |
| JPS5490193A (en) | 1979-07-17 |
| YU42169B (en) | 1988-06-30 |
| GB2010269B (en) | 1982-06-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19980202 |