DK284085A - ISOXAZOLOQUINOLINON DERIVATIVES, THEIR PREPARATION AND USE - Google Patents
ISOXAZOLOQUINOLINON DERIVATIVES, THEIR PREPARATION AND USE Download PDFInfo
- Publication number
- DK284085A DK284085A DK284085A DK284085A DK284085A DK 284085 A DK284085 A DK 284085A DK 284085 A DK284085 A DK 284085A DK 284085 A DK284085 A DK 284085A DK 284085 A DK284085 A DK 284085A
- Authority
- DK
- Denmark
- Prior art keywords
- carbon atoms
- radical containing
- alkyl radical
- derivatives
- isoxazoloquinolinon
- Prior art date
Links
- IXQREGLIGLUSKL-UHFFFAOYSA-N 1H-[1,2]oxazolo[3,4-h]quinolin-2-one Chemical class C1=CC2=NOC=C2C2=C1C=CC(=O)N2 IXQREGLIGLUSKL-UHFFFAOYSA-N 0.000 title abstract 2
- -1 alkyl radical Chemical class 0.000 abstract 6
- 125000004432 carbon atom Chemical group C* 0.000 abstract 6
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- KZBUYRJDOAKODT-UHFFFAOYSA-N Chlorine Chemical group ClCl KZBUYRJDOAKODT-UHFFFAOYSA-N 0.000 abstract 1
- WZKSXHQDXQKIQJ-UHFFFAOYSA-N F[C](F)F Chemical compound F[C](F)F WZKSXHQDXQKIQJ-UHFFFAOYSA-N 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Chemical group 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Lubricants (AREA)
- Color Television Systems (AREA)
- Diaphragms For Electromechanical Transducers (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
1. Derivatives of isoxazoloquinolinone characterized in that they answer to the general formula l see diagramm : EP0168309,P8,F1 in which R represents a hydrogen, fluorine, chlorine or bromine atom, a linear alkyl radical containing from 1 to 5 carbon atoms, or branched alkyl radical containing from 3 to 5 carbon atoms, an alkoxy radical containing from 1 to 5 carbon atoms, a nitro or trifluoromethyl radical and R1 represents a phenyl radical possibly substituted by a linear alkyl radical containing from 1 to 5 carbon atoms, or a branched alkyl radical containing from 3 to 5 carbon atoms, by an alkoxy radical containing from 1 to 5 carbon atoms, or by a halogen atom.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8409961A FR2566407B1 (en) | 1984-06-25 | 1984-06-25 | NOVEL ISOXAZOLOQUINOLEIN DERIVATIVES, PROCESS FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS, AND COMPOSITIONS CONTAINING THEM |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK284085D0 DK284085D0 (en) | 1985-06-24 |
| DK284085A true DK284085A (en) | 1985-12-26 |
Family
ID=9305387
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK284085A DK284085A (en) | 1984-06-25 | 1985-06-24 | ISOXAZOLOQUINOLINON DERIVATIVES, THEIR PREPARATION AND USE |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0168309B1 (en) |
| JP (1) | JPS6176491A (en) |
| KR (1) | KR860000296A (en) |
| AT (1) | ATE32899T1 (en) |
| CA (1) | CA1225993A (en) |
| DE (1) | DE3561818D1 (en) |
| DK (1) | DK284085A (en) |
| ES (1) | ES8604599A1 (en) |
| FI (1) | FI79322C (en) |
| FR (1) | FR2566407B1 (en) |
| GR (1) | GR851530B (en) |
| HU (1) | HU192234B (en) |
| IL (1) | IL75562A (en) |
| MA (1) | MA20461A1 (en) |
| NZ (1) | NZ212532A (en) |
| OA (1) | OA08045A (en) |
| PT (1) | PT80690B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4920117A (en) * | 1989-06-09 | 1990-04-24 | Hoechst-Roussel Pharmaceuticals Inc. | 4,5,5a,6-tetrahydro-3H-isoxazolo(5,4,3-kl)acridines, pharmaceutical compositions and use |
| US5182290A (en) * | 1991-08-27 | 1993-01-26 | Neurogen Corporation | Certain oxazoloquinolinones; a new class of GABA brain receptor ligands |
| JP2000514048A (en) | 1996-06-20 | 2000-10-24 | ボード オブ リージェンツ，ザ ユニバーシティ オブ テキサス システム | Compounds and methods for providing pharmacologically active preparations and uses thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2537140B1 (en) * | 1982-12-07 | 1986-07-18 | Roussel Uclaf | NOVEL 4-HYDROXY-3-QUINOLEINE CARBOXAMIDE DERIVATIVES, SALTS THEREOF, PROCESS FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS, AND COMPOSITIONS CONTAINING THEM |
-
1984
- 1984-06-25 FR FR8409961A patent/FR2566407B1/en not_active Expired
-
1985
- 1985-06-05 FI FI852249A patent/FI79322C/en not_active IP Right Cessation
- 1985-06-19 IL IL75562A patent/IL75562A/en unknown
- 1985-06-20 DE DE8585401234T patent/DE3561818D1/en not_active Expired
- 1985-06-20 EP EP85401234A patent/EP0168309B1/en not_active Expired
- 1985-06-20 AT AT85401234T patent/ATE32899T1/en active
- 1985-06-21 CA CA000484819A patent/CA1225993A/en not_active Expired
- 1985-06-24 MA MA20688A patent/MA20461A1/en unknown
- 1985-06-24 GR GR851530A patent/GR851530B/el unknown
- 1985-06-24 HU HU852472A patent/HU192234B/en not_active IP Right Cessation
- 1985-06-24 JP JP60136225A patent/JPS6176491A/en active Pending
- 1985-06-24 ES ES544488A patent/ES8604599A1/en not_active Expired
- 1985-06-24 PT PT80690A patent/PT80690B/en not_active IP Right Cessation
- 1985-06-24 NZ NZ212532A patent/NZ212532A/en unknown
- 1985-06-24 DK DK284085A patent/DK284085A/en not_active Application Discontinuation
- 1985-06-25 OA OA58619A patent/OA08045A/en unknown
- 1985-06-25 KR KR1019850004504A patent/KR860000296A/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| IL75562A (en) | 1988-07-31 |
| DK284085D0 (en) | 1985-06-24 |
| PT80690B (en) | 1987-03-31 |
| ATE32899T1 (en) | 1988-03-15 |
| FR2566407B1 (en) | 1986-09-26 |
| JPS6176491A (en) | 1986-04-18 |
| IL75562A0 (en) | 1985-10-31 |
| FI79322B (en) | 1989-08-31 |
| EP0168309A1 (en) | 1986-01-15 |
| FI852249A0 (en) | 1985-06-05 |
| PT80690A (en) | 1985-07-01 |
| EP0168309B1 (en) | 1988-03-09 |
| HUT38948A (en) | 1986-07-28 |
| HU192234B (en) | 1987-05-28 |
| KR860000296A (en) | 1986-01-27 |
| OA08045A (en) | 1987-01-31 |
| NZ212532A (en) | 1988-08-30 |
| MA20461A1 (en) | 1985-12-31 |
| ES544488A0 (en) | 1986-02-01 |
| GR851530B (en) | 1985-11-25 |
| DE3561818D1 (en) | 1988-04-14 |
| FR2566407A1 (en) | 1985-12-27 |
| FI852249L (en) | 1985-12-26 |
| ES8604599A1 (en) | 1986-02-01 |
| FI79322C (en) | 1989-12-11 |
| CA1225993A (en) | 1987-08-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |