ES2187038T3 - Glicosidos modificados, composiciones que los comprenden y procedimientos para su utilizacion. - Google Patents
Glicosidos modificados, composiciones que los comprenden y procedimientos para su utilizacion.Info
- Publication number
- ES2187038T3 ES2187038T3 ES98932361T ES98932361T ES2187038T3 ES 2187038 T3 ES2187038 T3 ES 2187038T3 ES 98932361 T ES98932361 T ES 98932361T ES 98932361 T ES98932361 T ES 98932361T ES 2187038 T3 ES2187038 T3 ES 2187038T3
- Authority
- ES
- Spain
- Prior art keywords
- modified
- variety
- glycosids
- procedures
- understand
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000000034 method Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 239000007787 solid Substances 0.000 abstract 3
- 239000000126 substance Substances 0.000 abstract 3
- 239000011521 glass Substances 0.000 abstract 2
- 229930182470 glycoside Natural products 0.000 abstract 2
- 150000002338 glycosides Chemical class 0.000 abstract 2
- 239000011159 matrix material Substances 0.000 abstract 2
- 238000000576 coating method Methods 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000007943 implant Substances 0.000 abstract 1
- 238000011065 in-situ storage Methods 0.000 abstract 1
- 238000001990 intravenous administration Methods 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 239000004005 microsphere Substances 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
- 230000002685 pulmonary effect Effects 0.000 abstract 1
- 239000003826 tablet Substances 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Biotechnology (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Crystallography & Structural Chemistry (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Medicinal Chemistry (AREA)
- Medicinal Preparation (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
Se proporcionan glucósidos modificados que pueden utilizarse para formar una variedad de materiales, incluyendo sistemas de administración sólida, y dispositivos o recubrimientos coloreados ópticamente transparentes. Los sistemas de administración sólida pueden utilizarse para la administración y la liberación de una variedad de sustancias que pueden estar en forma de comprimidos para administración oral o en forma de polvos, microesferas o implantes para por vía intravenosa, intradérmica, transdérmica, pulmonar u otra vía de administración. Los glucósidos modificados pueden procesarse para formar una matriz de vidrio vítreo con una sustancia, tal como un agente terapéutico, o un tinte ópticamente activo incorporado a la misma. En una realización, la matriz de vidrio vítreo se proporciona en una forma de dosificación sólida que es capaz de liberar una sustancia terapéutica in situ a diversas velocidades controladas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5172797P | 1997-07-03 | 1997-07-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2187038T3 true ES2187038T3 (es) | 2003-05-16 |
Family
ID=21973024
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES98932361T Expired - Lifetime ES2187038T3 (es) | 1997-07-03 | 1998-07-03 | Glicosidos modificados, composiciones que los comprenden y procedimientos para su utilizacion. |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0994887B1 (es) |
| JP (1) | JP2002510316A (es) |
| AT (1) | ATE228528T1 (es) |
| AU (1) | AU8229998A (es) |
| DE (1) | DE69809746T2 (es) |
| DK (1) | DK0994887T3 (es) |
| ES (1) | ES2187038T3 (es) |
| PT (1) | PT994887E (es) |
| WO (1) | WO1999001463A2 (es) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6586006B2 (en) * | 1994-08-04 | 2003-07-01 | Elan Drug Delivery Limited | Solid delivery systems for controlled release of molecules incorporated therein and methods of making same |
| US6352722B1 (en) | 1997-12-23 | 2002-03-05 | Quadrant Holdings Cambridge Limited | Derivatized carbohydrates, compositions comprised thereof and methods of use thereof |
| GB9916316D0 (en) | 1999-07-12 | 1999-09-15 | Quadrant Holdings Cambridge | Dry powder compositions |
| CN1431919A (zh) | 2000-04-03 | 2003-07-23 | 巴特勒记忆研究所 | 装置和制剂 |
| GB0017999D0 (en) | 2000-07-21 | 2000-09-13 | Smithkline Beecham Biolog | Novel device |
| JP2004526674A (ja) | 2000-12-01 | 2004-09-02 | バテル・メモリアル・インスティテュート | 液体処方物中における生体分子の安定化のための方法 |
| EP1752189A3 (en) * | 2001-04-20 | 2007-02-21 | Alza Corporation | Microprojection array having a beneficial agent containing coating |
| GB0208608D0 (en) * | 2002-04-13 | 2002-05-22 | Glaxo Group Ltd | Composition |
| GB0208609D0 (en) * | 2002-04-13 | 2002-05-22 | Glaxo Group Ltd | Compositions |
| EP1428526A1 (en) * | 2002-12-13 | 2004-06-16 | Rijksuniversiteit Groningen | Formulation for fast dissolution of lipophilic compounds |
| JP4722386B2 (ja) * | 2003-08-22 | 2011-07-13 | 広島県 | 糖脂質及びその製造方法 |
| WO2006014930A2 (en) * | 2004-07-26 | 2006-02-09 | Cotherix, Inc. | Treatment of pulmonary hypertension by inhaled iloprost with a microparticle formulation |
| WO2007013160A1 (ja) | 2005-07-28 | 2007-02-01 | Saga University | ラジカル滅菌装置 |
| WO2023077447A1 (zh) * | 2021-11-05 | 2023-05-11 | 中国科学院过程工程研究所 | 环肽玻璃及含有环肽的药物组合物玻璃 |
| CN114014908B (zh) * | 2021-11-05 | 2023-08-22 | 中国科学院过程工程研究所 | 环肽玻璃及含有环肽的药物组合物玻璃 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CZ297431B6 (cs) * | 1994-08-04 | 2006-12-13 | Quadrant Holdings Cambridge Limited | Prostredek obsahující dodávací systém pevné dávkypro prímou aplikaci v pevné forme a zpusob jeho výroby |
-
1998
- 1998-07-03 JP JP50667799A patent/JP2002510316A/ja not_active Abandoned
- 1998-07-03 ES ES98932361T patent/ES2187038T3/es not_active Expired - Lifetime
- 1998-07-03 DK DK98932361T patent/DK0994887T3/da active
- 1998-07-03 PT PT98932361T patent/PT994887E/pt unknown
- 1998-07-03 AU AU82299/98A patent/AU8229998A/en not_active Abandoned
- 1998-07-03 AT AT98932361T patent/ATE228528T1/de not_active IP Right Cessation
- 1998-07-03 EP EP98932361A patent/EP0994887B1/en not_active Expired - Lifetime
- 1998-07-03 DE DE69809746T patent/DE69809746T2/de not_active Expired - Fee Related
- 1998-07-03 WO PCT/GB1998/001962 patent/WO1999001463A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| DE69809746T2 (de) | 2004-09-30 |
| EP0994887A2 (en) | 2000-04-26 |
| DE69809746D1 (de) | 2003-01-09 |
| EP0994887B1 (en) | 2002-11-27 |
| JP2002510316A (ja) | 2002-04-02 |
| DK0994887T3 (da) | 2003-03-17 |
| ATE228528T1 (de) | 2002-12-15 |
| WO1999001463A3 (en) | 1999-03-25 |
| PT994887E (pt) | 2003-04-30 |
| WO1999001463A2 (en) | 1999-01-14 |
| AU8229998A (en) | 1999-01-25 |
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