DK543386A - Thienooxazinoner deres fremstilling og anvendelse - Google Patents

Thienooxazinoner deres fremstilling og anvendelse

Info

Publication number: DK543386A
Authority: DK; Denmark
Prior art keywords: thienooxazinones; preparation
Prior art date: 1985-11-14

Application number

DK543386A

Other languages

English (en)

Other versions

DK543386D0 (da

Inventor

Werner Hallenbach

Hans Lindel

Friedrich Berschauer

Martin Scheer

Anno De Jong

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-11-14

Filing date

1986-11-13

Publication date

1987-05-15

1986-11-13 Application filed by Bayer Ag filed Critical Bayer Ag

1986-11-13 Publication of DK543386D0 publication Critical patent/DK543386D0/da

1987-05-15 Publication of DK543386A publication Critical patent/DK543386A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/78—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Pregnancy & Childbirth (AREA)
Gynecology & Obstetrics (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Fodder In General (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK543386A 1985-11-14 1986-11-13 Thienooxazinoner deres fremstilling og anvendelse DK543386A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19853540377 DE3540377A1 (de)	1985-11-14	1985-11-14	Thienooxazinone, verfahren zu ihrer herstellung und ihre verwendung als leistungsfoerderer

Publications (2)

Publication Number	Publication Date
DK543386D0 DK543386D0 (da)	1986-11-13
DK543386A true DK543386A (da)	1987-05-15

Family

ID=6285959

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK543386A DK543386A (da)	1985-11-14	1986-11-13	Thienooxazinoner deres fremstilling og anvendelse

Country Status (7)

Country	Link
US (1)	US4760063A (da)
EP (1)	EP0223140A2 (da)
JP (1)	JPS62114989A (da)
DE (1)	DE3540377A1 (da)
DK (1)	DK543386A (da)
IL (1)	IL80588A0 (da)
ZA (1)	ZA868609B (da)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5693374A (en)	1994-06-23	1997-12-02	Fuji Photo Film Co., Ltd.	Alpha-resorcyclic acid ester derivatives and recording materials using the same
US6344476B1 (en)	1997-05-23	2002-02-05	Bayer Corporation	Inhibition of p38 kinase activity by aryl ureas
US7517880B2 (en) *	1997-12-22	2009-04-14	Bayer Pharmaceuticals Corporation	Inhibition of p38 kinase using symmetrical and unsymmetrical diphenyl ureas
US7329670B1 (en)	1997-12-22	2008-02-12	Bayer Pharmaceuticals Corporation	Inhibition of RAF kinase using aryl and heteroaryl substituted heterocyclic ureas
US20080300281A1 (en) *	1997-12-22	2008-12-04	Jacques Dumas	Inhibition of p38 Kinase Activity Using Aryl and Heteroaryl Substituted Heterocyclic Ureas
US20080269265A1 (en) *	1998-12-22	2008-10-30	Scott Miller	Inhibition Of Raf Kinase Using Symmetrical And Unsymmetrical Substituted Diphenyl Ureas
US7928239B2 (en)	1999-01-13	2011-04-19	Bayer Healthcare Llc	Inhibition of RAF kinase using quinolyl, isoquinolyl or pyridyl ureas
RU2319693C9 (ru) *	1999-01-13	2008-08-20	Байер Копэрейшн	Производные мочевины (варианты), фармацевтическая композиция (варианты) и способ лечения заболевания, связанного с ростом раковых клеток (варианты)
US8124630B2 (en)	1999-01-13	2012-02-28	Bayer Healthcare Llc	ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
EP1140840B1 (en)	1999-01-13	2006-03-22	Bayer Pharmaceuticals Corp.	-g(v)-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
WO2000041698A1 (en)	1999-01-13	2000-07-20	Bayer Corporation	φ-CARBOXY ARYL SUBSTITUTED DIPHENYL UREAS AS p38 KINASE INHIBITORS
HN2000000051A (es) *	1999-05-19	2001-02-02	Pfizer Prod Inc	Derivados heterociclicos utiles como agentes anticancerosos
US7235576B1 (en)	2001-01-12	2007-06-26	Bayer Pharmaceuticals Corporation	Omega-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
US7371763B2 (en)	2001-04-20	2008-05-13	Bayer Pharmaceuticals Corporation	Inhibition of raf kinase using quinolyl, isoquinolyl or pyridyl ureas
RU2324696C2 (ru) *	2001-08-30	2008-05-20	Ализайм Терапевтикс Лимитед	Тиено-(1,3)-оксазин-4-оны, обладающие ингибирующей активностью по отношению к липазе
SI2305255T1 (sl) *	2001-12-03	2012-10-30	Bayer Healthcare Llc	Arilsečninske spojine v kombinaciji z drugimi citostatičnimi ali citotoksičnimi sredstvi za zdravljenje človeških rakov
JP4668536B2 (ja) *	2001-12-20	2011-04-13	オーエスアイ・ファーマスーティカルズ・インコーポレーテッド	膵臓リパーゼ阻害化合物、その合成および使用
US20040023961A1 (en) *	2002-02-11	2004-02-05	Bayer Corporation	Aryl ureas with raf kinase and angiogenisis inhibiting activity
AU2003209119A1 (en)	2002-02-11	2003-09-04	Bayer Pharmaceuticals Corporation	Pyridine, quinoline, and isoquinoline n-oxides as kinase inhibitors
WO2003068228A1 (en)	2002-02-11	2003-08-21	Bayer Pharmaceuticals Corporation	Aryl ureas with angiogenesis inhibiting activity
CN1318404C (zh)	2002-02-11	2007-05-30	拜耳制药公司	作为激酶抑制剂的芳基脲类化合物
US7557129B2 (en)	2003-02-28	2009-07-07	Bayer Healthcare Llc	Cyanopyridine derivatives useful in the treatment of cancer and other disorders
DE602004007382T2 (de)	2003-05-20	2008-04-17	Bayer Pharmaceuticals Corp., West Haven	Diaryl-harnstoffe für durch pdgfr vermittelte krankheiten
NZ544920A (en)	2003-07-23	2009-11-27	Bayer Healthcare Llc	4{4-[3-(4-chloro-3-trifluoromethylphenyl)-ureido]-3-fluorophenoxy}-pyridine-2-carboxylic acid methylamide and metabolites for the treatment and prevention of diseases and conditions
WO2005110994A2 (en)	2004-04-30	2005-11-24	Bayer Pharmaceuticals Corporation	Substituted pyrazolyl urea derivatives useful in the treatment of cancer

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2315303A1 (de) *	1973-03-27	1974-10-17	Bayer Ag	Verfahren zur herstellung von n-substituierten 2-amino-3,1-benzoxazin-4-onen
US4036979A (en) *	1974-01-25	1977-07-19	American Cyanamid Company	Compositions containing 4,5,6,7-tetrahydrobenz[b]thien-4-yl-ureas or derivatives and methods of enhancing growth rate
US4234581A (en) *	1975-09-10	1980-11-18	Mead Johnson & Company	Thieno[2,3-d]oxazines

1985
- 1985-11-14 DE DE19853540377 patent/DE3540377A1/de not_active Withdrawn
1986
- 1986-11-03 EP EP86115191A patent/EP0223140A2/de not_active Withdrawn
- 1986-11-06 JP JP61262869A patent/JPS62114989A/ja active Pending
- 1986-11-11 IL IL80588A patent/IL80588A0/xx unknown
- 1986-11-12 US US06/929,921 patent/US4760063A/en not_active Expired - Fee Related
- 1986-11-13 ZA ZA868609A patent/ZA868609B/xx unknown
- 1986-11-13 DK DK543386A patent/DK543386A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
US4760063A (en)	1988-07-26
EP0223140A2 (de)	1987-05-27
DK543386D0 (da)	1986-11-13
ZA868609B (en)	1987-07-29
IL80588A0 (en)	1987-02-27
DE3540377A1 (de)	1987-05-21
JPS62114989A (ja)	1987-05-26

Publication	Publication Date	Title
DK21986D0 (da)	1986-01-17	Tiazolidindionderivater og deres fremstilling og anvendelse
DK289886A (da)	1986-12-22	Substituerede 3-phenyl-4-cyanopyrrol-derivater samt deres fremstilling og anvendelse
DK543386A (da)	1987-05-15	Thienooxazinoner deres fremstilling og anvendelse
DK129386A (da)	1986-09-22	Iodpropargylethere, deres fremstilling og anvendelse
DK546186A (da)	1987-05-17	Substituerede benzylethere, deres fremstilling og anvendelse
DK29686A (da)	1986-07-23	13beta-alkyl-milbemycinderivater samt deres fremstilling og anvendelse
DK519586D0 (da)	1986-10-30	1-aryl-4-nitro-pyrazoler, deres fremstilling og anvendelse
DK365286D0 (da)	1986-07-31	7-oxabicycloheptan-substituerede disyre-diamid-prosta-glandin-analoge og deres anvendelse
DK515386A (da)	1987-04-30	Benzoylurinstofsalte samt deres fremstilling og anvendelse
DK380286D0 (da)	1986-08-08	Sulfonamider, deres fremstilling og anvendelse
DK617886D0 (da)	1986-12-19	1-aryl-pyrazoler, deres fremstilling og anvendelse
DK396886D0 (da)	1986-08-20	Gem-dihalogen-1,8-diamino-4-azaoctaner, deres fremstilling og anvendelse
DK172486D0 (da)	1986-04-16	Heterocyclyl-penem-forbindelser samt deres fremstilling og anvendelse
DK548586A (da)	1987-05-19	Thienylsulfonylguanidin-derivater, deres fremstilling og anvendelse
DK377786A (da)	1987-02-09	1-aryl-5-hydrazino-pyrazoler, deres fremstilling og anvendelse
DK77286A (da)	1986-08-21	1-0-acylerede hexosederivater samt deres fremstilling og anvendelse
DK206686A (da)	1986-11-07	Acylaminomethyl-penem-forbindelser samt deres fremstilling og anvendelse
DK393986D0 (da)	1986-08-19	Lactamamider, deres fremstilling og anvendelse
DK437986A (da)	1987-03-14	1-amino-3-phenyl-propan-2-ol-derivater samt deres fremstilling og anvendelse
DK478586A (da)	1987-04-09	Polyhydroxyalkyl-oligourinstoffer og deres anvendelse
DK451486D0 (da)	1986-09-22	Alkenylazoler, deres fremstilling og anvendelse
DK195086D0 (da)	1986-04-29	Substituerede azolylmethylethere, deres fremstilling og anvendelse somfungicide midler
DK540786A (da)	1987-05-14	2-hydroxybenzamider, deres fremstilling og anvendelse
DK482385D0 (da)	1985-10-21	Fluorerede resorcinolethere samt deres fremstilling og anvendelse
DK471185D0 (da)	1985-10-15	4-acylresorcinolethere samt deres fremstilling og anvendelse

Legal Events

Date	Code	Title
1987-12-07	ATS	Application withdrawn
1988-11-07	ATS	Application withdrawn
1989-02-13	ATS	Application withdrawn