DK7483A - Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf - Google Patents

Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf Download PDF

Info

Publication number: DK7483A
Authority: DK; Denmark
Prior art keywords: sublicencillanic; aminoal; dioxides; derivatives; preparation
Prior art date: 1982-01-11

Application number

DK7483A

Other languages

English (en)

Other versions

DK7483D0 (da

DK166883B1 (da

Inventor

Wayne Ernest Barth

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-01-11

Filing date

1983-01-10

Publication date

1983-07-12

1982-06-14 Priority claimed from US06/388,323 external-priority patent/US4427678A/en

1982-10-21 Priority claimed from US06/434,371 external-priority patent/US4452796A/en

1983-01-10 Application filed by Pfizer filed Critical Pfizer

1983-01-10 Publication of DK7483D0 publication Critical patent/DK7483D0/da

1983-07-12 Publication of DK7483A publication Critical patent/DK7483A/da

1993-07-26 Application granted granted Critical

1993-07-26 Publication of DK166883B1 publication Critical patent/DK166883B1/da

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Medicinal Preparation (AREA)

DK007483A 1982-01-11 1983-01-10 Analogifremgangsmaade til fremstilling af 6-aminoalkylpenicillansyre-1,1-dioxider samt derivater eller salte deraf DK166883B1 (da)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
US33879782A	1982-01-11	1982-01-11
US33879782		1982-01-11
US38832482A	1982-06-14	1982-06-14
US06/388,323 US4427678A (en)	1982-01-11	1982-06-14	6-Aminomethylpenicillanic acid 1,1-dioxide derivatives as beta-lactamase inhibitors
US38832482		1982-06-14
US38832382		1982-06-14
US06/434,371 US4452796A (en)	1982-06-14	1982-10-21	6-Aminoalkylpenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
US43437182		1982-10-21

Publications (3)

Publication Number	Publication Date
DK7483D0 DK7483D0 (da)	1983-01-10
DK7483A true DK7483A (da)	1983-07-12
DK166883B1 DK166883B1 (da)	1993-07-26

Family

ID=27502592

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK007483A DK166883B1 (da)	1982-01-11	1983-01-10	Analogifremgangsmaade til fremstilling af 6-aminoalkylpenicillansyre-1,1-dioxider samt derivater eller salte deraf

Country Status (20)

Country	Link
EP (1)	EP0084925B1 (da)
JP (1)	JPH0689005B2 (da)
AU (1)	AU538468B2 (da)
BG (1)	BG42676A3 (da)
CA (1)	CA1190921A (da)
DD (2)	DD209462A5 (da)
DE (1)	DE3362826D1 (da)
DK (1)	DK166883B1 (da)
ES (2)	ES518912A0 (da)
FI (1)	FI79112C (da)
GR (1)	GR77152B (da)
HU (1)	HU189211B (da)
IE (1)	IE54390B1 (da)
IL (1)	IL67647A (da)
NO (6)	NO830046L (da)
NZ (1)	NZ202982A (da)
PL (1)	PL142315B1 (da)
PT (1)	PT76077B (da)
RO (2)	RO84910B (da)
YU (1)	YU43646B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4502990A (en) *	1983-06-06	1985-03-05	Pfizer Inc.	Process for 6-(aminomethyl)penicillanic acid 1,1-dioxide and derivatives thereof
US4499017A (en) *	1983-06-06	1985-02-12	Pfizer Inc.	Beta-lactamase inhibiting 6-(alkoxyamino-methyl) penicillanic acid 1,1-dioxide and derivatives
JPS60239489A (ja) *	1984-05-15	1985-11-28	Meiji Seika Kaisha Ltd	６−エピペニシリンスルホン化合物及びその製造方法
GB2206579B (en) *	1987-07-10	1991-05-29	Erba Farmitalia	6a and 6b-(substituted methyl)-penicillanic acid derivatives
AU2008253257B2 (en) *	2007-05-21	2013-10-03	Hans Rudolf Pfaendler	Bactericidal anti-MRSA active pharmaceutical composition containing carbapenems

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4237051A (en) *	1979-04-19	1980-12-02	Schering Corporation	Stereospecific production of 6- or 7-carbon-substituted-β-lactams
DE2927004A1 (de) *	1979-07-04	1981-05-27	Bayer Ag, 5090 Leverkusen	Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) *	1979-10-22	1981-09-01	Pfizer Inc.	Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

1983
- 1983-01-04 RO RO109609A patent/RO84910B/ro unknown
- 1983-01-04 RO RO83113375A patent/RO87705A/ro unknown
- 1983-01-05 EP EP83300042A patent/EP0084925B1/en not_active Expired
- 1983-01-05 DE DE8383300042T patent/DE3362826D1/de not_active Expired
- 1983-01-07 GR GR70215A patent/GR77152B/el unknown
- 1983-01-07 NO NO830046A patent/NO830046L/no unknown
- 1983-01-10 CA CA000419181A patent/CA1190921A/en not_active Expired
- 1983-01-10 PT PT76077A patent/PT76077B/pt not_active IP Right Cessation
- 1983-01-10 BG BG059284A patent/BG42676A3/xx unknown
- 1983-01-10 IE IE42/83A patent/IE54390B1/en not_active IP Right Cessation
- 1983-01-10 IL IL67647A patent/IL67647A/xx not_active IP Right Cessation
- 1983-01-10 HU HU8370A patent/HU189211B/hu not_active IP Right Cessation
- 1983-01-10 FI FI830081A patent/FI79112C/fi not_active IP Right Cessation
- 1983-01-10 YU YU44/83A patent/YU43646B/xx unknown
- 1983-01-10 DK DK007483A patent/DK166883B1/da active
- 1983-01-10 NZ NZ202982A patent/NZ202982A/en unknown
- 1983-01-10 AU AU10232/83A patent/AU538468B2/en not_active Ceased
- 1983-01-11 DD DD83247166A patent/DD209462A5/de not_active IP Right Cessation
- 1983-01-11 PL PL1983240108A patent/PL142315B1/pl unknown
- 1983-01-11 DD DD83262053A patent/DD218365A5/de not_active IP Right Cessation
- 1983-01-11 JP JP58002768A patent/JPH0689005B2/ja not_active Expired - Lifetime
- 1983-01-11 ES ES518912A patent/ES518912A0/es active Granted
- 1983-08-30 ES ES525238A patent/ES8507147A1/es not_active Expired
- 1983-09-22 NO NO833415A patent/NO833415L/no unknown
- 1983-09-22 NO NO833416A patent/NO833416L/no unknown
1984
- 1984-03-20 NO NO841069A patent/NO841069L/no unknown
- 1984-03-20 NO NO841070A patent/NO841070L/no unknown
- 1984-03-20 NO NO841068A patent/NO841068L/no unknown

Also Published As

Publication number	Publication date
DD209462A5 (de)	1984-05-09
GR77152B (da)	1984-09-07
JPS58126889A (ja)	1983-07-28
FI79112C (fi)	1989-11-10
YU43646B (en)	1989-10-31
NO841068L (no)	1983-07-12
IL67647A0 (en)	1983-05-15
NO833416L (no)	1983-07-12
ES8403489A1 (es)	1984-03-16
ES525238A0 (es)	1985-08-16
NO841070L (no)	1983-07-12
RO87705A (ro)	1985-10-31
EP0084925A1 (en)	1983-08-03
RO84910A (ro)	1984-08-17
NZ202982A (en)	1986-04-11
NO833415L (no)	1983-07-12
DE3362826D1 (en)	1986-05-15
IL67647A (en)	1986-08-31
IE54390B1 (en)	1989-09-13
IE830042L (en)	1983-07-11
RO84910B (ro)	1984-09-30
YU4483A (en)	1986-02-28
RO87705B (ro)	1985-10-01
DK7483D0 (da)	1983-01-10
JPH0689005B2 (ja)	1994-11-09
PT76077A (en)	1983-02-01
AU538468B2 (en)	1984-08-16
EP0084925B1 (en)	1986-04-09
DK166883B1 (da)	1993-07-26
AU1023283A (en)	1983-07-21
HU189211B (en)	1986-06-30
PL240108A1 (en)	1985-08-13
PL142315B1 (en)	1987-10-31
DD218365A5 (de)	1985-02-06
CA1190921A (en)	1985-07-23
ES518912A0 (es)	1984-03-16
FI830081L (fi)	1983-07-12
ES8507147A1 (es)	1985-08-16
NO841069L (no)	1983-07-12
FI830081A0 (fi)	1983-01-10
BG42676A3 (en)	1988-01-15
PT76077B (en)	1986-01-09
FI79112B (fi)	1989-07-31
NO830046L (no)	1983-07-12

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NO821087L (no)	1982-10-07	Fremgangsmaate for fremstilling av cyklobutan-derivater.
DK112582A (da)	1982-09-17	Fremgangsmaade til fremstilling af triazolonderivater
DK307883A (da)	1984-01-06	Carbostyrilderivater samt fremgangsmaade til fremstilling deraf
DK66582A (da)	1982-08-18	Fremgangsmaade til fremstilling af carbostyrilderivater
DK158269C (da)	1990-10-08	Analogifremgangsmaade til fremstilling af morpholinyldaunorubicin- eller morpholinyldoxorubicinderivater
DK106897A (da)	1997-09-17	Fremgangsmåde til fremstilling af urinstofderivater
DK491582A (da)	1983-05-10	Fremgangsmaade til fremstilling af morphinanderivater
DK352082A (da)	1983-02-08	Fremgangsmaade til fremstilling af ergopeptinderivater
FI832004A7 (fi)	1983-12-04	Menetelmä 1-sulfo-2-oksoatsetidiini- johdannaisten valmistamiseksi.
ES517862A0 (es)	1984-03-01	Derivados de alcanosulfonanilida.
NO155693C (no)	1987-05-13	Fremgangsmaate for fremstilling av eburnamoninderivater.
ES522823A0 (es)	1984-08-16	Derivados de 6 -metilprednisolona.
DK116982A (da)	1982-09-18	Fremgangsmaade til fremstilling af alkylendioxybenzenderivater
DK7483A (da)	1983-07-12	Fremgangsmaade til fremstilling af 6-aminoalkylpencillansyre-1,1-dioxider samt derivater deraf
FI832919A7 (fi)	1984-02-14	Menetelmä N-substituoidun nikotiiniamidi-1-oksidin ja sen suolojen valmistamiseksi.
DK113483D0 (da)	1983-03-08	Fremgangsmade til fremstilling af 3,4-diphenyl-5-methylpyrazolderivater
NO157143C (no)	1988-01-27	Fremgangsmaate for fremstilling av karbapen-2-em-derivater.
DK70482A (da)	1982-08-20	Fremgangsmaade til fremstilling af diazolderivater
DK423284A (da)	1985-03-09	Naphthalenylimidazopyridin og derivater heraf samt fremgangsmaade til fremstilling af saadanne forbindelser
DK364483D0 (da)	1983-08-10	14-aminosteroid-derivater samt fremgangsmade til fremstilling deraf
DK570082A (da)	1983-06-26	4-cyan-2-azetidinoner samt fremgangsmaade til fremstilling af saadanne
ES517428A0 (es)	1983-08-16	Procedimiento de preparacion de derivados bencilidenicos.
DK375882A (da)	1983-02-27	Fremgangsmaade til fremstilling af benzisoxazolderivater
DK135081A (da)	1981-10-04	Fr&mgangsmaade til fremstilling af thiazoler
ES522653A0 (es)	1984-09-16	Procedimiento de preparacion de derivados de piperacina.