DK479984D0 - CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION - Google Patents
CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATIONInfo
- Publication number
- DK479984D0 DK479984D0 DK479984A DK479984A DK479984D0 DK 479984 D0 DK479984 D0 DK 479984D0 DK 479984 A DK479984 A DK 479984A DK 479984 A DK479984 A DK 479984A DK 479984 D0 DK479984 D0 DK 479984D0
- Authority
- DK
- Denmark
- Prior art keywords
- procedures
- preparation
- cephalosporine derivatives
- cephalosporine
- derivatives
- Prior art date
Links
- HOKIDJSKDBPKTQ-UHFFFAOYSA-N 3-(acetyloxymethyl)-7-[(5-amino-5-carboxypentanoyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical class S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)C(NC(=O)CCCC(N)C(O)=O)C12 HOKIDJSKDBPKTQ-UHFFFAOYSA-N 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3336757A DE3336757A1 (en) | 1983-10-08 | 1983-10-08 | CEPHALOSPORINE DERIVATIVES AND METHOD FOR THEIR PRODUCTION |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK479984D0 true DK479984D0 (en) | 1984-10-05 |
| DK479984A DK479984A (en) | 1985-04-09 |
Family
ID=6211418
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK479984A DK479984A (en) | 1983-10-08 | 1984-10-05 | CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP0137441A3 (en) |
| JP (1) | JPS6097982A (en) |
| DE (1) | DE3336757A1 (en) |
| DK (1) | DK479984A (en) |
| GR (1) | GR80573B (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8401093D0 (en) * | 1984-01-16 | 1984-02-15 | Fujisawa Pharmaceutical Co | Cephem compounds |
| NO165842C (en) * | 1984-04-23 | 1991-04-17 | Takeda Chemical Industries Ltd | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE CEFEM COMPOUNDS. |
| PH22107A (en) * | 1984-06-07 | 1988-06-01 | Takeda Chemical Industries Ltd | 3-pyrazolo(1,5-a)pyrdinium cephem compounds |
| JPH0613530B2 (en) * | 1984-06-08 | 1994-02-23 | 武田薬品工業株式会社 | Cem compound |
| US4665066A (en) * | 1984-12-24 | 1987-05-12 | Eli Lilly And Company | 3-thiazolomethyl cephalosporins as antibiotics |
| NO166283C (en) * | 1985-03-01 | 1991-06-26 | Takeda Chemical Industries Ltd | METHOD OF ANALOGUE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 7BETA- (2- (5-AMINO-1,2,4-THIADIAZOL-3-YL) -2 (Z) -SUBSTITUTE TOXYIMINOACETAMIDO) -3- (HETEROCYCLYLMETHYL) -CYLMETHYL-Methyl-3 . |
| GB8519606D0 (en) * | 1985-08-05 | 1985-09-11 | Fujisawa Pharmaceutical Co | 3 7-d substituted-3-cephem compounds |
| JPH07107069B2 (en) * | 1985-09-03 | 1995-11-15 | 大塚化学株式会社 | Novel derivative of cefalosporin compound, process for producing the same and pharmaceutical composition containing the derivative |
| DE3687200T2 (en) * | 1985-09-03 | 1993-05-27 | Otsuka Kagaku Kk | CEPHALOSPORINE DERIVATIVES. |
| US4826834A (en) * | 1985-09-27 | 1989-05-02 | Takeda Chemical Industries, Ltd. | Cephem compounds |
| CN86107947A (en) | 1985-11-22 | 1987-05-27 | 藤沢药品工业株式会社 | New cephem compounds and preparation method thereof |
| US4921851A (en) * | 1986-06-09 | 1990-05-01 | Takeda Chemical Industries, Ltd. | Cephem compounds, their production and use |
| JP2519054B2 (en) * | 1986-06-09 | 1996-07-31 | 武田薬品工業株式会社 | New cephem compound |
| DE3707019A1 (en) * | 1987-03-05 | 1988-09-15 | Hoechst Ag | CEPHALOSPORINE DERIVATIVES AND METHOD FOR THEIR PRODUCTION |
| US5173485A (en) * | 1988-03-09 | 1992-12-22 | Fujisawa Pharmaceutical Company, Ltd. | Cephem compounds |
| GB8805642D0 (en) * | 1988-03-09 | 1988-04-07 | Fujisawa Pharmaceutical Co | New cephem compounds & processes for preparation thereof |
| US5215982A (en) * | 1989-11-10 | 1993-06-01 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds |
| US5194433A (en) * | 1990-11-13 | 1993-03-16 | Bristol-Myers Squibb Company | Antibiotic c-3 catechol-substituted cephalosporin compounds, compositions and method of use thereof |
| KR0157073B1 (en) * | 1992-10-01 | 1998-11-16 | 김태훈 | Cephalosporin derivatives |
| TW526202B (en) | 1998-11-27 | 2003-04-01 | Shionogi & Amp Co | Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IE49100B1 (en) * | 1978-10-27 | 1985-07-24 | Glaxo Group Ltd | Cephalosporin compounds |
| ES485937A1 (en) * | 1978-11-15 | 1980-07-01 | Glaxo Group Ltd | Cephalosporin antibiotics |
| AU536966B2 (en) * | 1979-02-23 | 1984-05-31 | Glaxo Group Limited | Cephalosporin antibiotics |
| US4401668A (en) * | 1981-10-02 | 1983-08-30 | Eli Lilly And Company | Pyrazinium substituted cephalosporins |
-
1983
- 1983-10-08 DE DE3336757A patent/DE3336757A1/en not_active Withdrawn
-
1984
- 1984-10-02 EP EP84111745A patent/EP0137441A3/en not_active Withdrawn
- 1984-10-05 GR GR80573A patent/GR80573B/en unknown
- 1984-10-05 DK DK479984A patent/DK479984A/en not_active Application Discontinuation
- 1984-10-08 JP JP59211207A patent/JPS6097982A/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| GR80573B (en) | 1985-02-01 |
| EP0137441A2 (en) | 1985-04-17 |
| DK479984A (en) | 1985-04-09 |
| DE3336757A1 (en) | 1985-04-25 |
| JPS6097982A (en) | 1985-05-31 |
| EP0137441A3 (en) | 1986-01-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ATS | Application withdrawn |