ECSP15001225A - TRICYCLIC COMPOUNDS SUBSTITUTED AS INHIBITORS OF THE FIBROBLAST GROWTH FACTOR RECEPTOR - Google Patents
TRICYCLIC COMPOUNDS SUBSTITUTED AS INHIBITORS OF THE FIBROBLAST GROWTH FACTOR RECEPTORInfo
- Publication number
- ECSP15001225A ECSP15001225A ECIEPI20151225A ECPI201501225A ECSP15001225A EC SP15001225 A ECSP15001225 A EC SP15001225A EC IEPI20151225 A ECIEPI20151225 A EC IEPI20151225A EC PI201501225 A ECPI201501225 A EC PI201501225A EC SP15001225 A ECSP15001225 A EC SP15001225A
- Authority
- EC
- Ecuador
- Prior art keywords
- inhibitors
- growth factor
- tricyclic compounds
- factor receptor
- fibroblast growth
- Prior art date
Links
- 108091008794 FGF receptors Proteins 0.000 title abstract 3
- 150000001875 compounds Chemical group 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 102000044168 Fibroblast Growth Factor Receptor Human genes 0.000 title 1
- 102000052178 fibroblast growth factor receptor activity proteins Human genes 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos tricíclicos de la fórmula I, y composiciones farmacéuticas de los mismos, que son inhibidores de una o más enzimas del FGFR y son útiles en el tratamiento de enfermedades asociadas con el FGFR tales como cáncer.The present invention relates to tricyclic compounds of formula I, and pharmaceutical compositions thereof, which are inhibitors of one or more FGFR enzymes and are useful in the treatment of diseases associated with FGFR such as cancer.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261659245P | 2012-06-13 | 2012-06-13 | |
| US201261740012P | 2012-12-20 | 2012-12-20 | |
| US201361774841P | 2013-03-08 | 2013-03-08 | |
| US201561691463P | 2015-01-21 | 2015-01-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP15001225A true ECSP15001225A (en) | 2017-03-31 |
Family
ID=73007100
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECIEPI20151225A ECSP15001225A (en) | 2012-06-13 | 2015-01-13 | TRICYCLIC COMPOUNDS SUBSTITUTED AS INHIBITORS OF THE FIBROBLAST GROWTH FACTOR RECEPTOR |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP15001225A (en) |
-
2015
- 2015-01-13 EC ECIEPI20151225A patent/ECSP15001225A/en unknown
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