DK540879A - METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF - Google Patents
METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOFInfo
- Publication number
- DK540879A DK540879A DK540879A DK540879A DK540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A DK 540879 A DK540879 A DK 540879A
- Authority
- DK
- Denmark
- Prior art keywords
- piperidinoquinazoline
- derivatives
- salts
- amino
- preparing
- Prior art date
Links
- MDGLKMXWHKGENE-UHFFFAOYSA-N 2-piperidin-1-ylquinazolin-4-amine Chemical class N=1C2=CC=CC=C2C(N)=NC=1N1CCCCC1 MDGLKMXWHKGENE-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7903398 | 1979-01-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK540879A true DK540879A (en) | 1980-08-01 |
Family
ID=10502852
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK540879A DK540879A (en) | 1979-01-31 | 1979-12-18 | METHOD OF PREPARING 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES AND SALTS THEREOF |
Country Status (28)
| Country | Link |
|---|---|
| JP (1) | JPS55104278A (en) |
| AR (1) | AR222208A1 (en) |
| AT (1) | AT373595B (en) |
| BE (1) | BE881448A (en) |
| CA (1) | CA1131636A (en) |
| CS (1) | CS231970B2 (en) |
| DD (1) | DD148720A5 (en) |
| DE (1) | DE3003323A1 (en) |
| DK (1) | DK540879A (en) |
| ES (1) | ES488129A0 (en) |
| FI (1) | FI63936C (en) |
| FR (1) | FR2447919A1 (en) |
| GR (1) | GR73626B (en) |
| HU (1) | HU184233B (en) |
| IE (1) | IE800178L (en) |
| IL (1) | IL59252A (en) |
| IT (1) | IT1149902B (en) |
| LU (1) | LU82115A1 (en) |
| NL (1) | NL8000571A (en) |
| NO (1) | NO800230L (en) |
| NZ (1) | NZ192744A (en) |
| PH (1) | PH15436A (en) |
| PL (1) | PL121890B1 (en) |
| PT (1) | PT70749A (en) |
| SE (1) | SE8000699L (en) |
| SU (1) | SU895291A3 (en) |
| YU (1) | YU22980A (en) |
| ZA (1) | ZA80557B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2483920A1 (en) * | 1980-06-09 | 1981-12-11 | Synthelabo | Antihypertensive piperidino quinazoline(s) - prepd. from benzyloxy piperidine and a 2:halo-4:amino 6,7-di:methoxy quinazoline |
| ES8405389A1 (en) * | 1981-09-09 | 1983-11-01 | Orion Yhtymae Oy | Substituted piperidinyl quinazolines. |
| US5280032A (en) * | 1989-02-14 | 1994-01-18 | Toyama Chemical Co., Ltd. | 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same |
| WO2013070852A2 (en) * | 2011-11-08 | 2013-05-16 | Emory University | Compounds and compositions used to epigenetically transform cells and methods related thereto |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1088068A (en) * | 1977-11-16 | 1980-10-21 | Simon F. Campbell | Piperidino-quinazolines |
| GB2021108B (en) * | 1978-05-18 | 1982-07-21 | Pfizer Ltd | 6,7 - di - 4 - amino - 2 - quinazolines |
-
1979
- 1979-01-30 IE IE800178A patent/IE800178L/en unknown
- 1979-12-18 DK DK540879A patent/DK540879A/en not_active Application Discontinuation
-
1980
- 1980-01-28 PH PH23559A patent/PH15436A/en unknown
- 1980-01-29 IT IT19537/80A patent/IT1149902B/en active
- 1980-01-29 SE SE8000699A patent/SE8000699L/en not_active Application Discontinuation
- 1980-01-29 CS CS80607A patent/CS231970B2/en unknown
- 1980-01-29 YU YU00229/80A patent/YU22980A/en unknown
- 1980-01-29 NZ NZ192744A patent/NZ192744A/en unknown
- 1980-01-29 FI FI800252A patent/FI63936C/en not_active IP Right Cessation
- 1980-01-29 AT AT0046980A patent/AT373595B/en not_active IP Right Cessation
- 1980-01-29 IL IL59252A patent/IL59252A/en unknown
- 1980-01-30 BE BE0/199187A patent/BE881448A/en not_active IP Right Cessation
- 1980-01-30 CA CA344,714A patent/CA1131636A/en not_active Expired
- 1980-01-30 NO NO800230A patent/NO800230L/en unknown
- 1980-01-30 JP JP990580A patent/JPS55104278A/en active Granted
- 1980-01-30 PL PL1980221683A patent/PL121890B1/en unknown
- 1980-01-30 ZA ZA00800557A patent/ZA80557B/en unknown
- 1980-01-30 HU HU80202A patent/HU184233B/en unknown
- 1980-01-30 DE DE19803003323 patent/DE3003323A1/en not_active Ceased
- 1980-01-30 NL NL8000571A patent/NL8000571A/en not_active Application Discontinuation
- 1980-01-30 PT PT70749A patent/PT70749A/en unknown
- 1980-01-30 FR FR8002012A patent/FR2447919A1/en active Granted
- 1980-01-30 AR AR279793A patent/AR222208A1/en active
- 1980-01-30 SU SU802877159A patent/SU895291A3/en active
- 1980-01-31 DD DD80218769A patent/DD148720A5/en unknown
- 1980-01-31 ES ES488129A patent/ES488129A0/en active Granted
- 1980-01-31 LU LU82115A patent/LU82115A1/en unknown
- 1980-02-11 GR GR61081A patent/GR73626B/el unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ATS | Application withdrawn |