ES369479A1 - (1)benzothieno(2 3-d)pyrimidine derivatives - Google Patents
(1)benzothieno(2 3-d)pyrimidine derivativesInfo
- Publication number
- ES369479A1 ES369479A1 ES369479A ES369479A ES369479A1 ES 369479 A1 ES369479 A1 ES 369479A1 ES 369479 A ES369479 A ES 369479A ES 369479 A ES369479 A ES 369479A ES 369479 A1 ES369479 A1 ES 369479A1
- Authority
- ES
- Spain
- Prior art keywords
- amino
- dissociated
- lower alkyl
- amino group
- benzothiene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229940083082 pyrimidine derivative acting on arteriolar smooth muscle Drugs 0.000 title 1
- 150000003230 pyrimidines Chemical class 0.000 title 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 3
- 125000002837 carbocyclic group Chemical group 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- SYSQUGFVNFXIIT-UHFFFAOYSA-N n-[4-(1,3-benzoxazol-2-yl)phenyl]-4-nitrobenzenesulfonamide Chemical class C1=CC([N+](=O)[O-])=CC=C1S(=O)(=O)NC1=CC=C(C=2OC3=CC=CC=C3N=2)C=C1 SYSQUGFVNFXIIT-UHFFFAOYSA-N 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/62—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by hydrogenation of carbon-to-carbon double or triple bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
- C07C45/676—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton by elimination of carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Procedure for obtaining [1] benzothiene/2,3-3/-pyrimidines and their 5,6,7,8-tetrahydro derivatives, which carry at least one aromatic carbocyclic moiety on the carbocyclic ring, and that in position 4 show an amino-lower alkyl-amino group, characterized in that in a 4-Y- [1] benzothiene [2,3-d] pyrimidine, which has at least one residue in the carbocyclic ring, aromatic carbocyclic, and where Y means a moiety transformable into an amino-lower alkyl-amino group, 6 into a 5,6,7,8-tetrahydro derivative thereof, AND is transformed into an amino-lower alkyl-amino group and, if desired, in the compounds obtained, within the scope of the definition of the final products, substituents are introduced, modified or dissociated, and/or, the mixtures of isomers obtained are dissociated into the pure cis- and trans-isomers and/or the racemates obtained are dissociated in the optical antipodes and/or the free bases obtained they are transformed into their salts, or the obtained salts You start on free bases. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1052268A CH508649A (en) | 1968-07-15 | 1968-07-15 | New pyrimidine derivates and their manufacture |
| CH865169A CH530412A (en) | 1968-07-15 | 1969-06-05 | Process for the preparation of (1) benzothieno- (2,3-d) pyrimidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES369479A1 true ES369479A1 (en) | 1971-06-16 |
Family
ID=25703582
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES369479A Expired ES369479A1 (en) | 1968-07-15 | 1969-07-14 | (1)benzothieno(2 3-d)pyrimidine derivatives |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US3634427A (en) |
| AR (1) | AR194562A1 (en) |
| AT (4) | AT292689B (en) |
| BE (1) | BE736045A (en) |
| BR (1) | BR6910708D0 (en) |
| CA (1) | CA933523A (en) |
| CH (1) | CH530412A (en) |
| DE (1) | DE1934172A1 (en) |
| ES (1) | ES369479A1 (en) |
| FR (1) | FR2012951A1 (en) |
| GB (1) | GB1277743A (en) |
| IE (1) | IE33226B1 (en) |
| NL (1) | NL6910807A (en) |
| OA (1) | OA03378A (en) |
| SU (1) | SU416946A3 (en) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3966733A (en) * | 1973-07-26 | 1976-06-29 | E. R. Squibb & Sons, Inc. | Intermediates for certain benzothiadiazepine and benzothiadiazocine compounds |
| US3875162A (en) * | 1973-07-26 | 1975-04-01 | Squibb & Sons Inc | Certain 6H-pyrimido{8 1,2-c{9 {8 1,3,5{9 benzothiadiaza compounds |
| US4054656A (en) * | 1975-09-10 | 1977-10-18 | Mead Johnson & Company | Thieno[2,3-d]pyrimidine antiallergic agents |
| GB1570494A (en) | 1975-11-28 | 1980-07-02 | Ici Ltd | Thienopyrimidine derivatives and their use as pesticides |
| NO150804C (en) * | 1982-04-13 | 1984-12-27 | Thune Eureka As | DEVICE FOR HEAT TREATMENT OF A CONTINUOUS WIRE OR FILLET |
| US5679683A (en) * | 1994-01-25 | 1997-10-21 | Warner-Lambert Company | Tricyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family |
| IL112248A0 (en) | 1994-01-25 | 1995-03-30 | Warner Lambert Co | Tricyclic heteroaromatic compounds and pharmaceutical compositions containing them |
| IL112249A (en) | 1994-01-25 | 2001-11-25 | Warner Lambert Co | Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds |
| CN105061460B (en) * | 2015-08-18 | 2017-06-30 | 沈阳药科大学 | Tetrahydro benzo [4,5] thieno [2,3 d] pyrimidines and its application containing sulfide based structural |
| CN105061461B (en) * | 2015-08-18 | 2017-06-30 | 沈阳药科大学 | Tetrahydro benzo [4,5] thieno [2,3 d] pyrimidines and its application containing benzylamine structure |
| KR20250065420A (en) * | 2015-12-25 | 2025-05-12 | 가부시키가이샤 한도오따이 에네루기 켄큐쇼 | Compound, light-emitting element, display device, electronic device, and lighting device |
| JP2019006763A (en) | 2017-06-22 | 2019-01-17 | 株式会社半導体エネルギー研究所 | Organic compound, light-emitting element, light-emitting device, electronic apparatus, and lighting device |
-
1969
- 1969-06-05 CH CH865169A patent/CH530412A/en unknown
- 1969-07-02 FR FR6922264A patent/FR2012951A1/fr not_active Withdrawn
- 1969-07-05 DE DE19691934172 patent/DE1934172A1/en active Pending
- 1969-07-07 CA CA056328A patent/CA933523A/en not_active Expired
- 1969-07-08 US US840035A patent/US3634427A/en not_active Expired - Lifetime
- 1969-07-08 OA OA53665A patent/OA03378A/en unknown
- 1969-07-10 GB GB34766/69A patent/GB1277743A/en not_active Expired
- 1969-07-14 AT AT517670A patent/AT292689B/en active
- 1969-07-14 AT AT517570A patent/AT292688B/en active
- 1969-07-14 AT AT674769A patent/AT289784B/en active
- 1969-07-14 NL NL6910807A patent/NL6910807A/xx unknown
- 1969-07-14 ES ES369479A patent/ES369479A1/en not_active Expired
- 1969-07-14 SU SU1485634A patent/SU416946A3/en active
- 1969-07-14 AT AT517770A patent/AT292690B/en not_active IP Right Cessation
- 1969-07-14 BE BE736045D patent/BE736045A/xx unknown
- 1969-07-15 BR BR210708/69A patent/BR6910708D0/en unknown
- 1969-07-15 IE IE968/69A patent/IE33226B1/en unknown
-
1970
- 1970-06-01 AR AR229038A patent/AR194562A1/en active
Also Published As
| Publication number | Publication date |
|---|---|
| BR6910708D0 (en) | 1973-02-15 |
| BE736045A (en) | 1970-01-14 |
| FR2012951A1 (en) | 1970-03-27 |
| GB1277743A (en) | 1972-06-14 |
| AT289784B (en) | 1971-05-10 |
| IE33226B1 (en) | 1974-04-17 |
| SU416946A3 (en) | 1974-02-25 |
| CH530412A (en) | 1972-11-15 |
| AT292690B (en) | 1971-09-10 |
| DE1934172A1 (en) | 1970-01-22 |
| US3634427A (en) | 1972-01-11 |
| AR194562A1 (en) | 1973-07-31 |
| AT292688B (en) | 1971-09-10 |
| OA03378A (en) | 1970-12-15 |
| IE33226L (en) | 1970-01-15 |
| CA933523A (en) | 1973-09-11 |
| NL6910807A (en) | 1970-01-19 |
| AT292689B (en) | 1971-09-10 |
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