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EE200300083A - Bitsüklilised pürrooli amiidid kui glükogeeni fosforülaasi inhibiitorid - Google Patents

Bitsüklilised pürrooli amiidid kui glükogeeni fosforülaasi inhibiitorid

Info

Publication number
EE200300083A
EE200300083A EEP200300083A EEP200300083A EE200300083A EE 200300083 A EE200300083 A EE 200300083A EE P200300083 A EEP200300083 A EE P200300083A EE P200300083 A EEP200300083 A EE P200300083A EE 200300083 A EE200300083 A EE 200300083A
Authority
EE
Estonia
Prior art keywords
glycogen phosphorylase
phosphorylase inhibitors
pyrrole amides
bicyclic pyrrole
amide derivatives
Prior art date
Application number
EEP200300083A
Other languages
English (en)
Inventor
B. Bartlett Julie
Freeman Sue
Kenny Peter
Morley Andrew
Whittamore Paul
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of EE200300083A publication Critical patent/EE200300083A/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Enzymes And Modification Thereof (AREA)
EEP200300083A 2000-09-06 2001-08-31 Bitsüklilised pürrooli amiidid kui glükogeeni fosforülaasi inhibiitorid EE200300083A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0021831.3A GB0021831D0 (en) 2000-09-06 2000-09-06 Chemical compounds
PCT/SE2001/001880 WO2002020530A1 (en) 2000-09-06 2001-08-31 Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors

Publications (1)

Publication Number Publication Date
EE200300083A true EE200300083A (et) 2004-12-15

Family

ID=9898927

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300083A EE200300083A (et) 2000-09-06 2001-08-31 Bitsüklilised pürrooli amiidid kui glükogeeni fosforülaasi inhibiitorid

Country Status (30)

Country Link
US (1) US20030232875A1 (et)
EP (1) EP1317459B1 (et)
JP (1) JP2004508376A (et)
KR (1) KR100802369B1 (et)
CN (2) CN1896078A (et)
AT (1) ATE263772T1 (et)
AU (2) AU8283301A (et)
BG (1) BG107624A (et)
BR (1) BR0113606A (et)
CA (1) CA2417594A1 (et)
CZ (1) CZ2003616A3 (et)
DE (1) DE60102710T2 (et)
DK (1) DK1317459T3 (et)
EE (1) EE200300083A (et)
ES (1) ES2217183T3 (et)
GB (1) GB0021831D0 (et)
HU (1) HUP0400784A3 (et)
IL (1) IL154291A0 (et)
IS (1) IS2110B (et)
MX (1) MXPA03001512A (et)
NO (1) NO20031024D0 (et)
NZ (1) NZ524011A (et)
PL (1) PL361024A1 (et)
PT (1) PT1317459E (et)
RU (1) RU2003104013A (et)
SK (1) SK2592003A3 (et)
TR (1) TR200401659T4 (et)
UA (1) UA73781C2 (et)
WO (1) WO2002020530A1 (et)
ZA (1) ZA200301013B (et)

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DE10225635C1 (de) * 2002-06-07 2003-12-24 Aventis Pharma Gmbh N-Benzoylureido-Zimtsäurederivate, Verfahren zu deren Herstellung und deren Verwendung
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US7186735B2 (en) 2002-08-07 2007-03-06 Sanofi-Aventis Deutschland Gmbh Acylated arylcycloalkylamines and their use as pharmaceuticals
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Also Published As

Publication number Publication date
ES2217183T3 (es) 2004-11-01
DK1317459T3 (da) 2004-07-12
NO20031024L (no) 2003-03-05
NO20031024D0 (no) 2003-03-05
AU2001282833B2 (en) 2006-07-06
UA73781C2 (en) 2005-09-15
SK2592003A3 (en) 2003-08-05
DE60102710D1 (de) 2004-05-13
JP2004508376A (ja) 2004-03-18
BR0113606A (pt) 2003-06-24
HUP0400784A3 (en) 2007-09-28
KR100802369B1 (ko) 2008-02-14
IS6727A (is) 2003-02-24
CA2417594A1 (en) 2002-03-14
RU2003104013A (ru) 2004-08-20
NZ524011A (en) 2004-08-27
KR20030025305A (ko) 2003-03-28
ATE263772T1 (de) 2004-04-15
EP1317459B1 (en) 2004-04-07
GB0021831D0 (en) 2000-10-18
IL154291A0 (en) 2003-09-17
ZA200301013B (en) 2004-05-05
BG107624A (bg) 2004-01-30
US20030232875A1 (en) 2003-12-18
WO2002020530A1 (en) 2002-03-14
CZ2003616A3 (cs) 2003-05-14
CN1473163A (zh) 2004-02-04
EP1317459A1 (en) 2003-06-11
IS2110B (is) 2006-05-15
CN1264846C (zh) 2006-07-19
MXPA03001512A (es) 2003-06-09
PT1317459E (pt) 2004-08-31
HUP0400784A2 (hu) 2004-07-28
AU8283301A (en) 2002-03-22
HK1055299A1 (en) 2004-01-02
PL361024A1 (en) 2004-09-20
DE60102710T2 (de) 2005-04-14
CN1896078A (zh) 2007-01-17
TR200401659T4 (tr) 2004-09-21

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