DK629889A - Aminosyrederivater, deres fremstilling og anvendelse som laegemidler - Google Patents

Aminosyrederivater, deres fremstilling og anvendelse som laegemidler Download PDF

Info

Publication number: DK629889A
Authority: DK; Denmark
Prior art keywords: preparation; amino acid; pharmaceuticals; acid derivatives; radical
Prior art date: 1988-12-14

Application number

DK629889A

Other languages

Danish (da)

English (en)

Other versions

DK629889D0 (da

Inventor

Wolfgang Rueger

Hansjoerg Urbach

Dieter Ruppert

Bernward Schoelkens

Original Assignee

Hoechst Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-12-14

Filing date

1989-12-13

Publication date

1990-06-15

1989-12-13 Application filed by Hoechst Ag filed Critical Hoechst Ag

1989-12-13 Publication of DK629889D0 publication Critical patent/DK629889D0/da

1990-06-15 Publication of DK629889A publication Critical patent/DK629889A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0227—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Virology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Pyridine Compounds (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)

DK629889A 1988-12-14 1989-12-13 Aminosyrederivater, deres fremstilling og anvendelse som laegemidler DK629889A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE3842067A DE3842067A1 (de)	1988-12-14	1988-12-14	Enzym-hemmende aminosaeurederivate, verfahren zu ihrer herstellung, diese enthaltende mittel und ihre verwendung

Publications (2)

Publication Number	Publication Date
DK629889D0 DK629889D0 (da)	1989-12-13
DK629889A true DK629889A (da)	1990-06-15

Family

ID=6369139

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK629889A DK629889A (da)	1988-12-14	1989-12-13	Aminosyrederivater, deres fremstilling og anvendelse som laegemidler

Country Status (16)

Country	Link
US (1)	US5185324A (no)
EP (1)	EP0373549B1 (no)
JP (1)	JPH02204475A (no)
KR (1)	KR900009691A (no)
AT (1)	ATE93863T1 (no)
AU (1)	AU632519B2 (no)
CA (1)	CA2005422A1 (no)
DE (2)	DE3842067A1 (no)
DK (1)	DK629889A (no)
ES (1)	ES2059688T3 (no)
FI (1)	FI895921A7 (no)
HU (1)	HU205369B (no)
IL (1)	IL92660A0 (no)
NO (1)	NO895002L (no)
PT (1)	PT92558B (no)
ZA (1)	ZA899507B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6313094B1 (en)	1990-12-11	2001-11-06	Japan Energy Corporation	β-amino-α-hydroxycarboxylic acid derivatives and HIV protease inhibitors
US5554728A (en) *	1991-07-23	1996-09-10	Nexstar Pharmaceuticals, Inc.	Lipid conjugates of therapeutic peptides and protease inhibitors
US5888992A (en) *	1992-03-11	1999-03-30	Narhex Limited	Polar substituted hydrocarbons
US6071895A (en) *	1992-03-11	2000-06-06	Narhex Limited	Polar-substituted hydrocarbons
CA2130754C (en) *	1992-03-11	2005-02-08	Damian W. Grobelny	Amine derivatives of oxo- and hydroxy-substituted hydrocarbons
DE69333270T2 (de)	1992-03-11	2004-08-05	Narhex Ltd.	Aminderivate von oxo- und hydroxy- substituierten kohlenwasserstoffen
US5559256A (en) *	1992-07-20	1996-09-24	E. R. Squibb & Sons, Inc.	Aminediol protease inhibitors
IL110898A0 (en) *	1993-09-10	1994-11-28	Narhex Australia Pty Ltd	Polar-substituted hydrocarbons
AU725432B2 (en) *	1996-04-17	2000-10-12	Centaur Pharmaceuticals, Inc.	Nitrone free radical trap treatment of dementia associated with AIDS virus (HIV-1) infection
FR3012460B1 (fr)	2013-10-25	2015-12-11	Michelin & Cie	Composition de caoutchouc comprenant un elastomere dienique portant des fonctions imidazole reparties de facon aleatoire le long de la chaine
FR3012451B1 (fr)	2013-10-25	2016-11-11	Michelin & Cie	Compose 1,3-dipolaire portant une fonction imidazole
FR3012458B1 (fr)	2013-10-25	2015-10-30	Michelin & Cie	Composition de caoutchouc comprenant un additif compose 1,3-dipolaire portant une fonction imidazole
WO2021220231A1 (en)	2020-05-01	2021-11-04	Pi Industries Ltd.	Composition of propineb and metominostrobin
EP4079748A1 (en) *	2021-04-23	2022-10-26	Insusense ApS	Modulators of sortilin activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1987004349A1 (en) *	1986-01-16	1987-07-30	Joseph Dellaria	Peptide analogs
DE3626130A1 (de) *	1986-08-01	1988-02-11	Merck Patent Gmbh	Aminosaeurederivate

1988
- 1988-12-14 DE DE3842067A patent/DE3842067A1/de not_active Withdrawn
1989
- 1989-12-11 ES ES89122794T patent/ES2059688T3/es not_active Expired - Lifetime
- 1989-12-11 AT AT89122794T patent/ATE93863T1/de not_active IP Right Cessation
- 1989-12-11 EP EP89122794A patent/EP0373549B1/de not_active Expired - Lifetime
- 1989-12-11 DE DE89122794T patent/DE58905462D1/de not_active Expired - Fee Related
- 1989-12-12 US US07/448,903 patent/US5185324A/en not_active Expired - Fee Related
- 1989-12-12 IL IL92660A patent/IL92660A0/xx unknown
- 1989-12-12 KR KR1019890018354A patent/KR900009691A/ko not_active Withdrawn
- 1989-12-12 FI FI895921A patent/FI895921A7/fi not_active IP Right Cessation
- 1989-12-13 PT PT92558A patent/PT92558B/pt not_active IP Right Cessation
- 1989-12-13 ZA ZA899507A patent/ZA899507B/xx unknown
- 1989-12-13 JP JP1321602A patent/JPH02204475A/ja active Pending
- 1989-12-13 AU AU46115/89A patent/AU632519B2/en not_active Expired - Fee Related
- 1989-12-13 DK DK629889A patent/DK629889A/da not_active Application Discontinuation
- 1989-12-13 NO NO89895002A patent/NO895002L/no unknown
- 1989-12-13 CA CA002005422A patent/CA2005422A1/en not_active Abandoned
- 1989-12-14 HU HU896606A patent/HU205369B/hu not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR900009691A (ko)	1990-07-05
PT92558A (pt)	1990-06-29
FI895921A0 (fi)	1989-12-12
DE58905462D1 (de)	1993-10-07
ES2059688T3 (es)	1994-11-16
FI895921A7 (fi)	1990-06-15
PT92558B (pt)	1995-08-09
NO895002D0 (no)	1989-12-13
JPH02204475A (ja)	1990-08-14
HUT53664A (en)	1990-11-28
EP0373549A2 (de)	1990-06-20
ATE93863T1 (de)	1993-09-15
HU205369B (en)	1992-04-28
EP0373549B1 (de)	1993-09-01
AU4611589A (en)	1990-06-28
EP0373549A3 (de)	1991-08-21
NO895002L (no)	1990-06-15
ZA899507B (en)	1990-08-29
DK629889D0 (da)	1989-12-13
IL92660A0 (en)	1990-08-31
HU896606D0 (en)	1990-02-28
DE3842067A1 (de)	1990-06-21
US5185324A (en)	1993-02-09
AU632519B2 (en)	1993-01-07
CA2005422A1 (en)	1990-06-14

Publication	Publication Date	Title
ES539658A0 (es)	1986-04-01	Procedimiento de preparacion de nuevos derivados de la xan- tina y de sus sales de adicion con acidos apropiados
DK629889A (da)	1990-06-15	Aminosyrederivater, deres fremstilling og anvendelse som laegemidler
NO834626L (no)	1984-06-18	Derivater av cis, endo-2-azabicyklo-(5.3.0)-dekan-3-karboksylsyre, fremgangsmaate til deres fremstilling, midler som inneholder disse og deres anvendelse
NO903952L (no)	1991-03-13	Fremgangsmaate for fremstilling av aminosyrederivater med reninhemmende egenskaper, og anvendelse av midler som inneholder disse.
DK499088D0 (da)	1988-09-08	1-oe(2-pyrimidinyl)-aminoalkylaapiperidinderivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende saadanne derivater
DK359387A (da)	1988-01-12	Oploesninger af oxazaphosphoriner med forbedret stabilitet og fremgangsmaade til deres fremstilling
DK0461986T3 (da)	1996-05-28	Hexahydroazepinderivater, en fremgangsmåde til fremstilling heraf og farmaceutiske midler indeholdende disse
DK0452204T3 (da)	1994-10-24	Hidtil ukendte 3-aminochromanderivater, fremgangsmåde til fremstilling heraf og farmaceutiske midler, som indeholder dem
DK440987D0 (da)	1987-08-24	Thyroninderivater, deres fremstilling og anvendelse
ES2054989T3 (es)	1994-08-16	Derivados de aminodiol inhibidores de renina.
DK279988D0 (da)	1988-05-20	Spiro(4,5)decanderivater, fremgangsmaade til deres fremstilling og farmaceutiske midler indeholdende dem
NO171020C (no)	1993-01-13	Nye tyroninderivater og anvendelse derav
DK0635491T3 (da)	1997-11-03	(Thia)cycloalkylab indoler, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse forbindelser.
FI870299A7 (fi)	1987-01-23	Amin, som aer anvaendbart som mellanprodukt vid framstaellning av l-aspartyl-d -aminosyradipeptidamider.
DK378885D0 (da)	1985-08-20	1-(n-(alfa-amino-alfa-methylacetyl)aminophenyl)-2-aminopropanonderivater, fremgangsmaade til deres fremstilling og deres anvendelse i terapien

Legal Events

Date	Code	Title	Description
1992-12-14	ATS	Application withdrawn