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EE05264B1 - Prukalopriidi vesilahus suukaudseks manustamiseks ning selle valmistamismeetod - Google Patents

Prukalopriidi vesilahus suukaudseks manustamiseks ning selle valmistamismeetod

Info

Publication number
EE05264B1
EE05264B1 EEP200100539A EEP200100539A EE05264B1 EE 05264 B1 EE05264 B1 EE 05264B1 EE P200100539 A EEP200100539 A EE P200100539A EE P200100539 A EEP200100539 A EE P200100539A EE 05264 B1 EE05264 B1 EE 05264B1
Authority
EE
Estonia
Prior art keywords
prucalopride
preparation
aqueous solution
oral administration
oral
Prior art date
Application number
EEP200100539A
Other languages
English (en)
Inventor
Andr� Jos�e De Proost Eddy
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of EE200100539A publication Critical patent/EE200100539A/et
Publication of EE05264B1 publication Critical patent/EE05264B1/et

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4525Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Urology & Nephrology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
EEP200100539A 1999-04-29 2000-04-20 Prukalopriidi vesilahus suukaudseks manustamiseks ning selle valmistamismeetod EE05264B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99201335 1999-04-29
PCT/EP2000/003739 WO2000066170A1 (en) 1999-04-29 2000-04-20 Prucalopride oral solution

Publications (2)

Publication Number Publication Date
EE200100539A EE200100539A (et) 2002-12-16
EE05264B1 true EE05264B1 (et) 2010-02-15

Family

ID=8240160

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100539A EE05264B1 (et) 1999-04-29 2000-04-20 Prukalopriidi vesilahus suukaudseks manustamiseks ning selle valmistamismeetod

Country Status (36)

Country Link
US (1) US6413988B1 (et)
EP (1) EP1176982B1 (et)
JP (1) JP4773619B2 (et)
KR (1) KR100669175B1 (et)
CN (1) CN1165345C (et)
AR (1) AR023815A1 (et)
AT (1) ATE254929T1 (et)
AU (1) AU770073B2 (et)
BG (1) BG65061B1 (et)
BR (1) BRPI0010150B8 (et)
CA (1) CA2371178C (et)
CZ (1) CZ294070B6 (et)
DE (1) DE60006799T2 (et)
DK (1) DK1176982T3 (et)
EA (1) EA003904B1 (et)
EE (1) EE05264B1 (et)
ES (1) ES2211546T3 (et)
HK (1) HK1045950B (et)
HR (1) HRP20010764B1 (et)
HU (1) HU228924B1 (et)
ID (1) ID30397A (et)
IL (2) IL146152A0 (et)
JO (1) JO2181B1 (et)
MX (1) MXPA01010953A (et)
MY (1) MY119880A (et)
NO (1) NO331448B1 (et)
NZ (1) NZ515119A (et)
PL (1) PL195674B1 (et)
PT (1) PT1176982E (et)
SI (1) SI1176982T1 (et)
SK (1) SK284847B6 (et)
TR (1) TR200103121T2 (et)
TW (1) TW592709B (et)
UA (1) UA68426C2 (et)
WO (1) WO2000066170A1 (et)
ZA (1) ZA200108820B (et)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050063998A1 (en) * 1999-10-26 2005-03-24 Francois Marc Karel Jozef Oral solution containing galantamine and a sweetening agent
AU2002231627A1 (en) * 2000-11-24 2002-06-03 Janssen Pharmaceutica N.V. Use of a triple combination comprising a 5HT3 antagonist, a 5HT4 agonist and a laxative for promoting intestinal lavage
EP1467991B1 (en) 2002-01-16 2005-05-18 Janssen Pharmaceutica N.V. Prucalopride-n-oxide
JP4526247B2 (ja) * 2002-07-08 2010-08-18 第一三共株式会社 経口用セファロスポリン製剤
FI20022007A0 (fi) * 2002-11-08 2002-11-08 Juvantia Pharma Ltd Oy Oromukosaalinen valmiste ja menetelmä sen valmistamiseksi
ES2388501T3 (es) 2004-08-12 2012-10-16 Helsinn Healthcare S.A. Uso de secretagogos de la hormona de crecimiento para estimular la motilidad del sistema gastrointestinal
GB201103397D0 (et) 2011-02-28 2011-04-13 Shire Movetis N V
US8568747B1 (en) 2012-10-05 2013-10-29 Silvergate Pharmaceuticals, Inc. Enalapril compositions
US9463183B1 (en) 2015-10-30 2016-10-11 Silvergate Pharmaceuticals, Inc. Lisinopril formulations
US9669008B1 (en) 2016-03-18 2017-06-06 Silvergate Pharmaceuticals, Inc. Enalapril formulations
CN119700664B (zh) * 2025-02-28 2025-06-20 山东新时代药业有限公司 含有活性成分琥珀酸普芦卡必利的注射液及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5374637A (en) * 1989-03-22 1994-12-20 Janssen Pharmaceutica N.V. N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
GB9005014D0 (en) * 1990-03-06 1990-05-02 Janssen Pharmaceutica Nv N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives
JPH05163154A (ja) * 1991-12-13 1993-06-29 Kanebo Ltd 経口液剤
TW490465B (en) * 1994-11-24 2002-06-11 Janssen Pharmaceutica Nv Enterokinetic benzamide, the preparation process and the pharmaceutical compositions thereof
AU770580B2 (en) * 1998-11-23 2004-02-26 Janssen Pharmaceutica N.V. Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia

Also Published As

Publication number Publication date
IL146152A (en) 2006-12-31
JP4773619B2 (ja) 2011-09-14
MY119880A (en) 2005-07-29
JO2181B1 (en) 2003-04-23
AU4913700A (en) 2000-11-17
AU770073B2 (en) 2004-02-12
KR100669175B1 (ko) 2007-01-17
ES2211546T3 (es) 2004-07-16
DK1176982T3 (da) 2004-03-29
PT1176982E (pt) 2004-04-30
CA2371178C (en) 2008-03-25
NZ515119A (en) 2003-05-30
SK284847B6 (sk) 2006-01-05
HRP20010764A2 (en) 2002-12-31
BR0010150A (pt) 2002-01-15
EE200100539A (et) 2002-12-16
TW592709B (en) 2004-06-21
EP1176982B1 (en) 2003-11-26
MXPA01010953A (es) 2002-05-06
PL195674B1 (pl) 2007-10-31
TR200103121T2 (tr) 2002-05-21
CZ294070B6 (cs) 2004-09-15
EP1176982A1 (en) 2002-02-06
BRPI0010150B8 (pt) 2021-05-25
UA68426C2 (uk) 2004-08-16
ID30397A (id) 2001-11-29
HU228924B1 (en) 2013-06-28
IL146152A0 (en) 2002-07-25
SK15192001A3 (sk) 2002-03-05
BRPI0010150B1 (pt) 2015-06-23
BG65061B1 (bg) 2007-01-31
DE60006799T2 (de) 2004-09-23
NO20014794D0 (no) 2001-10-02
ATE254929T1 (de) 2003-12-15
CA2371178A1 (en) 2000-11-09
NO20014794L (no) 2001-10-02
HK1045950B (zh) 2005-05-27
EA200101150A1 (ru) 2002-04-25
HUP0202324A3 (en) 2003-03-28
SI1176982T1 (en) 2004-04-30
CN1348386A (zh) 2002-05-08
ZA200108820B (en) 2003-01-27
WO2000066170A1 (en) 2000-11-09
CZ20013735A3 (cs) 2002-02-13
NO331448B1 (no) 2012-01-02
BG106031A (en) 2002-05-31
HRP20010764B1 (hr) 2011-01-31
US6413988B1 (en) 2002-07-02
HUP0202324A2 (hu) 2002-12-28
AR023815A1 (es) 2002-09-04
DE60006799D1 (de) 2004-01-08
JP2002543161A (ja) 2002-12-17
HK1045950A1 (en) 2002-12-20
KR20020004972A (ko) 2002-01-16
CN1165345C (zh) 2004-09-08
PL352062A1 (en) 2003-07-28
EA003904B1 (ru) 2003-10-30

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Legal Events

Date Code Title Description
GB1A Change in the ownership or in the address of the owner
KB4A Valid patent at the end of a year

Effective date: 20101231

HC1A Change of owner name