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EE9500055A - 1,4-dihüdropüridiin-3,5-dikarboksüülhappeestrite kasutamine ravimitena, ravimid ja nende valmistamismeetod - Google Patents

1,4-dihüdropüridiin-3,5-dikarboksüülhappeestrite kasutamine ravimitena, ravimid ja nende valmistamismeetod

Info

Publication number
EE9500055A
EE9500055A EE9500055A EE9500055A EE9500055A EE 9500055 A EE9500055 A EE 9500055A EE 9500055 A EE9500055 A EE 9500055A EE 9500055 A EE9500055 A EE 9500055A EE 9500055 A EE9500055 A EE 9500055A
Authority
EE
Estonia
Prior art keywords
medicaments
dihydropyridine
preparation
dicarboxylic acid
acid esters
Prior art date
Application number
EE9500055A
Other languages
English (en)
Estonian (et)
Inventor
Urbahns Klaus
Behner Otto
Goldmann Siegfried
Heine Hans-Georg
Junge Bodo
Schohe-Loop Rudolf
Wehinger Egbert
Wollweber Hartmund
Sommermeyer Henning
Glaser Thomas
Wittka Reilinde
De Vry Jean-Marie-Viktor
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of EE9500055A publication Critical patent/EE9500055A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
EE9500055A 1994-08-25 1995-08-24 1,4-dihüdropüridiin-3,5-dikarboksüülhappeestrite kasutamine ravimitena, ravimid ja nende valmistamismeetod EE9500055A (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4430094A DE4430094A1 (de) 1994-08-25 1994-08-25 Verwendung von 3,5-Dicarbonsäureester-1,4-Dihydropyridinen als Arzneimittel

Publications (1)

Publication Number Publication Date
EE9500055A true EE9500055A (et) 1996-04-15

Family

ID=6526498

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9500055A EE9500055A (et) 1994-08-25 1995-08-24 1,4-dihüdropüridiin-3,5-dikarboksüülhappeestrite kasutamine ravimitena, ravimid ja nende valmistamismeetod

Country Status (14)

Country Link
US (2) US5665741A (xx)
EP (1) EP0705819A1 (xx)
JP (1) JPH0859468A (xx)
KR (1) KR960007563A (xx)
CN (1) CN1128757A (xx)
AU (1) AU3011295A (xx)
CA (1) CA2156673A1 (xx)
DE (1) DE4430094A1 (xx)
EE (1) EE9500055A (xx)
FI (1) FI953957L (xx)
HU (1) HUT74617A (xx)
IL (1) IL115030A0 (xx)
NO (1) NO953322L (xx)
PL (1) PL310146A1 (xx)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000078719A1 (en) * 1999-06-23 2000-12-28 Ajinomoto Co., Inc. Dihydropyridine derivative
ATE511858T1 (de) * 2002-02-05 2011-06-15 Astellas Pharma Inc 2,4,6-triamino-1,3,5-triazin-derivat
US20050075359A1 (en) * 2003-03-14 2005-04-07 Rikako Kono Large conductance calcium-activated K channel opener
AU2012342226B2 (en) * 2011-11-24 2017-09-28 Richter Gedeon Nyrt. 1,4- dihydropyridine derivatives with Hsp modulating activity
CN104710441B (zh) * 2014-12-18 2017-01-18 苏州科技学院 吡啶五甲酸二钾化合物及其制备方法
US20230416203A1 (en) * 2020-11-30 2023-12-28 Nanyang Technological University Potent and selective inhibitors of the calcium-activated potassium channel, kca3.1, for use as platform therapeutics

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1813436C3 (de) * 1968-12-07 1979-01-11 Bayer Ag, 5090 Leverkusen N-Substituierte 2,6-Dimethyl-l,4dihydropyridine
US3883543A (en) * 1969-05-10 1975-05-13 Bayer Ag N-alkyl-1,4-dihydropyridines
DE1923990C3 (de) * 1969-05-10 1978-11-23 Bayer Ag Verfahren zur Herstellung von N-substituierten M-Dihydropyridin-S.S-dicarbonsäureestern
JPS4899181A (xx) * 1972-04-04 1973-12-15
DE2815578C2 (de) 1978-04-11 1986-01-16 Bayer Ag, 5090 Leverkusen Neue pharmazeutische Verwendung von Nimodipin
EP0287828A1 (de) * 1987-03-27 1988-10-26 Byk Gulden Lomberg Chemische Fabrik GmbH Neue Zwischenprodukte und Verfahren
DE4011695A1 (de) * 1990-04-11 1991-10-17 Bayer Ag Verwendung von n-alkylierten 1,4-dihydropyridindicarbonsaeureestern als arzneimittel, neue verbindungen und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
PL310146A1 (en) 1996-03-04
FI953957A7 (fi) 1996-02-26
NO953322L (no) 1996-02-26
US5665741A (en) 1997-09-09
FI953957L (fi) 1996-02-26
CN1128757A (zh) 1996-08-14
CA2156673A1 (en) 1996-02-26
JPH0859468A (ja) 1996-03-05
NO953322D0 (no) 1995-08-24
KR960007563A (ko) 1996-03-22
AU3011295A (en) 1996-03-07
IL115030A0 (en) 1995-12-08
US5955482A (en) 1999-09-21
HU9502509D0 (en) 1995-10-30
DE4430094A1 (de) 1996-02-29
FI953957A0 (fi) 1995-08-23
EP0705819A1 (de) 1996-04-10
HUT74617A (en) 1997-01-28

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