DK476885D0 - Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf - Google Patents
Heterocycliske forbindelser og fremgangsmaader til fremstilling herafInfo
- Publication number
- DK476885D0 DK476885D0 DK476885A DK476885A DK476885D0 DK 476885 D0 DK476885 D0 DK 476885D0 DK 476885 A DK476885 A DK 476885A DK 476885 A DK476885 A DK 476885A DK 476885 D0 DK476885 D0 DK 476885D0
- Authority
- DK
- Denmark
- Prior art keywords
- sub
- relations
- heterocyclic
- procedures
- preparing
- Prior art date
Links
- 238000000034 method Methods 0.000 title 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 230000000895 acaricidal effect Effects 0.000 abstract 1
- 239000000642 acaricide Substances 0.000 abstract 1
- 230000000507 anthelmentic effect Effects 0.000 abstract 1
- 239000000921 anthelmintic agent Substances 0.000 abstract 1
- 229940124339 anthelmintic agent Drugs 0.000 abstract 1
- 229940125681 anticonvulsant agent Drugs 0.000 abstract 1
- 239000001961 anticonvulsive agent Substances 0.000 abstract 1
- 239000002249 anxiolytic agent Substances 0.000 abstract 1
- 230000000949 anxiolytic effect Effects 0.000 abstract 1
- 229940005530 anxiolytics Drugs 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 239000003326 hypnotic agent Substances 0.000 abstract 1
- 230000000147 hypnotic effect Effects 0.000 abstract 1
- 239000002917 insecticide Substances 0.000 abstract 1
- 239000002664 nootropic agent Substances 0.000 abstract 1
- 230000001777 nootropic effect Effects 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Tropical Medicine & Parasitology (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cosmetics (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Lubricants (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Priority Applications (60)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK476885A DK476885D0 (da) | 1985-10-17 | 1985-10-17 | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
| US06/912,777 US4870073A (en) | 1985-10-17 | 1986-09-26 | Heterocyclic compounds and their preparation and use |
| US06/912,776 US4774245A (en) | 1985-10-17 | 1986-09-26 | Imidazoquinoxaline compounds |
| US06/912,775 US4771051A (en) | 1985-05-17 | 1986-09-26 | 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments |
| EP87114729A EP0274009B1 (en) | 1985-10-17 | 1986-10-01 | Oxadiazolylacetonitriles, their preparation and use |
| ES86307541T ES2011448B3 (es) | 1985-10-17 | 1986-10-01 | Preparacion de un compuesto heterocido y uso del mismo |
| AT86307542T ATE48844T1 (de) | 1985-10-17 | 1986-10-01 | Heterocyclische verbindungen, ihre herstellung und verwendung. |
| DE8787114729T DE3686723T2 (de) | 1985-10-17 | 1986-10-01 | Oxadiazolylacetonitrile, ihre herstellung und anwendung. |
| CA000519558A CA1297099C (en) | 1985-10-17 | 1986-10-01 | Quinazoline compounds and their preparation and use |
| DE8686307541T DE3664211D1 (en) | 1985-10-17 | 1986-10-01 | Heterocyclic compounds and their preparation and use |
| CA000519557A CA1275411C (en) | 1985-10-17 | 1986-10-01 | Heterocyclic compounds and their preparation and use |
| EP86307542A EP0225013B1 (en) | 1985-10-17 | 1986-10-01 | Heterocyclic compounds and their preparation and use |
| EP86307541A EP0226282B1 (en) | 1985-10-17 | 1986-10-01 | Heterocyclic compounds and their preparation and use |
| DE8686307542T DE3667665D1 (de) | 1985-10-17 | 1986-10-01 | Heterocyclische verbindungen, ihre herstellung und verwendung. |
| CA000519556A CA1293723C (en) | 1985-10-17 | 1986-10-01 | 1,2,4-oxadiazolyl derivatives of imidazo-: benzazepine, benzodiazepine, benzoxazepine and benzothiazepine |
| EP86307543A EP0220845A1 (en) | 1985-10-17 | 1986-10-01 | Heterocyclic compounds and their preparation and use |
| AT86307541T ATE44381T1 (de) | 1985-10-17 | 1986-10-01 | Heterocyclische verbindungen und ihre herstellung und verwendung. |
| ES86307542T ES2014234B3 (es) | 1985-10-17 | 1986-10-01 | Compuestos heterociclicos, su preparacion y usos |
| AT87114729T ATE80392T1 (de) | 1985-10-17 | 1986-10-01 | Oxadiazolylacetonitrile, ihre herstellung und anwendung. |
| NO864063A NO165840C (no) | 1985-10-17 | 1986-10-13 | Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazo-quinazolinforbindelser. |
| NO864062A NO163776C (no) | 1985-10-17 | 1986-10-13 | Analogifremgangsmaate til fremstilling av terapeutisk aktive imidazoquinoksaliner. |
| FI864124A FI864124A7 (fi) | 1985-10-17 | 1986-10-13 | Heterocykliska foereningar och deras framstaellning samt anvaendning. |
| FI864126A FI83871C (fi) | 1985-10-17 | 1986-10-13 | Foerfarande foer framstaellning av saosom psykofarmaceutiska medel anvaendbara 4,5-dihydro-5-oxo-imidazo (1,5-a)kinazolinderivat. |
| NO864061A NO864061L (no) | 1985-10-17 | 1986-10-13 | Hetrocykliske forbindelser og fremstilling og anvendelse av disse. |
| FI864125A FI82050C (fi) | 1985-10-17 | 1986-10-13 | Foerfarande foer framstaellning som laekemedel anvaendbara 3-oxadiazolylderivat av imidazol(1,5-a) kinoxaliner och 1-oxdiazolylderivat av imidazo(1,5-a)pyrrolo(2,1-c) kinoxaliner. |
| IL80319A IL80319A (en) | 1985-10-17 | 1986-10-15 | 4,5-dihydro-3-(substituted 1,2,4-oxadiazolyl)-imidazo-(1,5-a)pyrrolo(2,1-c)-quinoxaline derivatives,their preparation and pharmaceutical compositions containing them |
| IL80318A IL80318A0 (en) | 1985-10-17 | 1986-10-15 | Bridged 1-phenylimidazole derivatives,their preparation and pharmaceutical compositions containing them |
| IL80320A IL80320A (en) | 1985-10-17 | 1986-10-15 | 3-substituted-4,5-dihydro-5-oxo-imidazo(1,5-a)quinazoline derivatives,their preparation and pharmaceutical compositions containing them |
| PH34375A PH22556A (en) | 1985-10-17 | 1986-10-16 | Heterocyclic compounds, pharmaceutical compositions containing the same and method of use thereof |
| IE273386A IE59642B1 (en) | 1985-10-17 | 1986-10-16 | Heterocyclic compounds and their preparation and use |
| NZ217957A NZ217957A (en) | 1985-10-17 | 1986-10-16 | 3-oxadiazole-imidazo quinoxalines, their preparation, and pharmaceutical compositions |
| IE273486A IE59830B1 (en) | 1985-10-17 | 1986-10-16 | Heterocyclic compounds and their preparation and use |
| NZ217958A NZ217958A (en) | 1985-10-17 | 1986-10-16 | Derivatives of imidazo benzazepine and pharmaceutical compositions |
| PH34376A PH24902A (en) | 1985-10-17 | 1986-10-16 | Quinazoline compounds,a pharmaceutical preparation containing said compounds and a method of treating a central nervous system ailment in a human |
| IE930093A IE63631B1 (en) | 1985-10-17 | 1986-10-16 | Oxadiazolylacetonitriles their preparation and use |
| NZ217959A NZ217959A (en) | 1985-10-17 | 1986-10-16 | Imidazoquinazoline derivatives and pharmaceutical compositions |
| AU64180/86A AU586043B2 (en) | 1985-10-17 | 1986-10-17 | Imidazo``1,5-a``quinazoline derivatives, their preparation and use. |
| KR1019860008728A KR940010034B1 (ko) | 1985-10-17 | 1986-10-17 | 헤테로사이클릭 퀴녹살린 화합물의 제조방법 |
| AU64179/86A AU591937B2 (en) | 1985-10-17 | 1986-10-17 | Imidazo(15-a)quinoxaline derivatives and their preparation and use |
| DK499586A DK155007C (da) | 1985-10-17 | 1986-10-17 | Imidazo(1,5-a)quinazolinforbindelse, praeparat indeholdende samme samt isocyanomethyl-oxadiazol til brug som udgangsmateriale ved fremstillingen af forbindelsen |
| JP61247307A JPH0753731B2 (ja) | 1985-10-17 | 1986-10-17 | 複素環式キノキサリン化合物、その製造方法並びその用途 |
| PT83571A PT83571B (en) | 1985-10-17 | 1986-10-17 | Process for the preparation of heterocyclic compounds of 1-phenyl-imidazoles and of pharmaceutical compounds containing them |
| DK499486A DK155006C (da) | 1985-10-17 | 1986-10-17 | Kondenserede imidazolderivater og farmaceutisk praeparat indeholdende en saadan forbindelse |
| PT83572A PT83572B (pt) | 1985-10-17 | 1986-10-17 | Processo para a preparacao de compostos heterociclicos de quinoxalina e de composicoes farmaceuticas que os contem |
| KR1019860008729A KR940010035B1 (ko) | 1985-10-17 | 1986-10-17 | 헤테로사이클릭 퀴나졸린 화합물의 제조방법 |
| DK499686A DK154142C (da) | 1985-10-17 | 1986-10-17 | Imidazo(1,5-a)quinoxalinforbindelse samt praeparat indeholdende samme |
| JP61247308A JPH0751577B2 (ja) | 1985-10-17 | 1986-10-17 | 複素環キナゾリン化合物、その製造方法、並びに用途 |
| JP61247306A JPS62155278A (ja) | 1985-10-17 | 1986-10-17 | 複素環式化合物、その製法および使用 |
| AU64178/86A AU6417886A (en) | 1985-10-17 | 1986-10-17 | Heterocyclic compounds and and their preparation and use |
| PT83573A PT83573B (pt) | 1985-10-17 | 1986-10-17 | Processo de preparacao de compostos heterociclicos de quinazolina e de seus intermediarios e de composicoes farmaceuticas |
| ZA871535A ZA871535B (en) | 1985-10-17 | 1987-03-03 | Heterocyclic compounds and their preparation and use |
| US07/108,272 US4795749A (en) | 1985-10-17 | 1987-10-13 | Imidazopyrroloquinoxaline compounds |
| US07/143,364 US4780539A (en) | 1985-05-17 | 1988-01-12 | 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments |
| PH36839A PH25034A (en) | 1985-10-17 | 1988-04-25 | Process for the preparation of imidazoquinazoline compounds and intermediate for use in said process |
| US07/305,969 US4886797A (en) | 1985-10-17 | 1989-02-02 | Heterocyclic compounds and their preparation and use |
| US07/305,970 US4880799A (en) | 1985-10-17 | 1989-02-02 | Heterocyclic compounds and their preparation and use |
| GR89400192T GR3000177T3 (en) | 1985-10-17 | 1989-10-06 | Heterocyclic compounds and their preparation and use |
| GR90400114T GR3000367T3 (en) | 1985-10-17 | 1990-03-01 | Heterocyclic compounds and their preparation and use |
| GR920402804T GR3006440T3 (da) | 1985-10-17 | 1992-12-02 | |
| JP5260097A JPH072727B2 (ja) | 1985-10-17 | 1993-10-18 | キナゾリン化合物の製造に有用なオキサジアゾール誘導体 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK476885A DK476885D0 (da) | 1985-10-17 | 1985-10-17 | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK476885D0 true DK476885D0 (da) | 1985-10-17 |
Family
ID=8136485
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK476885A DK476885D0 (da) | 1985-05-17 | 1985-10-17 | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
Country Status (18)
| Country | Link |
|---|---|
| US (5) | US4870073A (da) |
| EP (2) | EP0220845A1 (da) |
| JP (2) | JPS62155278A (da) |
| KR (1) | KR940010034B1 (da) |
| AT (1) | ATE48844T1 (da) |
| AU (2) | AU6417886A (da) |
| CA (2) | CA1293723C (da) |
| DE (1) | DE3667665D1 (da) |
| DK (1) | DK476885D0 (da) |
| ES (1) | ES2014234B3 (da) |
| FI (2) | FI864124A7 (da) |
| GR (1) | GR3000367T3 (da) |
| IE (1) | IE59642B1 (da) |
| IL (1) | IL80319A (da) |
| NO (2) | NO163776C (da) |
| NZ (2) | NZ217957A (da) |
| PH (1) | PH22556A (da) |
| PT (2) | PT83571B (da) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK476885D0 (da) * | 1985-10-17 | 1985-10-17 | Ferrosan As | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
| EP0226282B1 (en) * | 1985-10-17 | 1989-07-05 | A/S Ferrosan | Heterocyclic compounds and their preparation and use |
| DK174086D0 (da) * | 1986-04-16 | 1986-04-16 | Ferrosan As | Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme |
| DK155524C (da) * | 1987-03-18 | 1989-09-11 | Ferrosan As | Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse |
| DK160876C (da) * | 1987-12-08 | 1991-10-14 | Novo Nordisk As | Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar |
| IL90315A0 (en) * | 1988-06-01 | 1989-12-15 | Ferrosan As | Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them |
| DK161148C (da) * | 1988-06-14 | 1991-11-18 | Novo Nordisk As | Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne |
| GB8823475D0 (en) * | 1988-10-06 | 1988-11-16 | Merck Sharp & Dohme | Chemical compounds |
| DK626288D0 (da) * | 1988-11-10 | 1988-11-10 | Ferrosan As | Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen |
| DK0389189T3 (da) * | 1989-03-23 | 1994-06-20 | Pfizer | Diazepin antiallergimidler |
| DK443589D0 (da) * | 1989-09-08 | 1989-09-08 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| DK588489D0 (da) * | 1989-11-22 | 1989-11-22 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| DK588389D0 (da) * | 1989-11-22 | 1989-11-22 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| US5276028A (en) * | 1990-06-22 | 1994-01-04 | Nordisk A/S | Imidazoquinoxaline compounds |
| US5371080A (en) * | 1990-06-22 | 1994-12-06 | Novo Nordisk A/S | Imidazoquinazoline compounds and their use |
| DK151890D0 (da) * | 1990-06-22 | 1990-06-22 | Ferrosan As | Heterocykliske forbindelser deres fremstilling og brug |
| DK41191D0 (da) * | 1991-03-07 | 1991-03-07 | Novo Nordisk As | Heterocycliske forbindelser, deres fremstilling og anvendelse |
| EP0590022A1 (en) * | 1991-06-14 | 1994-04-06 | PHARMACIA & UPJOHN COMPANY | IMIDAZO 1,5-a]QUINOXALINES |
| US5561227A (en) * | 1991-07-23 | 1996-10-01 | Schering Corporation | Process for the stereospecific synthesis of azetidinones |
| EP0596015B1 (en) * | 1991-07-23 | 1997-10-01 | Schering Corporation | Substituted beta-lactam compounds useful as hypocholesterolemic agents and processes for the preparation thereof |
| WO1993012113A1 (en) * | 1991-12-17 | 1993-06-24 | The Upjohn Company | 3-SUBSTITUTED IMIDAZO (1,5-a) AND IMIDAZO (1,5-a)-TRIAZOLO (1,5-c) QUINOXALINES AND QUINAZOLINES WITH CNS ACTIVITY |
| US5244906A (en) * | 1992-01-23 | 1993-09-14 | Dowelanco | Insect control with substituted oxadiazole and thiadiazole compounds |
| DE69332019T2 (de) * | 1992-02-13 | 2002-11-28 | Pharmacia & Upjohn Co., Kalamazoo | 4-oxo-und 4h-imidazo(5,1-c)(1,4)benzoxazine nützlich als benzodiazepinrezeptor-bindemittel. |
| GB9212486D0 (en) * | 1992-06-12 | 1992-07-22 | Erba Carlo Spa | Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation |
| CA2143246C (en) * | 1994-03-16 | 2000-08-22 | Thierry Godel | Imidazodiazepines |
| GB2328940B (en) * | 1997-09-05 | 1999-12-08 | Dong Kook Pharm Co Ltd | A process for preparing benzodiazepine derivatives |
| CA2636043A1 (en) * | 2006-01-23 | 2007-08-02 | Amira Pharmaceuticals, Inc. | Tricyclic inhibitors of 5-lipoxygenase |
| US20090054412A1 (en) * | 2007-08-20 | 2009-02-26 | John Alan Kemp | Treatment of Sleep Disorders |
| CN101827597B (zh) | 2007-08-20 | 2013-03-13 | 伊沃泰克国际有限责任公司 | 睡眠障碍的治疗 |
| JO3156B1 (ar) | 2009-07-09 | 2017-09-20 | Novartis Ag | ايميدازولات مدمجة والتركيبات التي تشملها لعلاج الأمراض الطفيلية على مثال الملاريا |
| JP6964343B2 (ja) | 2015-11-20 | 2021-11-10 | フォーマ セラピューティクス,インコーポレイテッド | ユビキチン特異的プロテアーゼ1阻害剤としてのプリノン |
| JP7377717B2 (ja) | 2017-04-24 | 2023-11-10 | ノバルティス アーゲー | 2-アミノ-l-(2-(4-フルオロフェニル)-3-(4-フルオロフェニルアミノ)-8,8-ジメチル-5,6-ジヒドロイミダゾ[1,2-a]ピラジン-7(8h)-イル)エタノン及びそれらの組み合わせの治療レジメン |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4118386A (en) * | 1977-04-04 | 1978-10-03 | Hoffmann-La Roche Inc. | Synthesis of imidazo[1,5-a]diazepine-3-carboxylates |
| US4668678A (en) * | 1980-05-09 | 1987-05-26 | Usv Pharmaceutical Corporation | Triazoloquinoxalin-1,4-diones |
| CA1184175A (en) * | 1981-02-27 | 1985-03-19 | Walter Hunkeler | Imidazodiazepines |
| US4440929A (en) * | 1981-07-16 | 1984-04-03 | Usv Pharmaceutical Corporation | Imidazoquinoxaline compounds |
| DK151808C (da) * | 1982-11-16 | 1988-06-20 | Ferrosan As | Analogifremgangsmaade til fremstilling af oxadiazolylimidazo-oe1,4aa-benzodiazepinderivater |
| CA1252462A (en) * | 1984-01-19 | 1989-04-11 | Walter Hunkeler | Imidazodiazepine derivatives |
| US4771051A (en) * | 1985-05-17 | 1988-09-13 | A/S Ferrosan | 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments |
| DK476885D0 (da) * | 1985-10-17 | 1985-10-17 | Ferrosan As | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
| EP0226282B1 (en) * | 1985-10-17 | 1989-07-05 | A/S Ferrosan | Heterocyclic compounds and their preparation and use |
| FR2598147B1 (fr) * | 1986-04-30 | 1988-08-26 | Pasteur Institut | Immunogene isole de mollusques, son procede de preparation, reactifs de diagnostic des bilharzioses humaines, vaccins contre les schistosomiases et compositions immunisantes comprenant ledit immunogene. |
-
1985
- 1985-10-17 DK DK476885A patent/DK476885D0/da not_active Application Discontinuation
-
1986
- 1986-09-26 US US06/912,777 patent/US4870073A/en not_active Expired - Fee Related
- 1986-09-26 US US06/912,776 patent/US4774245A/en not_active Expired - Fee Related
- 1986-10-01 DE DE8686307542T patent/DE3667665D1/de not_active Expired - Lifetime
- 1986-10-01 CA CA000519556A patent/CA1293723C/en not_active Expired - Lifetime
- 1986-10-01 ES ES86307542T patent/ES2014234B3/es not_active Expired - Lifetime
- 1986-10-01 EP EP86307543A patent/EP0220845A1/en not_active Withdrawn
- 1986-10-01 AT AT86307542T patent/ATE48844T1/de not_active IP Right Cessation
- 1986-10-01 EP EP86307542A patent/EP0225013B1/en not_active Expired
- 1986-10-01 CA CA000519557A patent/CA1275411C/en not_active Expired - Lifetime
- 1986-10-13 NO NO864062A patent/NO163776C/no unknown
- 1986-10-13 FI FI864124A patent/FI864124A7/fi not_active IP Right Cessation
- 1986-10-13 FI FI864125A patent/FI82050C/fi not_active IP Right Cessation
- 1986-10-13 NO NO864061A patent/NO864061L/no unknown
- 1986-10-15 IL IL80319A patent/IL80319A/xx not_active IP Right Cessation
- 1986-10-16 IE IE273386A patent/IE59642B1/en not_active IP Right Cessation
- 1986-10-16 PH PH34375A patent/PH22556A/en unknown
- 1986-10-16 NZ NZ217957A patent/NZ217957A/xx unknown
- 1986-10-16 NZ NZ217958A patent/NZ217958A/xx unknown
- 1986-10-17 JP JP61247306A patent/JPS62155278A/ja active Pending
- 1986-10-17 JP JP61247307A patent/JPH0753731B2/ja not_active Expired - Lifetime
- 1986-10-17 KR KR1019860008728A patent/KR940010034B1/ko not_active Expired - Fee Related
- 1986-10-17 AU AU64178/86A patent/AU6417886A/en not_active Abandoned
- 1986-10-17 PT PT83571A patent/PT83571B/pt unknown
- 1986-10-17 AU AU64179/86A patent/AU591937B2/en not_active Ceased
- 1986-10-17 PT PT83572A patent/PT83572B/pt not_active IP Right Cessation
-
1987
- 1987-10-13 US US07/108,272 patent/US4795749A/en not_active Expired - Fee Related
-
1989
- 1989-02-02 US US07/305,969 patent/US4886797A/en not_active Expired - Fee Related
- 1989-02-02 US US07/305,970 patent/US4880799A/en not_active Expired - Fee Related
-
1990
- 1990-03-01 GR GR90400114T patent/GR3000367T3/el unknown
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| AHS | Application shelved for other reasons than non-payment | ||
| AHS | Application shelved for other reasons than non-payment |