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EE200100333A - Meetod 2-halo-3-nitro-4-aminopüridiini valmistamiseks ja selleks vajalike vaheühendite saamine - Google Patents

Meetod 2-halo-3-nitro-4-aminopüridiini valmistamiseks ja selleks vajalike vaheühendite saamine

Info

Publication number
EE200100333A
EE200100333A EEP200100333A EEP200100333A EE200100333A EE 200100333 A EE200100333 A EE 200100333A EE P200100333 A EEP200100333 A EE P200100333A EE P200100333 A EEP200100333 A EE P200100333A EE 200100333 A EE200100333 A EE 200100333A
Authority
EE
Estonia
Prior art keywords
aminopyridine
intermediates
halo
nitro
preparation
Prior art date
Application number
EEP200100333A
Other languages
English (en)
Inventor
C. Salazar Diane (Surnud)
Rodriguez Walter
P. Sherbine James
G. Woodward Rick
W. Sledeski Adam
R. Powers Matthew
K. O'brien Michael
Original Assignee
Aventis Pharmaceuticals Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharmaceuticals Products Inc. filed Critical Aventis Pharmaceuticals Products Inc.
Publication of EE200100333A publication Critical patent/EE200100333A/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
EEP200100333A 1998-12-21 1999-12-14 Meetod 2-halo-3-nitro-4-aminopüridiini valmistamiseks ja selleks vajalike vaheühendite saamine EE200100333A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11307798P 1998-12-21 1998-12-21
PCT/US1999/029643 WO2000037469A2 (en) 1998-12-21 1999-12-14 Process for preparing n6-substituted deaza-adenosine derivatives

Publications (1)

Publication Number Publication Date
EE200100333A true EE200100333A (et) 2002-08-15

Family

ID=22347487

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100333A EE200100333A (et) 1998-12-21 1999-12-14 Meetod 2-halo-3-nitro-4-aminopüridiini valmistamiseks ja selleks vajalike vaheühendite saamine

Country Status (28)

Country Link
US (1) US6184382B1 (et)
EP (1) EP1175420B1 (et)
JP (1) JP2002533343A (et)
KR (1) KR20010087425A (et)
CN (1) CN1122667C (et)
AP (1) AP1336A (et)
AT (1) ATE235493T1 (et)
AU (1) AU774155B2 (et)
BG (1) BG105624A (et)
BR (1) BR9917088A (et)
CA (1) CA2357760A1 (et)
CZ (1) CZ20012283A3 (et)
DE (1) DE69906392T2 (et)
DK (1) DK1175420T3 (et)
EA (1) EA003645B1 (et)
EE (1) EE200100333A (et)
ES (1) ES2191489T3 (et)
HK (1) HK1041607A1 (et)
HU (1) HUP0105224A3 (et)
ID (1) ID30118A (et)
IL (1) IL143843A0 (et)
NO (1) NO319789B1 (et)
NZ (1) NZ512500A (et)
PL (1) PL349154A1 (et)
PT (1) PT1175420E (et)
SK (1) SK284767B6 (et)
WO (1) WO2000037469A2 (et)
YU (1) YU51401A (et)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03006730A (es) * 1996-12-11 2003-10-24 Aventis Pharma Inc Preparacion de 4-hidroxi-3-nitro-2(1h)-piridona.
KR100446669B1 (ko) * 2002-04-04 2004-09-04 (주) 비엔씨바이오팜 2-(헤테로사이클릭-알킬아미노)피리딘 유도체, 그제조방법 및 이를 포함하는 항바이러스용 약학적 조성물
US7291603B2 (en) * 2002-07-24 2007-11-06 Ptc Therapeutics, Inc. Nucleoside compounds and their use for treating cancer and diseases associated with somatic mutations

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5561134A (en) * 1990-09-25 1996-10-01 Rhone-Poulenc Rorer Pharmaceuticals Inc. Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
US5652366A (en) * 1990-09-25 1997-07-29 Rhone-Poulenc Rorer Pharmaceuticals Inc. DI (1R)-(-)camphosulfonic acid) salt, preparation thereof and use thereof
EP0550631B1 (en) * 1990-09-25 1997-01-02 Rhone-Poulenc Rorer International (Holdings) Inc. Compounds having antihypertensive and anti-ischemic properties

Also Published As

Publication number Publication date
ATE235493T1 (de) 2003-04-15
YU51401A (sh) 2003-12-31
CN1333773A (zh) 2002-01-30
US6184382B1 (en) 2001-02-06
PL349154A1 (en) 2002-07-01
AP2001002200A0 (en) 2001-09-30
AU774155B2 (en) 2004-06-17
EP1175420B1 (en) 2003-03-26
ES2191489T3 (es) 2003-09-01
CA2357760A1 (en) 2000-06-29
WO2000037469A3 (en) 2000-09-14
SK284767B6 (sk) 2005-11-03
NO20013044L (no) 2001-08-20
PT1175420E (pt) 2003-08-29
IL143843A0 (en) 2002-04-21
BR9917088A (pt) 2006-01-31
NO319789B1 (no) 2005-09-12
CN1122667C (zh) 2003-10-01
DE69906392T2 (de) 2004-02-05
HUP0105224A3 (en) 2003-01-28
EP1175420A2 (en) 2002-01-30
HK1041607A1 (zh) 2002-07-12
BG105624A (en) 2002-01-31
JP2002533343A (ja) 2002-10-08
CZ20012283A3 (cs) 2001-10-17
WO2000037469B1 (en) 2000-11-02
DK1175420T3 (da) 2003-07-07
AP1336A (en) 2004-11-30
NO20013044D0 (no) 2001-06-19
DE69906392D1 (de) 2003-04-30
SK9072001A3 (en) 2001-12-03
HUP0105224A2 (en) 2002-06-29
EA003645B1 (ru) 2003-08-28
NZ512500A (en) 2003-01-31
EA200100697A1 (ru) 2001-12-24
KR20010087425A (ko) 2001-09-15
WO2000037469A2 (en) 2000-06-29
ID30118A (id) 2001-11-08
AU2181400A (en) 2000-07-12

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