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DK476985D0 - Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden - Google Patents

Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden

Info

Publication number
DK476985D0
DK476985D0 DK476985A DK476985A DK476985D0 DK 476985 D0 DK476985 D0 DK 476985D0 DK 476985 A DK476985 A DK 476985A DK 476985 A DK476985 A DK 476985A DK 476985 D0 DK476985 D0 DK 476985D0
Authority
DK
Denmark
Prior art keywords
procedure
imidazobenzodiazepines
intermediates
preparation
oxadiazolyl derivatives
Prior art date
Application number
DK476985A
Other languages
English (en)
Inventor
Frank Waetjen
Mogens Engelstoft
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan As filed Critical Ferrosan As
Priority to DK476985A priority Critical patent/DK476985D0/da
Publication of DK476985D0 publication Critical patent/DK476985D0/da
Priority to US06/816,732 priority patent/US4622320A/en
Priority to US06/816,731 priority patent/US4622321A/en
Priority to AU54013/86A priority patent/AU587802B2/en
Priority to DE198686102535T priority patent/DE197282T1/de
Priority to EP86102535A priority patent/EP0197282A1/en
Priority to DK094686A priority patent/DK157319C/da
Priority to PT82115A priority patent/PT82115B/pt
Priority to FI860894A priority patent/FI860894A7/fi
Priority to FI893143A priority patent/FI893143A7/fi
Priority to CA000503329A priority patent/CA1261322A/en
Priority to US06/837,100 priority patent/US4670433A/en
Priority to DE8686102951T priority patent/DE3660331D1/de
Priority to EP86102951A priority patent/EP0201678B1/en
Priority to AT86102951T priority patent/ATE35266T1/de
Priority to DE198686102951T priority patent/DE201678T1/de
Priority to NZ227855A priority patent/NZ227855A/xx
Priority to NO860857A priority patent/NO165545C/no
Priority to GR860639A priority patent/GR860639B/el
Priority to DE8686104605T priority patent/DE3661197D1/de
Priority to EP86104605A priority patent/EP0202441B1/en
Priority to AT86104605T priority patent/ATE38671T1/de
Priority to DE198686104605T priority patent/DE202441T1/de
Priority to US06/856,945 priority patent/US4745112A/en
Priority to CA000507955A priority patent/CA1256863A/en
Priority to CA000507957A priority patent/CA1256865A/en
Priority to CA000507956A priority patent/CA1256864A/en
Priority to GR861260A priority patent/GR861260B/el
Priority to AU57429/86A priority patent/AU590273B2/en
Priority to GR861261A priority patent/GR861261B/el
Priority to IL78791A priority patent/IL78791A/xx
Priority to IL78790A priority patent/IL78790A/xx
Priority to DK231686A priority patent/DK157194C/da
Priority to NZ227983A priority patent/NZ227983A/en
Priority to FI862062A priority patent/FI83325C/fi
Priority to IE130786A priority patent/IE59495B1/en
Priority to NZ216202A priority patent/NZ216202A/xx
Priority to ES555036A priority patent/ES8707206A1/es
Priority to DK231586A priority patent/DK154837C/da
Priority to PT82594A priority patent/PT82594B/pt
Priority to FI862061A priority patent/FI82049C/fi
Priority to PT82593A priority patent/PT82593B/pt
Priority to IE130686A priority patent/IE59494B1/en
Priority to NZ216203A priority patent/NZ216203A/xx
Priority to FI892920A priority patent/FI892920A0/fi
Priority to ES555035A priority patent/ES8707205A1/es
Priority to NO86861953A priority patent/NO162859C/no
Priority to NO861954A priority patent/NO163228C/no
Priority to IL90183A priority patent/IL90183A/xx
Priority to US06/912,775 priority patent/US4771051A/en
Priority to AT86307541T priority patent/ATE44381T1/de
Priority to DE8787114729T priority patent/DE3686723T2/de
Priority to DE8686307541T priority patent/DE3664211D1/de
Priority to EP87114729A priority patent/EP0274009B1/en
Priority to EP86307541A priority patent/EP0226282B1/en
Priority to CA000519558A priority patent/CA1297099C/en
Priority to ES86307541T priority patent/ES2011448B3/es
Priority to AT87114729T priority patent/ATE80392T1/de
Priority to NO864063A priority patent/NO165840C/no
Priority to FI864126A priority patent/FI83871C/fi
Priority to IL80320A priority patent/IL80320A/xx
Priority to IE273486A priority patent/IE59830B1/en
Priority to PH34376A priority patent/PH24902A/en
Priority to NZ217959A priority patent/NZ217959A/xx
Priority to IE930093A priority patent/IE63631B1/en
Priority to DK499586A priority patent/DK155007C/da
Priority to AU64180/86A priority patent/AU586043B2/en
Priority to KR1019860008729A priority patent/KR940010035B1/ko
Priority to JP61247308A priority patent/JPH0751577B2/ja
Priority to PT83573A priority patent/PT83573B/pt
Priority to US06/942,200 priority patent/US4727153A/en
Priority to US06/942,162 priority patent/US4772696A/en
Priority to US07/143,364 priority patent/US4780539A/en
Priority to DK063388A priority patent/DK159150C/da
Priority to DK063288A priority patent/DK160097C/da
Priority to PH36839A priority patent/PH25034A/en
Priority to CA000590382A priority patent/CA1266671A/en
Priority to NO890989A priority patent/NO890989D0/no
Priority to JP1065783A priority patent/JPH01279877A/ja
Priority to IL90183A priority patent/IL90183A0/xx
Priority to NO892008A priority patent/NO169228C/no
Priority to AU39333/89A priority patent/AU614407B2/en
Priority to GR89400192T priority patent/GR3000177T3/el
Priority to IL93355A priority patent/IL93355A0/xx
Priority to GR920402804T priority patent/GR3006440T3/el
Priority to JP5260097A priority patent/JPH072727B2/ja

Links

DK476985A 1985-03-08 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden DK476985D0 (da)

Priority Applications (86)

Application Number Priority Date Filing Date Title
DK476985A DK476985D0 (da) 1985-10-17 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden
US06/816,732 US4622320A (en) 1985-05-17 1986-01-06 Oxadiazolylimidazobenzodiazepine, compositions, and method
US06/816,731 US4622321A (en) 1985-05-17 1986-01-06 Oxadiazolylimidazobenzodiazepine, compositions, and method
AU54013/86A AU587802B2 (en) 1985-03-08 1986-02-24 Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
DE198686102535T DE197282T1 (de) 1985-03-08 1986-02-27 Oxadiazolyl-imidazobenzodiazepinderivate und methoden zu ihrer herstellung.
EP86102535A EP0197282A1 (en) 1985-03-08 1986-02-27 Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
DK094686A DK157319C (da) 1985-03-08 1986-02-28 Oxadiazolylimidazobenzodiazepinderivater
PT82115A PT82115B (pt) 1985-03-08 1986-02-28 Processo de preparacao de derivados de oxadiazolilimidazobenzodiazepina e dos seus intermediarios
FI860894A FI860894A7 (fi) 1985-03-08 1986-03-03 Nya oxadiazolyl -imidazobensodiazepinderivat och foerfarande foer framstaellning av dylika foereningar.
FI893143A FI893143A7 (fi) 1985-03-08 1986-03-03 Isosyanometyyliyhdiste ja menetelmä oksadiatsolyyli-imidatsobentsodiatsepiinijohdannaisten valmistamiseksi
CA000503329A CA1261322A (en) 1985-03-08 1986-03-05 Oxadiazolyl imidabenzodiazepine derivatives, a method of preparing the same, pharmaceutical compositions thereof, and method of treating therewith
US06/837,100 US4670433A (en) 1985-03-08 1986-03-06 Oxadiazolyl imidazobenzodiazepine derivatives pharmaceutical compositions thereof, and method of treating therewith
DE8686102951T DE3660331D1 (en) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
EP86102951A EP0201678B1 (en) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
AT86102951T ATE35266T1 (de) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6dihydro-5-methyl-6-oxo-4h-imidazo(1,5a)(1,4)benzodiazepin, verfahren zu seiner herstellung und pharmazeutische zubereitungen.
DE198686102951T DE201678T1 (de) 1985-05-17 1986-03-06 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin, verfahren zu seiner herstellung und pharmazeutische zubereitungen.
NZ227855A NZ227855A (en) 1985-03-08 1986-03-07 Isocyanomethyl derivatives of oxadiazoles
NO860857A NO165545C (no) 1985-03-08 1986-03-07 Analogifremgangsmaate for fremstilling av terapeutisk aktive nye oksadiazolimidazo-benzodiazepinderivater.
GR860639A GR860639B (en) 1985-03-08 1986-03-07 Novel oxadiazolyl imidazobenzodiazepine derivates and methods of preaparing such compounds
DE8686104605T DE3661197D1 (en) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
EP86104605A EP0202441B1 (en) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
AT86104605T ATE38671T1 (de) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepine, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
DE198686104605T DE202441T1 (de) 1985-05-17 1986-04-04 Oxadiazolylimidazobenzodiazepine, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
US06/856,945 US4745112A (en) 1985-05-17 1986-04-28 Oxadiazolylimidazobenzodiazepine, compositions, and method III
CA000507955A CA1256863A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method i
CA000507957A CA1256865A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method iii
CA000507956A CA1256864A (en) 1985-05-17 1986-04-30 Oxadiazolylimidazobenzodiazepine, compositions, and method ii
GR861260A GR861260B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound pharmaceutial composition containing said compound method of preparing said compound and method of treating a central nervous system ailment
AU57429/86A AU590273B2 (en) 1985-05-17 1986-05-14 Oxydiazolyl imidazobenzodiazepine compound, pharmaceutical composition containing said compound, method of preparing said compound and method of treating a central nervous system ailment
GR861261A GR861261B (en) 1985-05-17 1986-05-14 Oxadiazolyl imidazobenzodiazepine compound pharmaceutical composition containing said compound method of preparing said compound and method of treating a central nervous system ailment
IL78791A IL78791A (en) 1985-05-17 1986-05-15 7-substituted-3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)-(1,4)-benzodiazepines,pharmaceutical compositions containing them and method of preparing them
IL78790A IL78790A (en) 1985-05-17 1986-05-15 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl 6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepine,a pharmaceutical composition containing it and a method of preparing it
DK231686A DK157194C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme
NZ227983A NZ227983A (en) 1985-05-17 1986-05-16 5 cyclopropyl-3-isocyanomethyl-1,2,4-oxidiazole
FI862062A FI83325C (fi) 1985-05-17 1986-05-16 Foerfarande foer framstaellning av 7- substituerade 3-(5-cyklopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-metyl -6-oxo-4h-imidazo(1,5-a)(1,4) bensodiazepiner.
IE130786A IE59495B1 (en) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepines, process for their preparation and pharmaceutical compositions
NZ216202A NZ216202A (en) 1985-05-17 1986-05-16 An oxadiazolyl imidazobenzodiazepine compound and pharmaceutical compositions thereof
ES555036A ES8707206A1 (es) 1985-05-17 1986-05-16 Procedimiento para preparar derivados de oxadiazolilimidazobenzodiazepina
DK231586A DK154837C (da) 1985-05-17 1986-05-16 Oxadiazolylimidazobenzodiazepinforbindelse og farmaceutisk praeparat indeholdende samme
PT82594A PT82594B (pt) 1985-05-17 1986-05-16 Processo de preparacao da oxadiazolil-imidazobenzodiazepina e das composicoes farmaceuticas que a contem
FI862061A FI82049C (fi) 1985-05-17 1986-05-16 Foerfarande foer framstaellning av saosom laekemedel anvaendbar 3-(5-cyklopropyl-1,2,4-oxadiazol-3-yl) 5,6-dihydro-5-metyl-6-oxo-4h-imidazo-(1,5-a)(1,4)bensodiazepin.
PT82593A PT82593B (pt) 1985-05-17 1986-05-16 Processo de preparacao da oxadiazolil-imidazobenzodiazepina e das composicoes farmaceuticas que a contem
IE130686A IE59494B1 (en) 1985-05-17 1986-05-16 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5--methyl-6-oxo-4h-imidazo(1,4-a)(1,4)benzodiazepine, a process for its preparation and pharmaceutical compositions
NZ216203A NZ216203A (en) 1985-05-17 1986-05-16 Oxydiazolyl imidazobenzodiazepines and pharmaceutical compositions
FI892920A FI892920A0 (fi) 1985-05-17 1986-05-16 Substituerad 1,2,4-oxadiazol.
ES555035A ES8707205A1 (es) 1985-05-17 1986-05-16 Procedimiento para preparar un derivado de oxadiazolilimidazobenzodiazepina
NO86861953A NO162859C (no) 1985-05-17 1986-05-16 Analogifremgangsmaate for fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelser.
NO861954A NO163228C (no) 1985-05-17 1986-05-16 Analogifremgangsmaate til fremstilling av terapeutisk aktive oksadiazolylimidazobenzodiazepinforbindelse.
IL90183A IL90183A (en) 1985-05-17 1986-05-18 5-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazole
US06/912,775 US4771051A (en) 1985-05-17 1986-09-26 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
AT86307541T ATE44381T1 (de) 1985-10-17 1986-10-01 Heterocyclische verbindungen und ihre herstellung und verwendung.
DE8787114729T DE3686723T2 (de) 1985-10-17 1986-10-01 Oxadiazolylacetonitrile, ihre herstellung und anwendung.
DE8686307541T DE3664211D1 (en) 1985-10-17 1986-10-01 Heterocyclic compounds and their preparation and use
EP87114729A EP0274009B1 (en) 1985-10-17 1986-10-01 Oxadiazolylacetonitriles, their preparation and use
EP86307541A EP0226282B1 (en) 1985-10-17 1986-10-01 Heterocyclic compounds and their preparation and use
CA000519558A CA1297099C (en) 1985-10-17 1986-10-01 Quinazoline compounds and their preparation and use
ES86307541T ES2011448B3 (es) 1985-10-17 1986-10-01 Preparacion de un compuesto heterocido y uso del mismo
AT87114729T ATE80392T1 (de) 1985-10-17 1986-10-01 Oxadiazolylacetonitrile, ihre herstellung und anwendung.
NO864063A NO165840C (no) 1985-10-17 1986-10-13 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazo-quinazolinforbindelser.
FI864126A FI83871C (fi) 1985-10-17 1986-10-13 Foerfarande foer framstaellning av saosom psykofarmaceutiska medel anvaendbara 4,5-dihydro-5-oxo-imidazo (1,5-a)kinazolinderivat.
IL80320A IL80320A (en) 1985-10-17 1986-10-15 3-substituted-4,5-dihydro-5-oxo-imidazo(1,5-a)quinazoline derivatives,their preparation and pharmaceutical compositions containing them
IE273486A IE59830B1 (en) 1985-10-17 1986-10-16 Heterocyclic compounds and their preparation and use
PH34376A PH24902A (en) 1985-10-17 1986-10-16 Quinazoline compounds,a pharmaceutical preparation containing said compounds and a method of treating a central nervous system ailment in a human
NZ217959A NZ217959A (en) 1985-10-17 1986-10-16 Imidazoquinazoline derivatives and pharmaceutical compositions
IE930093A IE63631B1 (en) 1985-10-17 1986-10-16 Oxadiazolylacetonitriles their preparation and use
DK499586A DK155007C (da) 1985-10-17 1986-10-17 Imidazo(1,5-a)quinazolinforbindelse, praeparat indeholdende samme samt isocyanomethyl-oxadiazol til brug som udgangsmateriale ved fremstillingen af forbindelsen
AU64180/86A AU586043B2 (en) 1985-10-17 1986-10-17 Imidazo``1,5-a``quinazoline derivatives, their preparation and use.
KR1019860008729A KR940010035B1 (ko) 1985-10-17 1986-10-17 헤테로사이클릭 퀴나졸린 화합물의 제조방법
JP61247308A JPH0751577B2 (ja) 1985-10-17 1986-10-17 複素環キナゾリン化合物、その製造方法、並びに用途
PT83573A PT83573B (pt) 1985-10-17 1986-10-17 Processo de preparacao de compostos heterociclicos de quinazolina e de seus intermediarios e de composicoes farmaceuticas
US06/942,200 US4727153A (en) 1985-03-08 1986-12-16 Oxadiazolyl intermediates
US06/942,162 US4772696A (en) 1985-03-08 1986-12-16 Oxadiazolyl imidazobenzodiazepine process
US07/143,364 US4780539A (en) 1985-05-17 1988-01-12 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
DK063388A DK159150C (da) 1985-03-08 1988-02-08 Isocyanomethylforbindelse samt fremgangsmaade til fremstilling af et oxadiazolimidazobenzodiazepinderivat
DK063288A DK160097C (da) 1985-05-17 1988-02-08 Fremgangsmaade til fremstilling af 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4h-imidazo(1,5-a)(1,4)benzodiazepin samt 3-cyclopropyl-3-isocyanomethyl-1,2,4-oxadiazol til anvendelse som udgangsmateriale ved fremgangsmaaden
PH36839A PH25034A (en) 1985-10-17 1988-04-25 Process for the preparation of imidazoquinazoline compounds and intermediate for use in said process
CA000590382A CA1266671A (en) 1985-03-08 1989-02-07 Oxadiazolyl imidazobenzodiazepine derivatives, a method of preparing the same, pharmaceutical compositions thereof, and method of treating therewith
NO890989A NO890989D0 (no) 1985-03-08 1989-03-08 Isocyanometylforbindelse samt fremgangsmaate for fremstilling av et oksadiazolimidazobenzodiazepinderivat.
JP1065783A JPH01279877A (ja) 1985-05-17 1989-03-17 5―シクロプロピル―3―イソシアノメチル―1,2,4―オキサジアゾール
IL90183A IL90183A0 (en) 1985-05-17 1989-05-04 Substituted 1,2,4-oxadiazole
NO892008A NO169228C (no) 1985-05-17 1989-05-19 5-cyklopropyl-3-isocyanometyl-1,2,4-oksadiazol
AU39333/89A AU614407B2 (en) 1985-05-17 1989-08-04 Oxadiazolyl imidazobenzodiazepine compound, pharmaceutical composition containing said compound, method of preparing said compound and method of treating a central nervous system ailment
GR89400192T GR3000177T3 (en) 1985-10-17 1989-10-06 Heterocyclic compounds and their preparation and use
IL93355A IL93355A0 (en) 1985-03-08 1990-02-12 Isocyanomethyl derivatives
GR920402804T GR3006440T3 (da) 1985-10-17 1992-12-02
JP5260097A JPH072727B2 (ja) 1985-10-17 1993-10-18 キナゾリン化合物の製造に有用なオキサジアゾール誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK476985A DK476985D0 (da) 1985-10-17 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden

Publications (1)

Publication Number Publication Date
DK476985D0 true DK476985D0 (da) 1985-10-17

Family

ID=8136496

Family Applications (1)

Application Number Title Priority Date Filing Date
DK476985A DK476985D0 (da) 1985-03-08 1985-10-17 Fremgangsmaade til fremstilling af oxadiazolylderivater af imidazobenzodiazepiner og mellemprodukt til brug ved fremgangsmaaden

Country Status (1)

Country Link
DK (1) DK476985D0 (da)

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