DK530480A - Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin - Google Patents
Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicinInfo
- Publication number
- DK530480A DK530480A DK530480A DK530480A DK530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A DK 530480 A DK530480 A DK 530480A
- Authority
- DK
- Denmark
- Prior art keywords
- ethanon
- piperidyl
- quinolyl
- intermediates
- medicine
- Prior art date
Links
- SJPWBZYZHVUQRD-UHFFFAOYSA-N 2-piperidin-4-yl-1-quinolin-4-ylethanone Chemical class C=1C=NC2=CC=CC=C2C=1C(=O)CC1CCNCC1 SJPWBZYZHVUQRD-UHFFFAOYSA-N 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/34—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7931396A FR2471981A1 (fr) | 1979-12-21 | 1979-12-21 | Nouveaux derives de la (piperidyl-4)-2 (quinolyl-4)-1 ethanone, produits intermediaires et procedes pour leur preparation, et leur utilisation comme medicaments |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK530480A true DK530480A (da) | 1981-06-22 |
Family
ID=9233056
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK530480A DK530480A (da) | 1979-12-21 | 1980-12-12 | Hidtil ukendte derivater af 2-(4-piperidyl)-1-(4-quinolyl)-ethanon mellemprodukter og fremgangsmaader til deres fremstilling og deres anvendelse som medicin |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US4433150A (da) |
| EP (1) | EP0031753B1 (da) |
| JP (1) | JPS5699476A (da) |
| AT (1) | AT376670B (da) |
| CA (1) | CA1178589A (da) |
| DE (1) | DE3069243D1 (da) |
| DK (1) | DK530480A (da) |
| ES (3) | ES498017A0 (da) |
| FR (1) | FR2471981A1 (da) |
| IE (1) | IE51124B1 (da) |
| NO (1) | NO155137C (da) |
| PT (1) | PT72212A (da) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7908031A (nl) * | 1979-11-01 | 1981-06-01 | Acf Chemiefarma Nv | Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen. |
| US4442107A (en) * | 1980-03-06 | 1984-04-10 | Acf Chemiefarma N.V. | Quinoline derivatives, pharmaceutical compositions containing such compounds, and methods for treating cardiovascular conditions with them |
| FR2495470A1 (fr) * | 1980-12-05 | 1982-06-11 | Pharmindustrie | Nouveaux medicaments a base de derives de (quinolyl-4)-1 (piperidyl-4)-2 ethanol ou (quinolyl-4)-1 (piperidyl-4)-3 propanol |
| FR2582514B1 (fr) * | 1985-05-30 | 1988-02-19 | Rhone Poulenc Sante | Medicaments a base d'amides, nouveaux amides et leur preparation |
| US6103903A (en) | 1998-02-26 | 2000-08-15 | Neurogen Corporation | 4-(4-piperidylmethyhlamino) substituted heteroaryl fused pyridines: GABA brain receptor ligands |
| GB9917408D0 (en) * | 1999-07-23 | 1999-09-22 | Smithkline Beecham Plc | Compounds |
| GB9917406D0 (en) | 1999-07-23 | 1999-09-22 | Smithkline Beecham Plc | Compounds |
| US6376514B1 (en) * | 2000-10-17 | 2002-04-23 | The Procter & Gamble Co. | Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof |
| US6693099B2 (en) * | 2000-10-17 | 2004-02-17 | The Procter & Gamble Company | Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance |
| AR037641A1 (es) * | 2001-12-05 | 2004-11-17 | Tularik Inc | Moduladores de inflamacion |
| AR038240A1 (es) | 2002-01-29 | 2005-01-05 | Glaxo Group Ltd | Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para su preparacion |
| US7348434B2 (en) | 2003-08-08 | 2008-03-25 | Antony Bigot | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them |
| FR2858619B1 (fr) * | 2003-08-08 | 2006-12-22 | Aventis Pharma Sa | Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent |
| KR20090130347A (ko) * | 2007-05-09 | 2009-12-22 | 화이자 인코포레이티드 | 치환된 헤테로사이클릭 유도체 및 조성물 및 항균제로서의 이의 약학적 용도 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR31753E (fr) * | 1925-12-03 | 1927-06-11 | Appareil photographique pour prise de vues, agrandissement et projection | |
| FR42781E (fr) * | 1932-05-23 | 1933-10-10 | Perfectionnements aux machines rotatives à capsuler les bouteilles | |
| FR959917A (da) * | 1946-06-25 | 1950-04-07 | ||
| FR2177511A1 (en) * | 1972-03-28 | 1973-11-09 | Omnium Chimique Sa | Quinolyl pipiridylethyl ketones - with vasodilatory and antispasmodic activity |
| PT66682B (pt) * | 1976-06-18 | 1978-11-15 | Ind Biolog Francaise | /(quinolyl-4)-propyl-1/-4 piperidines leur preparation et leur utilisation comme medicaments /(quinolyl-4)-propyl/-4 piperidines leur preparation et leur utilisation comme medicaments |
| FR2354771A1 (fr) * | 1976-06-18 | 1978-01-13 | Mar Pha Etu Expl Marques | ((quinolyl-4)-3 propyl-1) -4 piperidines, leur preparation et leur utilisation comme medicaments |
| FR2485014A1 (fr) * | 1980-06-20 | 1981-12-24 | Pharmindustrie | Nouveaux derives de (quinolyl-2, -3 ou -4)-1 (piperidyl ou pyrrolidinyl-2 ou -3)-2 ou -3 ethanone ou propanone, procedes pour leur preparation, et leur utilisation comme medicaments |
-
1979
- 1979-12-21 FR FR7931396A patent/FR2471981A1/fr active Granted
-
1980
- 1980-12-02 US US06/212,293 patent/US4433150A/en not_active Expired - Lifetime
- 1980-12-12 EP EP80401788A patent/EP0031753B1/fr not_active Expired
- 1980-12-12 DE DE8080401788T patent/DE3069243D1/de not_active Expired
- 1980-12-12 DK DK530480A patent/DK530480A/da not_active Application Discontinuation
- 1980-12-15 AT AT0609680A patent/AT376670B/de not_active IP Right Cessation
- 1980-12-17 PT PT72212A patent/PT72212A/pt unknown
- 1980-12-19 IE IE2684/80A patent/IE51124B1/en unknown
- 1980-12-19 JP JP18031480A patent/JPS5699476A/ja active Pending
- 1980-12-19 CA CA000367172A patent/CA1178589A/fr not_active Expired
- 1980-12-19 NO NO803881A patent/NO155137C/no unknown
- 1980-12-19 ES ES498017A patent/ES498017A0/es active Granted
-
1981
- 1981-12-15 ES ES507997A patent/ES507997A0/es active Granted
- 1981-12-15 ES ES507998A patent/ES8207526A1/es not_active Expired
-
1982
- 1982-09-29 US US06/426,545 patent/US4505916A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AT376670B (de) | 1984-12-27 |
| IE51124B1 (en) | 1986-10-15 |
| IE802684L (en) | 1981-06-21 |
| EP0031753B1 (fr) | 1984-09-19 |
| US4505916A (en) | 1985-03-19 |
| JPS5699476A (en) | 1981-08-10 |
| EP0031753A1 (fr) | 1981-07-08 |
| NO155137C (no) | 1987-02-18 |
| FR2471981B1 (da) | 1983-03-25 |
| DE3069243D1 (en) | 1984-10-25 |
| ES8300745A1 (es) | 1982-11-01 |
| ES8207525A1 (es) | 1982-10-01 |
| NO155137B (no) | 1986-11-10 |
| ES507998A0 (es) | 1982-10-01 |
| US4433150A (en) | 1984-02-21 |
| ES8207526A1 (es) | 1982-10-01 |
| ES507997A0 (es) | 1982-10-01 |
| PT72212A (pt) | 1981-01-01 |
| ES498017A0 (es) | 1982-11-01 |
| FR2471981A1 (fr) | 1981-06-26 |
| CA1178589A (fr) | 1984-11-27 |
| ATA609680A (de) | 1984-05-15 |
| NO803881L (no) | 1981-06-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |